Utilization of High-Throughput Experimentation (HTE) and ChemBeads Toward the Development of an Aryl Bromide and Benzyl Bromide Photoredox Cross-Electrophile Coupling
Glogowski, Michal P., Cercizi, Noel, Lynch-Colameta, Tessa, Ridgers, Lance H., Phelan, James P., Rowley, Ann M., Rauch, Martin P.
Published in Organic letters (29.03.2024)
Published in Organic letters (29.03.2024)
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Discovery and SAR Study of Boronic Acid-Based Selective PDE3B Inhibitors from a Novel DNA-Encoded Library
Rowley, Ann M., Yao, Gang, Andrews, Logan, Bedermann, Aaron, Biddulph, Ross, Bingham, Ryan, Brady, Jennifer J., Buxton, Rachel, Cecconie, Ted, Cooper, Rona, Csakai, Adam, Gao, Enoch N., Grenier-Davies, Melissa C., Lawler, Meghan, Lian, Yiqian, Macina, Justyna, Macphee, Colin, Marcaurelle, Lisa, Martin, John, McCormick, Patricia, Pindoria, Rekha, Rauch, Martin, Rocque, Warren, Shen, Yingnian, Shewchuk, Lisa M., Squire, Michael, Stebbeds, Will, Tear, Westley, Wang, Xin, Ward, Paris, Xiao, Shouhua
Published in Journal of medicinal chemistry (08.02.2024)
Published in Journal of medicinal chemistry (08.02.2024)
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Discovery of a Selective Phosphoinositide-3-Kinase (PI3K)‑γ Inhibitor (IPI-549) as an Immuno-Oncology Clinical Candidate
Evans, Catherine A, Liu, Tao, Lescarbeau, André, Nair, Somarajan J, Grenier, Louis, Pradeilles, Johan A, Glenadel, Quentin, Tibbitts, Thomas, Rowley, Ann M, DiNitto, Jonathan P, Brophy, Erin E, O’Hearn, Erin L, Ali, Janid A, Winkler, David G, Goldstein, Stanley I, O’Hearn, Patrick, Martin, Christian M, Hoyt, Jennifer G, Soglia, John R, Cheung, Culver, Pink, Melissa M, Proctor, Jennifer L, Palombella, Vito J, Tremblay, Martin R, Castro, Alfredo C
Published in ACS medicinal chemistry letters (08.09.2016)
Published in ACS medicinal chemistry letters (08.09.2016)
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An Aldol-Based Build/Couple/Pair Strategy for the Synthesis of Medium- and Large-Sized Rings: Discovery of Macrocyclic Histone Deacetylase Inhibitors
Marcaurelle, Lisa A, Comer, Eamon, Dandapani, Sivaraman, Duvall, Jeremy R, Gerard, Baudouin, Kesavan, Sarathy, Lee, Maurice D, Liu, Haibo, Lowe, Jason T, Marie, Jean-Charles, Mulrooney, Carol A, Pandya, Bhaumik A, Rowley, Ann, Ryba, Troy D, Suh, Byung-Chul, Wei, Jingqiang, Young, Damian W, Akella, Lakshmi B, Ross, Nathan T, Zhang, Yan-Ling, Fass, Daniel M, Reis, Surya A, Zhao, Wen-Ning, Haggarty, Stephen J, Palmer, Michelle, Foley, Michael A
Published in Journal of the American Chemical Society (01.12.2010)
Published in Journal of the American Chemical Society (01.12.2010)
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Synthesis and Profiling of a Diverse Collection of Azetidine-Based Scaffolds for the Development of CNS-Focused Lead-like Libraries
Lowe, Jason T, Lee, Maurice D, Akella, Lakshmi B, Davoine, Emeline, Donckele, Etienne J, Durak, Landon, Duvall, Jeremy R, Gerard, Baudouin, Holson, Edward B, Joliton, Adrien, Kesavan, Sarathy, Lemercier, Berenice C, Liu, Haibo, Marié, Jean-Charles, Mulrooney, Carol A, Muncipinto, Giovanni, Welzel-O’Shea, Morgan, Panko, Laura M, Rowley, Ann, Suh, Byung-Chul, Thomas, Meryl, Wagner, Florence F, Wei, Jingqiang, Foley, Michael A, Marcaurelle, Lisa A
Published in Journal of organic chemistry (07.09.2012)
Published in Journal of organic chemistry (07.09.2012)
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Journal Article
Investigating Capnography Innovation for Better Patient Monitoring in the Resource Limited Surgical Setting
Nourian, Maziar M, Kolbay, Patrick, Hoehne, Soeren, Poursaid, Ahrash E, Rowley, Ann E, Harris, Mark J, Kuck, Kai
Published in Surgical innovation (01.02.2019)
Published in Surgical innovation (01.02.2019)
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Journal Article
One-Pot Catalytic Asymmetric Synthesis of Pyranones
Cheng, Kevin, Kelly, Ann Rowley, Kohn, Rachel A, Dweck, Jessica F, Walsh, Patrick J
Published in Organic letters (18.06.2009)
Published in Organic letters (18.06.2009)
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Journal Article
Targeting IRAK3 for Degradation to Enhance IL-12 Pro-inflammatory Cytokine Production
Rowley, Ann, Brown, Brian S., Stofega, Mary, Hoh, Hana, Mathew, Rebecca, Marin, Violeta, Ding, Rong-Xian, McClure, Ryan A., Bittencourt, Fabiola M., Chen, Jun, Gururaja, Tarikere, Kinoshita, Taisei, Wang, Xueqing, Rivkin, Alexey, Woller, Kevin R.
Published in ACS chemical biology (17.06.2022)
Published in ACS chemical biology (17.06.2022)
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Journal Article
Diversity-Oriented Synthesis-Facilitated Medicinal Chemistry: Toward the Development of Novel Antimalarial Agents
Comer, Eamon, Beaudoin, Jennifer A, Kato, Nobutaka, Fitzgerald, Mark E, Heidebrecht, Richard W, Lee, Maurice duPont, Masi, Daniela, Mercier, Marion, Mulrooney, Carol, Muncipinto, Giovanni, Rowley, Ann, Crespo-Llado, Keila, Serrano, Adelfa E, Lukens, Amanda K, Wiegand, Roger C, Wirth, Dyann F, Palmer, Michelle A, Foley, Michael A, Munoz, Benito, Scherer, Christina A, Duvall, Jeremy R, Schreiber, Stuart L
Published in Journal of medicinal chemistry (23.10.2014)
Published in Journal of medicinal chemistry (23.10.2014)
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Journal Article
Accessing Skeletal Diversity Using Catalyst Control: Formation of n and n + 1 Macrocyclic Triazole Rings
Kelly, Ann Rowley, Wei, Jingqiang, Kesavan, Sarathy, Marié, Jean-Charles, Windmon, Nicole, Young, Damian W, Marcaurelle, Lisa A
Published in Organic letters (04.06.2009)
Published in Organic letters (04.06.2009)
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Journal Article
Highly Enantio- and Diastereoselective One-Pot Synthesis of Acyclic Epoxy Alcohols with Three Contiguous Stereocenters
Lurain, Alice E, Maestri, Aaron, Kelly, Ann Rowley, Carroll, Patrick J, Walsh, Patrick J
Published in Journal of the American Chemical Society (27.10.2004)
Published in Journal of the American Chemical Society (27.10.2004)
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Journal Article
Practical asymmetric synthesis of β-hydroxy γ-amino acids via complimentary aldol reactions
Pandya, Bhaumik A., Dandapani, Sivaraman, Duvall, Jeremy R., Rowley, Ann, Mulrooney, Carol A., Ryba, Troy, Dombrowski, Michael, Harton, Marie, Young, Damian W., Marcaurelle, Lisa A.
Published in Tetrahedron (26.08.2011)
Published in Tetrahedron (26.08.2011)
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Journal Article
Tricyclic modulators of TNF signaling
Cox Phil B, Dietrich Justin, Vasudevan Anil, Frank Kristine E, Li Huan-Qui, Breinlinger Eric C, Friedman Michael M, Rowley Ann Marie, Wilson Noel, Longenecker Kenton, Osuma Augustine
Year of Publication 02.01.2018
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Year of Publication 02.01.2018
Patent
TRICYCLIC MODULATORS OF TNF SIGNALING
Dietrich, Justin D, Frank, Kristine E, Cox, Phil B, Vasudevan, Anil, Osuma, Augustine T, Li, Huan-Qui, Longenecker, Kenton L, Wilson, Noel S, Breinlinger, Eric C, Friedman, Michael M, Rowley, Ann Marie
Year of Publication 28.06.2018
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Year of Publication 28.06.2018
Patent
Tricyclic modulators of TNF signaling
Dietrich, Justin D, Frank, Kristine E, Gomtsyan, Arthur, Dombrowski, Amanda W, Schmidt, Robert, Breinlinger, Eric C, Friedman, Michael M, Cox, Phil B, Vasudevan, Anil, Osuma, Augustine T, Daanen, Jerome, Li, Huan-Qui, Longenecker, Kenton L, Wilson, Noel S, Rowley, Ann Marie, Djuric, Stevan
Year of Publication 23.04.2019
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Year of Publication 23.04.2019
Patent
TRICYCLIC MODULATORS OF TNF SIGNALING
OSUMA, Augustine, BREINLINGER, Eric, C, DJURIC, Stevan, DOMBROWSKI, Amanda, W, COX, Phil, B, ROWLEY, Ann, Marie, WILSON, Noel, FRIEDMAN, Michael, M, VASUDEVAN, Anil, DAANEN, Jerome, SCHMIDT, Robert, LI, Huan-Qui, GOMTSYAN, Arthur, LONGENECKER, Kenton, DIETRICH, Justin, FRANK, Kristine, E
Year of Publication 07.03.2018
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Year of Publication 07.03.2018
Patent