New ligands at the melatonin binding site MT3
Boussard, MF, Truche, S, Rousseau-Rojas, A, Briss, S, Descamps, S, Droual, M, Wierzbicki, M, Ferry, G, Audinot, Delagrange, P, Boutin, JA
Published in European journal of medicinal chemistry (01.03.2006)
Published in European journal of medicinal chemistry (01.03.2006)
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Deep generative models for ligand‐based de novo design applied to multi‐parametric optimization
Perron, Quentin, Mirguet, Olivier, Tajmouati, Hamza, Skiredj, Adam, Rojas, Anne, Gohier, Arnaud, Ducrot, Pierre, Bourguignon, Marie‐Pierre, Sansilvestri‐Morel, Patricia, Do Huu, Nicolas, Gellibert, Françoise, Gaston‐Mathé, Yann
Published in Journal of computational chemistry (15.04.2022)
Published in Journal of computational chemistry (15.04.2022)
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Approach to the specificity and selectivity between D2 and D3 receptors by mutagenesis and binding experiments part I: Expression and characterization of D2 and D3 receptor mutants
Legros, Céline, Rojas, Anne, Dupré, Clémence, Brasseur, Chantal, Riest‐Fery, Isabelle, Muller, Olivier, Ortuno, Jean‐Claude, Nosjean, Olivier, Guenin, Sophie‐Pénélope, Ferry, Gilles, Boutin, Jean A.
Published in Protein science (01.12.2022)
Published in Protein science (01.12.2022)
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Design and synthesis of novel N-sulfonyl-2-indoles that behave as 5-HT6 receptor ligands with significant selectivity for D-3 over D-2 receptors
Saavedra, Oscar M., Karila, Delphine, Brossard, Dominique, Rojas, Anne, Dupuis, Delphine, Gohier, Arnaud, la Cour, Clotilde Mannoury, Millan, Mark J., Ortuno, Jean-Claude, Hanessian, Stephen
Published in Bioorganic & medicinal chemistry (01.01.2017)
Published in Bioorganic & medicinal chemistry (01.01.2017)
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Journal Article
Design and synthesis of novel N-sulfonyl-2-indoles that behave as 5-HT6 receptor ligands with significant selectivity for D3 over D2 receptors
Saavedra, Oscar M., Karila, Delphine, Brossard, Dominique, Rojas, Anne, Dupuis, Delphine, Gohier, Arnaud, Mannoury la Cour, Clotilde, Millan, Mark J., Ortuno, Jean-Claude, Hanessian, Stephen
Published in Bioorganic & medicinal chemistry (01.01.2017)
Published in Bioorganic & medicinal chemistry (01.01.2017)
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Journal Article
Design and synthesis of novel N-sulfonyl-2-indoles that behave as 5-HT 6 receptor ligands with significant selectivity for D 3 over D 2 receptors
Saavedra, Oscar M, Karila, Delphine, Brossard, Dominique, Rojas, Anne, Dupuis, Delphine, Gohier, Arnaud, Mannoury la Cour, Clotilde, Millan, Mark J, Ortuno, Jean-Claude, Hanessian, Stephen
Published in Bioorganic & medicinal chemistry (01.01.2017)
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Published in Bioorganic & medicinal chemistry (01.01.2017)
Journal Article
New ligands at the melatonin binding site MT(3)
Boussard, Marie-Françoise, Truche, Sandrine, Rousseau-Rojas, Anne, Briss, Sylvie, Descamps, Sophie, Droual, Monique, Wierzbicki, Michel, Ferry, Gilles, Audinot, Valérie, Delagrange, Philippe, Boutin, Jean A
Published in European journal of medicinal chemistry (01.03.2006)
Get full text
Published in European journal of medicinal chemistry (01.03.2006)
Journal Article
New ligands at the melatonin binding site MT 3
Boussard, Marie-Françoise, Truche, Sandrine, Rousseau-Rojas, Anne, Briss, Sylvie, Descamps, Sophie, Droual, Monique, Wierzbicki, Michel, Ferry, Gilles, Audinot, Valérie, Delagrange, Philippe, Boutin, Jean A.
Published in European journal of medicinal chemistry (2006)
Published in European journal of medicinal chemistry (2006)
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Journal Article