Risk Attitudes in Late Adulthood: Do Parenthood Status and Family Size Matter?
Ho, Christine, Teerawichitchainan, Bussarawan, Tan, Joanne, Lie Tan, Eugene Rui
Published in Research on aging (01.05.2023)
Published in Research on aging (01.05.2023)
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Design, Synthesis, and Evaluation of NO-Donor Containing Carbonic Anhydrase Inhibitors To Lower Intraocular Pressure
Huang, Qinhua, Rui, Eugene Y, Cobbs, Morena, Dinh, Dac M, Gukasyan, Hovhannes J, Lafontaine, Jennifer A, Mehta, Saurabh, Patterson, Brian D, Rewolinski, David A, Richardson, Paul F, Edwards, Martin P
Published in Journal of medicinal chemistry (26.03.2015)
Published in Journal of medicinal chemistry (26.03.2015)
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Journal Article
737 Inhibition of P21-activated kinase 4 (PAK4) reverts immune exclusion and restores anti-tumor immunity in the tumor microenvironment
Zhou, Yu 'Jerry', Chu, Gina, Hendrickson, Eleanore, Gullo-Brown, Johnni, Chavez, Brandy, McAlpine, Indrawan, Rui, Eugene, Doran, Shawn, Timofeevski, Sergei, Heyen, Jonathan, Kinong, Jennifer, Tang, Szu-Yu, Oyer, Jon, Rayannavar, Vinayak, Nager, Andrew, Ching, Keith, Shi, Stephanie, Bhadra, Rajarshi, Dillon, Christopher, Gururajan, Murali
Published in Journal for immunotherapy of cancer (01.11.2021)
Published in Journal for immunotherapy of cancer (01.11.2021)
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Journal Article
Chemoenzymatic synthesis of small molecule human therapeutics
Ran, Ningqing, Rui, Eugene, Liu, Jinhua, Tao, Junhua
Published in Current pharmaceutical design (2009)
Published in Current pharmaceutical design (2009)
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Journal Article
Ocular pharmacokinetics and hypotensive activity of PF-04475270, an EP4 prostaglandin agonist in preclinical models
Prasanna, Ganesh, Fortner, Jay, Xiang, Cathie, Zhang, Eric, Carreiro, Samantha, Anderson, Scott, Sartnurak, Soisurin, Wu, Grace, Gukasyan, Hovhannes, Niesman, Michael, Nair, Sajiv, Rui, Eugene, Lafontaine, Jennifer, Almaden, Chau Doan, Wells, Peter, Krauss, Achim
Published in Experimental eye research (01.11.2009)
Published in Experimental eye research (01.11.2009)
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Journal Article
6-Methylsulfanyl-4H-pyrimido[1,6-a]pyrimidin-4-one
Quinhua Huang, Paul F. Richardson, Eugene Rui, Arnold L. Rheingold, Alex Yanovsky
Published in Acta crystallographica. Section E, Structure reports online (01.10.2009)
Published in Acta crystallographica. Section E, Structure reports online (01.10.2009)
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Journal Article
SAM-Competitive PRMT5 Inhibitor PF-06939999 Demonstrates Antitumor Activity in Splicing Dysregulated NSCLC with Decreased Liability of Drug Resistance
Jensen-Pergakes, Kristen, Tatlock, John, Maegley, Karen A, McAlpine, Indrawan J, McTigue, Michele, Xie, Tao, Dillon, Christopher P, Wang, Yuli, Yamazaki, Shinji, Spiegel, Noah, Shi, Manli, Nemeth, Amy, Miller, Natalie, Hendrickson, Eleanore, Lam, Hieu, Sherrill, John, Chung, Chi-Yeh, McMillan, Elizabeth A, Bryant, Shannon Karlicek, Palde, Prakash, Braganza, John, Brooun, Alexei, Deng, Ya-Li, Goshtasbi, Vesta, Kephart, Susan E, Kumpf, Robert A, Liu, Wei, Patman, Ryan L, Rui, Eugene, Scales, Stephanie, Tran-Dube, Michelle, Wang, Fen, Wythes, Martin, Paul, Thomas A
Published in Molecular cancer therapeutics (01.01.2022)
Published in Molecular cancer therapeutics (01.01.2022)
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Journal Article
Abstract 617: BH-30236, a novel macrocyclic CLK inhibitor modulating RNA splicing, demonstrates potent inhibition of cancer cell growth in a broad panel of cancer cell lines
Jiang, Ping, Li, Danan, Ling, Nancy, Zhai, Dayong, Deng, Wei, Rui, Eugene, Cui, J. Jean
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Journal Article
Design and Synthesis of Pyridone-Containing 3,4-Dihydroisoquinoline-1(2H)‑ones as a Novel Class of Enhancer of Zeste Homolog 2 (EZH2) Inhibitors
Kung, Pei-Pei, Rui, Eugene, Bergqvist, Simon, Bingham, Patrick, Braganza, John, Collins, Michael, Cui, Mei, Diehl, Wade, Dinh, Dac, Fan, Connie, Fantin, Valeria R, Gukasyan, Hovhannes J, Hu, Wenyue, Huang, Buwen, Kephart, Susan, Krivacic, Cody, Kumpf, Robert A, Li, Gary, Maegley, Karen A, McAlpine, Indrawan, Nguyen, Lisa, Ninkovic, Sacha, Ornelas, Martha, Ryskin, Michael, Scales, Stephanie, Sutton, Scott, Tatlock, John, Verhelle, Dominique, Wang, Fen, Wells, Peter, Wythes, Martin, Yamazaki, Shinji, Yip, Brian, Yu, Xiu, Zehnder, Luke, Zhang, Wei-Guo, Rollins, Robert A, Edwards, Martin
Published in Journal of medicinal chemistry (22.09.2016)
Published in Journal of medicinal chemistry (22.09.2016)
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Journal Article
STING Modulators of STING Stimulator of Interferon Genes
JALAIE MEHRAN, WYTHES MARTIN JAMES, GAJIWALA KETAN SATISH, SUN JIANMIN, RUI EUGENE YUANJIN, HUH CHAN WOO, PATMAN RYAN LLOYD
Year of Publication 25.03.2024
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Year of Publication 25.03.2024
Patent
Abstract 5944: Discovery of BH-30236: A novel macrocyclic CLK inhibitor targeting alternative splicing in cancers
Cui, J. Jean, Jiang, Ping, Deng, Wei, Zhai, Dayong, Ling, Nancy, Li, Danan, Wang, Zhenping, Hu, Yue, Darjania, Levan, Whitten, Jeff, Rogers, Evan, Rui, Eugene
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Journal Article
Abstract 1160: SAM competitive PRMT5 inhibitor PF06939999 demonstrates antitumor activity in splicing dysregulated NSCLC with decreased liability of drug resistance
Jensen-Pergakes, Kristen, Tatlock, John, Maegley, Karen, McAlpine, Indrawan, McTigue, Michele, Xie, Tao, Dillon, Christopher, Wang, Yuli, Yamazaki, Shinji, Spiegel, Noah, Shi, Manli, Nemeth, Amy, Miller, Natalie, Hendrickson, Eleanore, Lam, Hieu, Sherrill, John, Liu, Wei, Deng, Ya-Li, Chung, Chi-Yeh, McMillan, Elizabeth A., Palde, Prakash, Brooun, Alexei, Braganza, John, Kephart, Susan E., Kumpf, Robert, Patman, Ryan, Rui, Eugene, Scales, Stephanie, Tran-Dube, Michelle, Wang, Fen, Wythes, Martin, Paul, Thomas
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Journal Article
STING 의 조정제
JALAIE MEHRAN, WYTHES MARTIN JAMES, GAJIWALA KETAN SATISH, SUN JIANMIN, RUI EUGENE YUANJIN, HUH CHAN WOO, PATMAN RYAN LLOYD
Year of Publication 19.10.2023
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Year of Publication 19.10.2023
Patent
Abstract 4857: Discovery of PF-06855800, a SAM competitive PRMT5 inhibitor with potent antitumor activity
Mcalpine, Indrawan J., Tatlock, John, Billitti, Joseph, Braganza, John, Brooun, Alexei, Ya-Li, Deng, Hirakawa, Brad, Jensen-Pergakes, Kristen, Kumpf, Robert, Liu, Wei, Maegley, Karen, McTigue, Michele, Patman, Ryan, Rui, Eugene, Scales, Stephanie, Spiegel, Noah, Tran-Dubé, Michelle, Wang, Fen, Wang, Zhenxiong, Yamazaki, Shinji, Zhang, Tao, Wythes, Martin
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Characterization of the CHK1 Allosteric Inhibitor Binding Site
Vanderpool, Darin, Johnson, Ted O, Ping, Chen, Bergqvist, Simon, Alton, Gordon, Phonephaly, Soneprasith, Rui, Eugene, Luo, Chun, Deng, Ya-Li, Grant, Stephan, Quenzer, Terri, Margosiak, Steve, Register, James, Brown, Ed, Ermolieff, Jacques
Published in Biochemistry (Easton) (20.10.2009)
Published in Biochemistry (Easton) (20.10.2009)
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STING의 사이클로펜탄-기반 조절제
JALAIE MEHRAN, WYTHES MARTIN JAMES, MCALPINE INDRAWAN JAMES, PATMAN RYAN, RUI EUGENE YUANJIN, GAJIWALA KETAN S, FENSOME ANDREW, MADERNA ANDREAS
Year of Publication 24.11.2020
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Year of Publication 24.11.2020
Patent
STING 의 폴리헤테로시클릭 조정제
JALAIE MEHRAN, TRAN TUAN PHONG, WYTHES MARTIN JAMES, FISHER ETHAN LAWRENCE, ZHANG LEI, MCALPINE INDRAWAN JAMES, PATMAN RYAN, ZHOU DAHUI, GAJIWALA KETAN S, RUI EUGENE YUANJIN, FENSOME ANDREW, HUH CHAN WOO
Year of Publication 30.05.2022
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Year of Publication 30.05.2022
Patent