Sigma-1 receptors control neuropathic pain and macrophage infiltration into the dorsal root ganglion after peripheral nerve injury
Bravo-Caparrós, Inmaculada, Ruiz-Cantero, M Carmen, Perazzoli, Gloria, Cronin, Shane J F, Vela, José M, Hamed, Mohamed F, Penninger, Josef M, Baeyens, José M, Cobos, Enrique J, Nieto, Francisco R
Published in The FASEB journal (01.04.2020)
Published in The FASEB journal (01.04.2020)
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Journal Article
Sigma-1 receptor: A drug target for the modulation of neuroimmune and neuroglial interactions during chronic pain
Ruiz-Cantero, M. Carmen, González-Cano, Rafael, Tejada, Miguel Á., Santos-Caballero, Miriam, Perazzoli, Gloria, Nieto, Francisco R., Cobos, Enrique J.
Published in Pharmacological research (01.01.2021)
Published in Pharmacological research (01.01.2021)
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Journal Article
The sigma‐1 receptor curtails endogenous opioid analgesia during sensitization of TRPV1 nociceptors
Ruiz‐Cantero, M. Carmen, Cortés‐Montero, Elsa, Jain, Aakanksha, Montilla‐García, Ángeles, Bravo‐Caparrós, Inmaculada, Shim, Jaehoon, Sánchez‐Blázquez, Pilar, Woolf, Clifford J., Baeyens, José M., Cobos, Enrique J.
Published in British journal of pharmacology (01.04.2023)
Published in British journal of pharmacology (01.04.2023)
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Journal Article
Modulation by Sigma-1 Receptor of Morphine Analgesia and Tolerance: Nociceptive Pain, Tactile Allodynia and Grip Strength Deficits During Joint Inflammation
Montilla-García, Ángeles, Tejada, Miguel Á, Ruiz-Cantero, M Carmen, Bravo-Caparrós, Inmaculada, Yeste, Sandra, Zamanillo, Daniel, Cobos, Enrique J
Published in Frontiers in pharmacology (22.02.2019)
Published in Frontiers in pharmacology (22.02.2019)
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Journal Article
Tetrodotoxin, a Potential Drug for Neuropathic and Cancer Pain Relief?
González-Cano, Rafael, Ruiz-Cantero, M Carmen, Santos-Caballero, Miriam, Gómez-Navas, Carlos, Tejada, Miguel Á, Nieto, Francisco R
Published in Toxins (12.07.2021)
Published in Toxins (12.07.2021)
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Journal Article
Sigma-1 receptor agonism exacerbates immune-driven nociception: Role of TRPV1 + nociceptors
Ruiz-Cantero, M. Carmen, Huerta, Miguel Á., Tejada, Miguel Á., Santos-Caballero, Miriam, Fernández-Segura, Eduardo, Cañizares, Francisco J., Entrena, José M., Baeyens, José M., Cobos, Enrique J.
Published in Biomedicine & pharmacotherapy (01.11.2023)
Published in Biomedicine & pharmacotherapy (01.11.2023)
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Targeting immune-driven opioid analgesia by sigma-1 receptors: Opening the door to novel perspectives for the analgesic use of sigma-1 antagonists
Tejada, Miguel Á., Montilla-García, Ángeles, González-Cano, Rafael, Bravo-Caparrós, Inmaculada, Ruiz-Cantero, M. Carmen, Nieto, Francisco R., Cobos, Enrique J.
Published in Pharmacological research (01.05.2018)
Published in Pharmacological research (01.05.2018)
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Journal Article
The search for translational pain outcomes to refine analgesic development: Where did we come from and where are we going?
González-Cano, Rafael, Montilla-García, Ángeles, Ruiz-Cantero, M. Carmen, Bravo-Caparrós, Inmaculada, Tejada, Miguel Á., Nieto, Francisco R., Cobos, Enrique J.
Published in Neuroscience and biobehavioral reviews (01.06.2020)
Published in Neuroscience and biobehavioral reviews (01.06.2020)
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Journal Article
Nociceptor-immune interactomes reveal insult-specific immune signatures of pain
Jain, Aakanksha, Gyori, Benjamin M, Hakim, Sara, Jain, Ashish, Sun, Liang, Petrova, Veselina, Bhuiyan, Shamsuddin A, Zhen, Shannon, Wang, Qing, Kawaguchi, Riki, Bunga, Samuel, Taub, Daniel G, Ruiz-Cantero, M Carmen, Tong-Li, Candace, Andrews, Nicholas, Kotoda, Masakazu, Renthal, William, Sorger, Peter K, Woolf, Clifford J
Published in Nature immunology (01.07.2024)
Published in Nature immunology (01.07.2024)
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Journal Article
Discovery of AD258 as a Sigma Receptor Ligand with Potent Antiallodynic Activity
Dichiara, Maria, Ambrosio, Francesca Alessandra, Lee, Sang Min, Ruiz-Cantero, M. Carmen, Lombino, Jessica, Coricello, Adriana, Costa, Giosuè, Shah, Dhara, Costanzo, Giuliana, Pasquinucci, Lorella, Son, Kyung No, Cosentino, Giuseppe, González-Cano, Rafael, Marrazzo, Agostino, Aakalu, Vinay Kumar, Cobos, Enrique J., Alcaro, Stefano, Amata, Emanuele
Published in Journal of medicinal chemistry (24.08.2023)
Published in Journal of medicinal chemistry (24.08.2023)
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Journal Article
Dual Piperidine-Based Histamine H-3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain
Szczepanska, Katarzyna, Karcz, Tadeusz, Dichiara, Maria, Mogilski, Szczepan, Kalinowska-Tluscik, Justyna, Pilarski, Boguslaw, Leniak, Arkadiusz, Pietrus, Wojciech, Podlewska, Sabina, Popiolek-Barczyk, Katarzyna, Humphrys, Laura J., Ruiz-Cantero, M. Carmen, Reiner-Link, David, Leitzbach, Luisa, Lazewska, Dorota, Pockes, Steffen, Gorka, Michal, Zmyslowski, Adam, Calmels, Thierry, Cobos, Enrique J., Marrazzo, Agostino, Stark, Holger, Bojarski, Andrzej J., Amata, Emanuele, Kiec-Kononowicz, Katarzyna
Published in Journal of medicinal chemistry (27.07.2023)
Published in Journal of medicinal chemistry (27.07.2023)
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Journal Article
Dual Piperidine-Based Histamine H3 and Sigma‑1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain
Szczepańska, Katarzyna, Karcz, Tadeusz, Dichiara, Maria, Mogilski, Szczepan, Kalinowska-Tłuścik, Justyna, Pilarski, Bogusław, Leniak, Arkadiusz, Pietruś, Wojciech, Podlewska, Sabina, Popiołek-Barczyk, Katarzyna, Humphrys, Laura J., Ruiz-Cantero, M. Carmen, Reiner-Link, David, Leitzbach, Luisa, Łażewska, Dorota, Pockes, Steffen, Górka, Michał, Zmysłowski, Adam, Calmels, Thierry, Cobos, Enrique J., Marrazzo, Agostino, Stark, Holger, Bojarski, Andrzej J., Amata, Emanuele, Kieć-Kononowicz, Katarzyna
Published in Journal of medicinal chemistry (27.07.2023)
Published in Journal of medicinal chemistry (27.07.2023)
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Journal Article
Sigma-1 Receptors Control Neuropathic Pain and Peripheral Neuroinflammation After Nerve Injury in Female Mice: A Transcriptomic Study
Ruiz-Cantero, M. Carmen, Entrena, José M., Artacho-Cordón, Antonia, Huerta, Miguel Á., Portillo-Salido, Enrique, Nieto, Francisco R., Baeyens, José M., Costigan, Michael, González-Cano, Rafael, Cobos, Enrique J.
Published in Journal of neuroimmune pharmacology (20.08.2024)
Published in Journal of neuroimmune pharmacology (20.08.2024)
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Journal Article
Calmodulin Supports TRPA1 Channel Association with Opioid Receptors and Glutamate NMDA Receptors in the Nervous Tissue
Cortés-Montero, Elsa, Rodríguez-Muñoz, María, Ruiz-Cantero, María Del Carmen, Cobos, Enrique José, Sánchez-Blázquez, Pilar, Garzón-Niño, Javier
Published in International journal of molecular sciences (28.12.2020)
Published in International journal of molecular sciences (28.12.2020)
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Journal Article
Sigma-1 receptors control immune-driven peripheral opioid analgesia during inflammation in mice
Tejada, Miguel A., Montilla-García, Angeles, Cronin, Shane J., Cikes, Domagoj, Sánchez-Fernández, Cristina, González-Cano, Rafael, Ruiz-Cantero, M. Carmen, Penninger, Josef M., Vela, José M., Baeyens, José M., Cobos, Enrique J.
Published in Proceedings of the National Academy of Sciences - PNAS (01.08.2017)
Published in Proceedings of the National Academy of Sciences - PNAS (01.08.2017)
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Journal Article
Novel N‑Substituted Benzomorphan-Based Compounds: From MOR-Agonist/DOR-Antagonist to Biased/Unbiased MOR Agonists
Pasquinucci, Lorella, Parenti, Carmela, Ruiz-Cantero, M. Carmen, Georgoussi, Zafiroula, Pallaki, Paschalina, Cobos, Enrique J, Amata, Emanuele, Marrazzo, Agostino, Prezzavento, Orazio, Arena, Emanuela, Dichiara, Maria, Salerno, Loredana, Turnaturi, Rita
Published in ACS medicinal chemistry letters (14.05.2020)
Published in ACS medicinal chemistry letters (14.05.2020)
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