Novel Bisaryl Substituted Thiazoles and Oxazoles as Highly Potent and Selective Peroxisome Proliferator-Activated Receptor δ Agonists
Epple, Robert, Cow, Christopher, Xie, Yongping, Azimioara, Mihai, Russo, Ross, Wang, Xing, Wityak, John, Karanewsky, Donald S, Tuntland, Tove, Nguyêñ-Trân, Vân T. B, Cuc Ngo, Cara, Huang, David, Saez, Enrique, Spalding, Tracy, Gerken, Andrea, Iskandar, Maya, Seidel, H. Martin, Tian, Shin-Shay
Published in Journal of medicinal chemistry (14.01.2010)
Published in Journal of medicinal chemistry (14.01.2010)
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Journal Article
1,3,5-Trisubstituted aryls as highly selective PPARδ agonists
Epple, Robert, Azimioara, Mihai, Russo, Ross, Bursulaya, Badry, Tian, Shin-Shay, Gerken, Andrea, Iskandar, Maya
Published in Bioorganic & medicinal chemistry letters (01.06.2006)
Published in Bioorganic & medicinal chemistry letters (01.06.2006)
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Journal Article
3,4,5-Trisubstituted isoxazoles as novel PPARδ agonists: Part 1
Epple, Robert, Russo, Ross, Azimioara, Mihai, Cow, Christopher, Xie, Yongping, Wang, Xing, Wityak, John, Karanewsky, Don, Gerken, Andrea, Iskandar, Maya, Saez, Enrique, Martin Seidel, H., Tian, Shin-Shay
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
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Journal Article
3,4,5-Trisubstituted isoxazoles as novel PPARδ agonists. Part 2
Epple, Robert, Azimioara, Mihai, Russo, Ross, Xie, Yongping, Wang, Xing, Cow, Christopher, Wityak, John, Karanewsky, Don, Bursulaya, Badry, Kreusch, Andreas, Tuntland, Tove, Gerken, Andrea, Iskandar, Maya, Saez, Enrique, Martin Seidel, H., Tian, Shin-Shay
Published in Bioorganic & medicinal chemistry letters (01.11.2006)
Published in Bioorganic & medicinal chemistry letters (01.11.2006)
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Journal Article
Synthesis and SAR of succinamide peptidomimetic inhibitors of cathepsin S
Chatterjee, Arnab K., Liu, Hong, Tully, David C., Guo, Jianhua, Epple, Robert, Russo, Ross, Williams, Jennifer, Roberts, Michael, Tuntland, Tove, Chang, Jonathan, Gordon, Perry, Hollenbeck, Thomas, Tumanut, Christine, Li, Jun, Harris, Jennifer L.
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
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Journal Article
1,3,5-Trisubstituted aryls as highly selective PPARdelta agonists
Epple, Robert, Azimioara, Mihai, Russo, Ross, Bursulaya, Badry, Tian, Shin-Shay, Gerken, Andrea, Iskandar, Maya
Published in Bioorganic & medicinal chemistry letters (01.06.2006)
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Published in Bioorganic & medicinal chemistry letters (01.06.2006)
Journal Article
Bicyclic carbamates as inhibitors of papain-like cathepsin proteases
Epple, Robert, Urbina, Hugo D., Russo, Ross, Liu, Hong, Mason, Daniel, Bursulaya, Badry, Tumanut, Christine, Li, Jun, Harris, Jennifer L.
Published in Bioorganic & medicinal chemistry letters (01.03.2007)
Published in Bioorganic & medicinal chemistry letters (01.03.2007)
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Journal Article
Design and synthesis of arylaminoethyl amides as noncovalent inhibitors of cathepsin S. Part 1
Liu, Hong, Tully, David C., Epple, Robert, Bursulaya, Badry, Li, Jun, Harris, Jennifer L., Williams, Jennifer A., Russo, Ross, Tumanut, Christine, Roberts, Michael J., Alper, Phil B., He, Yun, Karanewsky, Donald S.
Published in Bioorganic & medicinal chemistry letters (15.11.2005)
Published in Bioorganic & medicinal chemistry letters (15.11.2005)
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Journal Article
COMPOUNDS AND METHODS FOR MODULATING G PROTEIN-COUPLED RECEPTORS
EPPLE ROBERT, LELAIS GERALD, AZIMIOARA MIHAI, COW CHRISTOPHER, RUSSO ROSS, NIKULIN VICTOR
Year of Publication 02.11.2009
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Year of Publication 02.11.2009
Patent
3,4,5-Trisubstituted isoxazoles as novel PPARdelta agonists: Part 1
Epple, Robert, Russo, Ross, Azimioara, Mihai, Cow, Christopher, Xie, Yongping, Wang, Xing, Wityak, John, Karanewsky, Don, Gerken, Andrea, Iskandar, Maya, Saez, Enrique, Martin Seidel, H, Tian, Shin-Shay
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
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Published in Bioorganic & medicinal chemistry letters (15.08.2006)
Journal Article
3,4,5-Trisubstituted isoxazoles as novel PPARdelta agonists. Part 2
Epple, Robert, Azimioara, Mihai, Russo, Ross, Xie, Yongping, Wang, Xing, Cow, Christopher, Wityak, John, Karanewsky, Don, Bursulaya, Badry, Kreusch, Andreas, Tuntland, Tove, Gerken, Andrea, Iskandar, Maya, Saez, Enrique, Martin Seidel, H, Tian, Shin-Shay
Published in Bioorganic & medicinal chemistry letters (01.11.2006)
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Published in Bioorganic & medicinal chemistry letters (01.11.2006)
Journal Article