Quinolines as a novel structural class of potent and selective PDE4 inhibitors: Optimisation for oral administration
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Published in Bioorganic & medicinal chemistry letters (01.03.2009)
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The design of potent, non-peptidic inhibitors of hepatitis C protease
Andrews, David M., Chaignot, Helene M., Coomber, Barry A., Dowle, Mike D., Lucy Hind, S., Johnson, Martin R., Jones, Paul S., Mills, Gail, Patikis, Angela, Pateman, Tony J., Ed Robinson, J., Slater, Martin J., Trivedi, Naimisha
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Published in European journal of medicinal chemistry (01.04.2003)
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Andrews, David M, Carey, Seb J, Chaignot, Helene, Coomber, Barry A, Gray, Norman M, Hind, S. Lucy, Jones, Paul S, Mills, Gail, Robinson, J. Ed, Slater, Martin J
Published in Organic letters (12.12.2002)
Published in Organic letters (12.12.2002)
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Pyrrolidine-5,5-trans-lactams. 5. Pharmacokinetic Optimization of Inhibitors of Hepatitis C Virus NS3/4A Protease
Andrews, David M, Barnes, Michael C, Dowle, Mike D, Hind, S. Lucy, Johnson, Martin R, Jones, Paul S, Mills, Gail, Patikis, Angela, Pateman, Tony J, Redfern, Tracy J, Robinson, J. Ed, Slater, Martin J, Trivedi, Naimisha
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Published in Organic letters (27.11.2003)
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Pyrrolidine-5,5-trans-lactams. 2. The Use of X-ray Crystal Structure Data in the Optimization of P3 and P4 Substituents
Andrews, David M, Chaignot, Helene, Coomber, Barry A, Good, Andrew C, Hind, S. Lucy, Johnson, Martin R, Jones, Paul S, Mills, Gail, Robinson, J. Ed, Skarzynski, Tadeusz, Slater, Martin J, Somers, Donald O'N
Published in Organic letters (12.12.2002)
Published in Organic letters (12.12.2002)
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Sialidase inhibitors related to zanamivir: Synthesis and biological evaluation of 4H-pyran 6-ether and ketone
Smith, Paul W., Robinson, J.Ed, Evans, Derek N., Sollis, Steven L., Howes, Peter D., Trivedi, Naimisha, Bethell, Richard C.
Published in Bioorganic & medicinal chemistry letters (22.02.1999)
Published in Bioorganic & medicinal chemistry letters (22.02.1999)
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Pyrrolidine-5,5-trans-lactams - 3. Alternative regiochemical outcome of the acyl-iminium coupling reaction
Andrews, DM, Borthwick, AD, Chaignot, H, Jones, PS, Robinson, E, Shah, P, Slater, MJ, Upton, RJ
Published in Synthesis (Stuttgart) (01.01.2003)
Published in Synthesis (Stuttgart) (01.01.2003)
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