Preclinical Testing of the Nitroimidazopyran PA-824 for Activity against Mycobacterium tuberculosis in a Series of In Vitro and In Vivo Models
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Structure-based design of inhibitors of purine nucleoside phosphorylase. 2. 9-Alicyclic and 9-heteroalicyclic derivatives of 9-deazaguanine
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Synthesis and biological evaluation of trehalose analogs as potential inhibitors of mycobacterial cell wall biosynthesis
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Enhancement of Nucleoside Cytotoxicity through Nucleotide Prodrugs
Rose, Jerry D, Parker, William B, Someya, Hitoshi, Shaddix, Sue C, Montgomery, John A, Secrist, John A
Published in Journal of medicinal chemistry (26.09.2002)
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Structure-based design of inhibitors of purine nucleoside phosphorylase. 3. 9-Arylmethyl derivatives of 9-deazaguanine substituted on the arylmethyl group
Erion, Mark D, Niwas, Shri, Rose, Jerry D, Ananthan, Subramaniam, Allen, Mark, Secrist, John A, Babu, Y. Sudhakar, Bugg, Charles E, Guida, Wayne C
Published in Journal of medicinal chemistry (01.11.1993)
Published in Journal of medicinal chemistry (01.11.1993)
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Structure-based design of inhibitors of purine nucleoside phosphorylase. 1. 9-(Arylmethyl) derivatives of 9-deazaguanine
Montgomery, John A., Niwas, Shri, Rose, Jerry D., Secrist, John A., Babu, Y. Sudhakar, Bugg, Charles E., Erion, Mark D., Guida, Wayne C., Ealick, Steven E.
Published in Journal of medicinal chemistry (1993)
Published in Journal of medicinal chemistry (1993)
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New anticancer agents: synthesis of 1,2-dihydropyrido[3,4-b]pyrazines (1-deaza-7,8-dihydropteridines)
Temple, Carroll, Wheeler, Glynn P, Elliott, Robert D, Rose, Jerry D, Kussner, Conrad L, Comber, Robert N, Montgomery, John A
Published in Journal of medicinal chemistry (01.09.1982)
Published in Journal of medicinal chemistry (01.09.1982)
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Synthesis of potential anticancer agents: imidazo[4,5-c]pyridines and imidazo[4,5-b]pyridines
Temple, Carroll, Rose, Jerry D, Comber, Robert N, Rener, Gregory A
Published in Journal of medicinal chemistry (01.10.1987)
Published in Journal of medicinal chemistry (01.10.1987)
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Structure-based design of inhibitors of purine nucleoside phosphorylase. 3. 9-Arylmethyl derivatives of 9-deazaguanine substituted on the arylmethyl group. [Erratum to document cited in CA119(25):271601v]
Erion, Mark D, Niwas, Shri, Rose, Jerry D, Ananthan, Subramaniam, Allen, Mark, Secrist, John A, Babu, Y. Sudhakar, Bugg, Charles E, Guida, Wayne C
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Published in Journal of medicinal chemistry (01.04.1994)
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Chemical conversion of folic acid to pteroic acid
Temple, Carroll, Rose, Jerry D, Montgomery, John A
Published in Journal of organic chemistry (01.08.1981)
Published in Journal of organic chemistry (01.08.1981)
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1,2-Dihydropyrido[3,4-b]pyrazines: structure-activity relationships
Temple, Carroll, Wheeler, Glynn P, Elliott, Robert D, Rose, Jerry D, Comber, Robert N, Montgomery, John A
Published in Journal of medicinal chemistry (01.01.1983)
Published in Journal of medicinal chemistry (01.01.1983)
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Synthesis of pseudocofactor analogs as potential inhibitors of the folate enzymes
Temple, Carroll, Bennett, L. Lee, Rose, Jerry D, Elliott, Robert D, Montgomery, John H
Published in Journal of medicinal chemistry (01.02.1982)
Published in Journal of medicinal chemistry (01.02.1982)
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Preparation and purification of L-(.+-.)-5-formyl-5,6,7,8-tetrahydrofolic acid
Temple, Carroll, Elliott, Robert D, Rose, Jerry D, Montgomery, John A
Published in Journal of medicinal chemistry (01.06.1979)
Published in Journal of medicinal chemistry (01.06.1979)
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Synthesis of potential antimalarial agents. V. Pyrido[2,3-b]pyrazines
Temple, Carroll, Rose, Jerry D, Elliott, Robert Daryl, Montgomery, John A
Published in Journal of medicinal chemistry (01.09.1970)
Published in Journal of medicinal chemistry (01.09.1970)
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Synthesis of potential antimalarial agents. II. 6,8-Disubstituted pyrido[2,3-b]pyrazines
Temple, Carroll, Rose, Jerry D, Elliott, Robert D, Montgomery, John A
Published in Journal of medicinal chemistry (01.11.1968)
Published in Journal of medicinal chemistry (01.11.1968)
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Structure-based design of inhibitors of purine nucleoside phosphorylase. 3. 9-Arylmethyl derivatives of 9-deazaguanine substituted on the methylene group
Erion, M D, Niwas, S, Rose, J D, Ananthan, S, Allen, M, Secrist, 3rd, J A, Babu, Y S, Bugg, C E, Guida, W C, Ealick, S E
Published in Journal of medicinal chemistry (26.11.1993)
Published in Journal of medicinal chemistry (26.11.1993)
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