Recent advances in small molecule stimulation of regeneration and repair
Silpa, Laurence, Sim, Rachel, Russell, Angela J.
Published in Bioorganic & medicinal chemistry letters (01.04.2022)
Published in Bioorganic & medicinal chemistry letters (01.04.2022)
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Journal Article
Modified minimal-size fragments of heparan sulfate as inhibitors of endosulfatase-2 (Sulf-2)
Kennett, Alice, Epple, Sven, van der Valk, Gabriella, Georgiou, Irene, Gout, Evelyne, Vives, Romain R., Russell, Angela J.
Published in Chemical communications (Cambridge, England) (04.01.2024)
Published in Chemical communications (Cambridge, England) (04.01.2024)
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Journal Article
Biased agonists of GPR84 and insights into biological control
Luscombe, Vincent B., Wang, Pinqi, Russell, Angela J., Greaves, David R.
Published in British journal of pharmacology (01.05.2024)
Published in British journal of pharmacology (01.05.2024)
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Journal Article
Structure-based development of new RAS-effector inhibitors from a combination of active and inactive RAS-binding compounds
Cruz-Migoni, Abimael, Canning, Peter, Quevedo, Camilo E., Bataille, Carole J. R., Bery, Nicolas, Miller, Ami, Russell, Angela J., Phillips, Simon E. V., Carr, Stephen B., Rabbitts, Terence H.
Published in Proceedings of the National Academy of Sciences - PNAS (12.02.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (12.02.2019)
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Journal Article
Small molecule inhibitors of RAS-effector protein interactions derived using an intracellular antibody fragment
Quevedo, Camilo E, Cruz-Migoni, Abimael, Bery, Nicolas, Miller, Ami, Tanaka, Tomoyuki, Petch, Donna, Bataille, Carole J R, Lee, Lydia Y W, Fallon, Phillip S, Tulmin, Hanna, Ehebauer, Matthias T, Fernandez-Fuentes, Narcis, Russell, Angela J, Carr, Stephen B, Phillips, Simon E V, Rabbitts, Terence H
Published in Nature communications (09.08.2018)
Published in Nature communications (09.08.2018)
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Journal Article
Correction: Modified minimal-size fragments of heparan sulfate as inhibitors of endosulfatase-2 (Sulf-2)
Kennett, Alice, Epple, Sven, van der Valk, Gabriella, Georgiou, Irene, Gout, Evelyne, Vivès, Romain R, Russell, Angela J
Published in Chemical communications (Cambridge, England) (23.04.2024)
Published in Chemical communications (Cambridge, England) (23.04.2024)
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Journal Article
Combining experimental strategies for successful target deconvolution
Wilkinson, Isabel V.L., Terstappen, Georg C., Russell, Angela J.
Published in Drug discovery today (01.11.2020)
Published in Drug discovery today (01.11.2020)
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Journal Article
Augmentation of Creatine in the Heart
Zervou, Sevasti, Whittington, Hannah J, Russell, Angela J, Lygate, Craig A
Published in Mini reviews in medicinal chemistry (01.01.2016)
Published in Mini reviews in medicinal chemistry (01.01.2016)
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Journal Article
Activation of the Immune-Metabolic Receptor GPR84 Enhances Inflammation and Phagocytosis in Macrophages
Recio, Carlota, Lucy, Daniel, Purvis, Gareth S D, Iveson, Poppy, Zeboudj, Lynda, Iqbal, Asif J, Lin, Daniel, O'Callaghan, Chris, Davison, Lucy, Griesbach, Esther, Russell, Angela J, Wynne, Graham M, Dib, Lea, Monaco, Claudia, Greaves, David R
Published in Frontiers in immunology (20.06.2018)
Published in Frontiers in immunology (20.06.2018)
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Journal Article
From arylamine N-acetyltransferase to folate-dependent acetyl CoA hydrolase: impact of folic acid on the activity of (HUMAN)NAT1 and its homologue (MOUSE)NAT2
Laurieri, Nicola, Dairou, Julien, Egleton, James E, Stanley, Lesley A, Russell, Angela J, Dupret, Jean-Marie, Sim, Edith, Rodrigues-Lima, Fernando
Published in PloS one (13.05.2014)
Published in PloS one (13.05.2014)
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Journal Article
20 Years an Orphan: Is GPR84 a Plausible Medium-Chain Fatty Acid-Sensing Receptor?
Luscombe, Vincent B, Lucy, Daniel, Bataille, Carole J R, Russell, Angela J, Greaves, David R
Published in DNA and cell biology (01.11.2020)
Published in DNA and cell biology (01.11.2020)
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Journal Article
DLL4-Notch Signaling Mediates Tumor Resistance to Anti-VEGF Therapy In Vivo
LI, Ji-Liang, SAINSON, Richard C. A, WU, Herren, CHOWDHURY, Partha S, RUSSELL, Angela J, MONTGOMERY, Craig P, POULSOM, Richard, HARRIS, Adrian L, EIN OON, Chern, TURLEY, Helen, LEEK, Russell, SHELDON, Helen, BRIDGES, Esther, SHI, Wen, SNELL, Cameron, BOWDEN, Emma T
Published in Cancer research (Chicago, Ill.) (15.09.2011)
Published in Cancer research (Chicago, Ill.) (15.09.2011)
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Journal Article
Kinetic insights into agonist-dependent signalling bias at the pro-inflammatory G-protein coupled receptor GPR84
Luscombe, Vincent B, Baena-López, Luis Alberto, Bataille, Carole J R, Russell, Angela J, Greaves, David R
Published in European journal of pharmacology (05.10.2023)
Published in European journal of pharmacology (05.10.2023)
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Journal Article
Development of Highly Potent, G‑Protein Pathway Biased, Selective, and Orally Bioavailable GPR84 Agonists
Wang, Pinqi, Raja, Arun, Luscombe, Vincent B., Bataille, Carole J. R., Lucy, Daniel, Rogga, Vanessa V., Greaves, David R., Russell, Angela J.
Published in Journal of medicinal chemistry (11.01.2024)
Published in Journal of medicinal chemistry (11.01.2024)
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Journal Article
Increasing Diversity in Admissions to Postgraduate Study
Conway, Stuart J, Kawamura, Akane, Marr, Tracey M, Platt, Frances, Russell, Angela J
Published in Journal of medicinal chemistry (28.04.2022)
Published in Journal of medicinal chemistry (28.04.2022)
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Journal Article
Optimization of 3,5-Dimethylisoxazole Derivatives as Potent Bromodomain Ligands
Hewings, David S, Fedorov, Oleg, Filippakopoulos, Panagis, Martin, Sarah, Picaud, Sarah, Tumber, Anthony, Wells, Christopher, Olcina, Monica M, Freeman, Katherine, Gill, Andrew, Ritchie, Alison J, Sheppard, David W, Russell, Angela J, Hammond, Ester M, Knapp, Stefan, Brennan, Paul E, Conway, Stuart J
Published in Journal of medicinal chemistry (25.04.2013)
Published in Journal of medicinal chemistry (25.04.2013)
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Journal Article
Chemical Proteomics and Phenotypic Profiling Identifies the Aryl Hydrocarbon Receptor as a Molecular Target of the Utrophin Modulator Ezutromid
Wilkinson, Isabel V. L., Perkins, Kelly J., Dugdale, Hannah, Moir, Lee, Vuorinen, Aini, Chatzopoulou, Maria, Squire, Sarah E., Monecke, Sebastian, Lomow, Alexander, Geese, Marcus, Charles, Philip D., Burch, Peter, Tinsley, Jonathan M., Wynne, Graham M., Davies, Stephen G., Wilson, Francis X., Rastinejad, Fraydoon, Mohammed, Shabaz, Davies, Kay E., Russell, Angela J.
Published in Angewandte Chemie International Edition (03.02.2020)
Published in Angewandte Chemie International Edition (03.02.2020)
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Journal Article
Disrupting Hypoxia-Induced Bicarbonate Transport Acidifies Tumor Cells and Suppresses Tumor Growth
McIntyre, Alan, Hulikova, Alzbeta, Ledaki, Ioanna, Snell, Cameron, Singleton, Dean, Steers, Graham, Seden, Peter, Jones, Dylan, Bridges, Esther, Wigfield, Simon, Li, Ji-Liang, Russell, Angela, Swietach, Pawel, Harris, Adrian L
Published in Cancer research (Chicago, Ill.) (01.07.2016)
Published in Cancer research (Chicago, Ill.) (01.07.2016)
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