The ferroptosis inducing compounds RSL3 and ML162 are not direct inhibitors of GPX4 but of TXNRD1
Cheff, Dorian M., Huang, Chuying, Scholzen, Karoline C., Gencheva, Radosveta, Ronzetti, Michael H., Cheng, Qing, Hall, Matthew D., Arnér, Elias S.J.
Published in Redox biology (01.06.2023)
Published in Redox biology (01.06.2023)
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Journal Article
Dome1-JAK-STAT signaling between parasite and host integrates vector immunity and development
Rana, Vipin S, Kitsou, Chrysoula, Dutta, Shraboni, Ronzetti, Michael H, Zhang, Min, Bernard, Quentin, Smith, Alexis A, Tomás-Cortázar, Julen, Yang, Xiuli, Wu, Ming-Jie, Kepple, Oleksandra, Li, Weizhong, Dwyer, Jennifer E, Matias, Jaqueline, Baljinnyam, Bolormaa, Oliver, Jonathan D, Rajeevan, Nallakkandi, Pedra, Joao H F, Narasimhan, Sukanya, Wang, Yan, Munderloh, Ulrike, Fikrig, Erol, Simeonov, Anton, Anguita, Juan, Pal, Utpal
Published in Science (American Association for the Advancement of Science) (13.01.2023)
Published in Science (American Association for the Advancement of Science) (13.01.2023)
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Journal Article
Real-Time Cellular Thermal Shift Assay to Monitor Target Engagement
Sanchez, Tino W., Ronzetti, Michael H., Owens, Ashley E., Antony, Maria, Voss, Ty, Wallgren, Eric, Talley, Daniel, Balakrishnan, Krishna, Leyes Porello, Sebastian E., Rai, Ganesha, Marugan, Juan J., Michael, Samuel G., Baljinnyam, Bolormaa, Southall, Noel, Simeonov, Anton, Henderson, Mark J.
Published in ACS chemical biology (16.09.2022)
Published in ACS chemical biology (16.09.2022)
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Journal Article
Application of temperature-responsive HIS-tag fluorophores to differential scanning fluorimetry screening of small molecule libraries
Ronzetti, Michael H, Baljinnyam, Bolormaa, Itkin, Zina, Jain, Sankalp, Rai, Ganesha, Zakharov, Alexey V, Pal, Utpal, Simeonov, Anton
Published in Frontiers in pharmacology (24.11.2022)
Published in Frontiers in pharmacology (24.11.2022)
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Journal Article
Discovery of small molecule inhibitors that effectively disrupt IQGAP1-Cdc42 interaction in breast cancer cells
Sayedyahossein, Samar, Smith, Jessica, Barnaeva, Elena, Li, Zhigang, Choe, Jun, Ronzetti, Michael, Dextras, Christopher, Hu, Xin, Marugan, Juan, Southall, Noel, Baljinnyam, Bolormaa, Thines, Louise, Tran, Andy D, Ferrer, Marc, Sacks, David B
Published in Scientific reports (17.10.2022)
Published in Scientific reports (17.10.2022)
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Journal Article
A unique borrelial protein facilitates microbial immune evasion
Foor, Shelby D, Brangulis, Kalvis, Shakya, Anil K, Rana, Vipin S, Bista, Sandhya, Kitsou, Chrysoula, Ronzetti, Michael, Alreja, Adit B, Linden, Sara B, Altieri, Amanda S, Baljinnyam, Bolormaa, Akopjana, Inara, Nelson, Daniel C, Simeonov, Anton, Herzberg, Osnat, Caimano, Melissa J, Pal, Utpal
Published in mBio (31.10.2023)
Published in mBio (31.10.2023)
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Journal Article
Advances in luminescence-based technologies for drug discovery
Baljinnyam, Bolormaa, Ronzetti, Michael, Simeonov, Anton
Published in Expert opinion on drug discovery (02.01.2023)
Published in Expert opinion on drug discovery (02.01.2023)
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Journal Article
Application of biophysical methods for improved protein production and characterization: A case study on an high‐temperature requirement A‐family bacterial protease
Ronzetti, Michael, Baljinnyam, Bolormaa, Jalal, Ishrat, Pal, Utpal, Simeonov, Anton
Published in Protein science (01.12.2022)
Published in Protein science (01.12.2022)
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Journal Article
Applications of Differential Scanning Fluorometry and Related Technologies in Characterization of Protein-Ligand Interactions
Baljinnyam, Bolormaa, Ronzetti, Michael, Yasgar, Adam, Simeonov, Anton
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2020)
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2020)
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Journal Article
Mannose receptor (CD206) activation in tumor-associated macrophages enhances adaptive and innate antitumor immune responses
Jaynes, Jesse M, Sable, Rushikesh, Ronzetti, Michael, Bautista, Wendy, Knotts, Zachary, Abisoye-Ogunniyan, Abisola, Li, Dandan, Calvo, Raul, Dashnyam, Myagmarjav, Singh, Anju, Guerin, Theresa, White, Jason, Ravichandran, Sarangan, Kumar, Parimal, Talsania, Keyur, Chen, Vicky, Ghebremedhin, Anghesom, Karanam, Balasubramanyam, Bin Salam, Ahmad, Amin, Ruksana, Odzorig, Taivan, Aiken, Taylor, Nguyen, Victoria, Bian, Yansong, Zarif, Jelani C, de Groot, Amber E, Mehta, Monika, Fan, Lixin, Hu, Xin, Simeonov, Anton, Pate, Nathan, Abu-Asab, Mones, Ferrer, Marc, Southall, Noel, Ock, Chan-Young, Zhao, Yongmei, Lopez, Henry, Kozlov, Serguei, de Val, Natalia, Yates, Clayton C, Baljinnyam, Bolormaa, Marugan, Juan, Rudloff, Udo
Published in Science translational medicine (12.02.2020)
Published in Science translational medicine (12.02.2020)
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Journal Article
Abstract B49: Precision targeting of M2-like macrophages by the innate defense regulator RP-182 in pancreatic cancer and noncancerous diseases
Sable, Rushikesh, Jaynes, Jesse, Ronzetti, Michael, Guzman, Wendy, Knotts, Zachary, Val, Natalia de, Morgan, Juan, Yates, Clayton, Bolormaa, Baljinnyam, Rudloff, Udo
Published in Cancer research (Chicago, Ill.) (15.12.2019)
Published in Cancer research (Chicago, Ill.) (15.12.2019)
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Journal Article
Controlled Proteolysis of an Essential Virulence Determinant Dictates Infectivity of Lyme Disease Pathogens
Thakur, Meghna, Bista, Sandhya, Foor, Shelby D, Dutta, Shraboni, Yang, Xiuli, Ronzetti, Michael, Rana, Vipin S, Kitsou, Chrysoula, Linden, Sara B, Altieri, Amanda S, Baljinnyam, Bolormaa, Nelson, Daniel C, Simeonov, Anton, Pal, Utpal
Published in Infection and immunity (19.05.2022)
Published in Infection and immunity (19.05.2022)
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Journal Article
A real-time cellular thermal shift assay (RT-CETSA) to monitor target engagement
Sanchez, Tino W, Ronzetti, Michael H, Owens, Ashley E, Antony, Maria, Voss, Ty, Wallgren, Eric, Talley, Daniel, Balakrishnan, Krishna, Rai, Ganesha, Marugan, Juan J, Sam, Michael, Baljinnyam, Bolormaa, Southall, Noel, Simeonov, Anton, Henderson, Mark J
Published in bioRxiv (27.01.2022)
Published in bioRxiv (27.01.2022)
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