Model-Based Analysis of Biopharmaceutic Experiments To Improve Mechanistic Oral Absorption Modeling: An Integrated in Vitro in Vivo Extrapolation Perspective Using Ketoconazole as a Model Drug
Pathak, Shriram M, Ruff, Aaron, Kostewicz, Edmund S, Patel, Nikunjkumar, Turner, David B, Jamei, Masoud
Published in Molecular pharmaceutics (04.12.2017)
Published in Molecular pharmaceutics (04.12.2017)
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Abstract 1482: M4645 is a potent and highly selective inhibitor of disease relevant cKIT mutations for the treatment of metastatic or recurrent GIST
Linde, Nina, Blum, Andreas, Dorsch, Dieter, Graedler, Ulrich, Busch, Michael, Glaser, Nina, Petersson, Carl, Ruff, Aaron, Sherbetjian, Eva, Esdar, Christina
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Identification of M4205A Highly Selective Inhibitor of KIT Mutations for Treatment of Unresectable Metastatic or Recurrent Gastrointestinal Stromal Tumors
Blum, Andreas, Dorsch, Dieter, Linde, Nina, Brandstetter, Susanne, Buchstaller, Hans-Peter, Busch, Michael, Glaser, Nina, Grädler, Ulrich, Ruff, Aaron, Petersson, Carl, Schieferstein, Hanno, Sherbetjian, Eva, Esdar, Christina
Published in Journal of medicinal chemistry (23.02.2023)
Published in Journal of medicinal chemistry (23.02.2023)
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Evaluating the predictability of the in vitro transfer model and in vivo rat studies as a surrogate to investigate the supersaturation and precipitation behaviour of different Albendazole formulations for humans
Ruff, Aaron, Holm, René, Kostewicz, Edmund S.
Published in European journal of pharmaceutical sciences (15.07.2017)
Published in European journal of pharmaceutical sciences (15.07.2017)
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Advances and challenges in PBPK modeling – Analysis of factors contributing to the oral absorption of atazanavir, a poorly soluble weak base
Berlin, Mark, Ruff, Aaron, Kesisoglou, Filippos, Xu, Wei, Wang, Michael Hong, Dressman, Jennifer B.
Published in European journal of pharmaceutics and biopharmaceutics (01.06.2015)
Published in European journal of pharmaceutics and biopharmaceutics (01.06.2015)
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A toolbox for the upscaling of ethanolic human serum albumin (HSA) desolvation
Wacker, Matthias, Zensi, Anja, Kufleitner, Jürgen, Ruff, Aaron, Schütz, Jessica, Stockburger, Tobias, Marstaller, Thomas, Vogel, Vitali
Published in International journal of pharmaceutics (29.07.2011)
Published in International journal of pharmaceutics (29.07.2011)
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