Hybrid Compound Design To Overcome the Gatekeeper T338M Mutation in cSrc
Getlik, Matthäus, Grütter, Christian, Simard, Jeffrey R, Klüter, Sabine, Rabiller, Matthias, Rode, Haridas B, Robubi, Armin, Rauh, Daniel
Published in Journal of medicinal chemistry (09.07.2009)
Published in Journal of medicinal chemistry (09.07.2009)
Get full text
Journal Article
High-Throughput Screening To Identify Inhibitors Which Stabilize Inactive Kinase Conformations in p38α
Simard, Jeffrey R, Pawar, Vijaykumar, Aust, Beate, Wolf, Alexander, Rabiller, Matthias, Wulfert, Sabine, Robubi, Armin, Klüter, Sabine, Ottmann, Christian, Rauh, Daniel
Published in Journal of the American Chemical Society (30.12.2009)
Published in Journal of the American Chemical Society (30.12.2009)
Get full text
Journal Article
The Tumor Suppressor DiRas3 Forms a Complex with H-Ras and C-RAF Proteins and Regulates Localization, Dimerization, and Kinase Activity of C-RAF
Baljuls, Angela, Beck, Matthias, Oenel, Ayla, Robubi, Armin, Kroschewski, Ruth, Hekman, Mirko, Rudel, Thomas, Rapp, Ulf R.
Published in The Journal of biological chemistry (29.06.2012)
Published in The Journal of biological chemistry (29.06.2012)
Get full text
Journal Article
Structure-based design, synthesis and biological evaluation of N-pyrazole, N′-thiazole urea inhibitors of MAP kinase p38α
Getlik, Matthäus, Grütter, Christian, Simard, Jeffrey R., Nguyen, Hoang D., Robubi, Armin, Aust, Beate, van Otterlo, Willem A.L., Rauh, Daniel
Published in European journal of medicinal chemistry (01.02.2012)
Published in European journal of medicinal chemistry (01.02.2012)
Get full text
Journal Article
RAF Kinase Inhibitors in Cancer Treatment: Like a Bull in a China Shop
Robubi, Armin, Waldmann, Herbert, Rauh, Daniel
Published in Chembiochem : a European journal of chemical biology (16.08.2010)
Published in Chembiochem : a European journal of chemical biology (16.08.2010)
Get full text
Journal Article
Supplementary material to the paper "B-Raf and C-Raf signaling investigated in a simplified model of the mitogenic kinase cascade"
Robubi, Armin, Mueller, Tobias, Fueller, Jochen, Hekman, Mirko, Rapp, Ulf R., Dandekar, Thomas
Published in Biological chemistry (25.11.2005)
Published in Biological chemistry (25.11.2005)
Get full text
Journal Article
B-Raf and C-Raf signaling investigated in a simplified model of the mitogenic kinase cascade
Robubi, Armin, Mueller, Tobias, Fueller, Jochen, Hekman, Mirko, Rapp, Ulf R., Dandekar, Thomas
Published in Biological chemistry (01.11.2005)
Published in Biological chemistry (01.11.2005)
Get full text
Journal Article
High-throughput screening to identify inhibitors which stabilize inactive kinase conformations in p38alpha
Simard, Jeffrey R, Grütter, Christian, Pawar, Vijaykumar, Aust, Beate, Wolf, Alexander, Rabiller, Matthias, Wulfert, Sabine, Robubi, Armin, Klüter, Sabine, Ottmann, Christian, Rauh, Daniel
Published in Journal of the American Chemical Society (30.12.2009)
Published in Journal of the American Chemical Society (30.12.2009)
Get full text
Journal Article