Fit-for-Purpose Development of the Enabling Route to Crizotinib (PF-02341066)
de Koning, Pieter D, McAndrew, Douglas, Moore, Robert, Moses, Ian B, Boyles, David C, Kissick, Kyle, Stanchina, Corey L, Cuthbertson, Timothy, Kamatani, Asayuki, Rahman, Leera, Rodriguez, Rick, Urbina, Armando, Sandoval (née Accacia), Alison, Rose, Peter R
Published in Organic process research & development (16.09.2011)
Published in Organic process research & development (16.09.2011)
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Development of a Scalable Synthesis for an Inhaled pan-JAK Inhibitor
Gontcharov, Alexander, Magano, Javier, Samp, Lacey, Houck, Tim L, Rose, Peter R, Rane, Anil, Coe, Jotham W, Kortum, Steven W, Chung, SeungWon, Jones, Peter, Pattavina, David
Published in Organic process research & development (20.09.2019)
Published in Organic process research & development (20.09.2019)
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Evaluation of Kilogram-Scale Sonagashira, Suzuki, and Heck Coupling Routes to Oncology Candidate CP-724,714
Ripin, David H. Brown, Bourassa, Dennis E, Brandt, Thomas, Castaldi, Michael J, Frost, Heather N, Hawkins, Joel, Johnson, Phillip J, Massett, Stephen S, Neumann, Karin, Phillips, James, Raggon, Jeffery W, Rose, Peter R, Rutherford, Jennifer L, Sitter, Barbara, Stewart, A. Morgan, Vetelino, Michael G, Wei, Lulin
Published in Organic process research & development (01.07.2005)
Published in Organic process research & development (01.07.2005)
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Development of a Practical and Efficient Synthesis of CP-945,598-01, a CB1 Antagonist for the Treatment of Obesity
Ragan, John A, Bourassa, Dennis E, Blunt, Jon, Breen, Darragh, Busch, Frank R, Cordi, Eric M, Damon, David B, Do, Nga, Engtrakul, Alanya, Lynch, Denis, McDermott, Ruth E, Mongillo, Joseph A, O’Sullivan, Maria M, Rose, Peter R, Vanderplas, Brian C
Published in Organic process research & development (20.03.2009)
Published in Organic process research & development (20.03.2009)
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Automated and Material-Sparing Workflow for the Measurement of Crystal Nucleation and Growth Kinetics
Arruda, Ryan J., Cally, Paul A.J., Wylie, Anthony, Shah, Nisha, Joel, Ibrahim, Leff, Zachary A., Clark, Alexander, Fountain, Griffin, Neves, Layane, Kratz, Joseph, Thorat, Alpana A., Marziano, Ivan, Rose, Peter R., Girard, Kevin P., Capellades, Gerard
Published in Crystal growth & design (03.05.2023)
Published in Crystal growth & design (03.05.2023)
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Early Process Development of PF-07054894, a Squaramide-Based Antagonist of C–C Chemokine Receptor Type 6 (CCR6)
Chinigo, Gary M., McInturff, Emma L., Bagley, Scott W., Barnhart, Richard W., Blakemore, David C., Han, Lu, Lee, Taegyo, Magano, Javier, McWilliams, J. Christopher, Monfette, Sebastien, Mousseau, James J., Pan, Senliang, Pedro, Dylan, Perfect, Hahdi H., Raggon, Jeffrey W., Rose, Peter R., Sagal, John, Trujillo, John I., Van Haitsma, Jared, Vetelino, Michael G., Yang, Xiaojing Helen
Published in Organic process research & development (21.06.2024)
Published in Organic process research & development (21.06.2024)
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Isolation and identification of an unusual impurity in an intermediate of Rimadyl((R)) (carprofen)
Tucker, JL, DeVries, KM, Hammen, PD, Rose, PR, Raymer, BK, Rescek, D
Published in Heterocycles (01.07.2003)
Published in Heterocycles (01.07.2003)
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Transition-metal chemistry of hexafluorobutadiene. Facile hydrolysis of (hexafluoro-1-metalla-3-cyclopentene)rhodium complexes to give tetrafluoro-1-metalla-3-cyclopenten-2-one and tetrafluoro-1-metalla-2-cyclopenten-4-one complexes. Crystal and molecular structures of trans-[cyclo][(RhCF2CF:CFCO)Cl(PPh3)2], mer-[cyclo][(RhCF2CF:CFCF2)Cl(PMe3)3], and mer-[cyclo][(RhCF:CFCOCF2)Cl(PMe3)3]
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Synthesis and Molecular Structure of the First Example of an .eta.4-Complex of Hexafluorobutadiene: [RuCl(.eta.5-C5Me5)(.eta.4-C4F6)]. Structural Comparison of Coordinated Butadiene and Its Perfluorinated Analog
Hughes, Russell P, Rose, Peter R, Zheng, Xiaoming, Rheingold, Arnold L
Published in Organometallics (01.05.1995)
Published in Organometallics (01.05.1995)
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Development of two synthetic routes to CE-178,253, a CB1 antagonist for the treatment of obesity
Brandt, Thomas A., Caron, Stephane, Damon, David B., DiBrino, Joseph, Ghosh, Arun, Griffith, David A., Kedia, Sandeep, Ragan, John A., Rose, Peter R., Vanderplas, Brian C., Wei, Lulin
Published in Tetrahedron (18.04.2009)
Published in Tetrahedron (18.04.2009)
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Development of two synthetic routes to CE-178,253, a CB1 antagonist for the treatment of obesity: Recent Advances in Synthetic Methodology: Development and Applications
BRANDT, Thomas A, CARON, Stéphane, LULIN WEI, DAMON, David B, DIBRINO, Joseph, GHOSH, Arun, GRIFFITH, David A, KEDIA, Sandeep, RAGAN, John A, ROSE, Peter R, VANDERPLAS, Brian C
Published in Tetrahedron (2009)
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Published in Tetrahedron (2009)
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Development of a Practical and Efficient Synthesis of CP-945,598-01, a CB 1 Antagonist for the Treatment of Obesity
Ragan, John A., Bourassa, Dennis E., Blunt, Jon, Breen, Darragh, Busch, Frank R., Cordi, Eric M., Damon, David B., Do, Nga, Engtrakul, Alanya, Lynch, Denis, McDermott, Ruth E., Mongillo, Joseph A., O’Sullivan, Maria M., Rose, Peter R., Vanderplas, Brian C.
Published in Organic process research & development (20.03.2009)
Published in Organic process research & development (20.03.2009)
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Construction of the (1 alpha,5 alpha,6 alpha)-6-amino-3-azabicyclo[3.1.0]hexane ring system
Braish, TF, Castaldi, M, Chan, S, Fox, DE, Keltonic, T, McGarry, J, Hawkins, JM, Norris, T
Published in Synlett (01.11.1996)
Published in Synlett (01.11.1996)
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Synthesis of trovafloxacin using various (1 alpha,5 alpha,6 alpha)-3-azabicyclo[3.1.0]hexane derivatives
Norris, T, Braish, TF, Butters, M, DeVries, KM, Hawkins, JM, Massett, SS, Rose, PR, Santafianos, D, Sklavounos, C
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2000)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2000)
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