Luminescence screening assays for the identification of sensitizers for lanthanides based on the controlled formation of ternary lanthanide complexes with DTPA-bisamide ligands
Ruston, Linette L, Robertson, Graeme M, Pikramenou, Zoe
Published in Chemistry, an Asian journal (01.03.2010)
Published in Chemistry, an Asian journal (01.03.2010)
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Use of aza-Cope rearrangement-Mannich cyclization reactions to achieve a general entry to Melodinus and Aspidosperma alkaloids. Stereocontrolled total syntheses of (.+-.)-deoxoapodine, (.+-.)-meloscine, and (.+-.)-epimeloscine and a formal synthesis of (.+-.)-1-acetylaspidoalbidine
Overman, Larry E, Robertson, Graeme M, Robichaud, Albert J
Published in Journal of the American Chemical Society (01.03.1991)
Published in Journal of the American Chemical Society (01.03.1991)
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Solution-phase synthesis of ICG-001, a β-turn peptidomimetic molecule inhibitor of β-catenin–Tcf-mediated transcription
Piergentili, Alessandro, Del Bello, Fabio, Gentili, Francesco, Giannella, Mario, Quaglia, Wilma, Vesprini, Cristian, Thomas, Russell J., Robertson, Graeme M.
Published in Tetrahedron (24.12.2007)
Published in Tetrahedron (24.12.2007)
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Modeling the pore structure of voltage-gated sodium channels in closed, open, and fast-inactivated conformation reveals details of site 1 toxin and local anesthetic binding
Scheib, Holger, McLay, Iain, Guex, Nicolas, Clare, Jeff J, Blaney, Frank E, Dale, Tim J, Tate, Simon N, Robertson, Graeme M
Published in Journal of molecular modeling (01.09.2006)
Published in Journal of molecular modeling (01.09.2006)
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Discovery and characterization of novel potent PARP-1 inhibitors endowed with neuroprotective properties: From TIQ-A to HYDAMTIQ
Pellicciari, Roberto, Camaioni, Emidio, Gilbert, Adam M., Macchiarulo, Antonio, Bikker, Jack A., Shah, Falgun, Bard, Joel, Costantino, Gabriele, Gioiello, Antimo, Robertson, Graeme M., Sabbatini, Paola, Venturoni, Francesco, Liscio, Paride, Carotti, Andrea, Bellocchi, Daniele, Cozzi, Andrea, Wood, Andrew, Gonzales, Cathleen, Zaleska, Margaret M., Ellingboe, John W., Moroni, Flavio
Published in MedChemComm (01.06.2011)
Published in MedChemComm (01.06.2011)
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Journal Article
Ask the experts: future of the pharmaceutical industry. Interview by Future Medicinal Chemistry
Cottens, Sylvain, Eaton, Mike, Fuhr, Joseph, Geary, Stewart, Johnson, Douglas S, Li, Ge, Raveglia, Luca, Robertson, Graeme M, Westwell, Andrew
Published in Future medicinal chemistry (01.11.2011)
Published in Future medicinal chemistry (01.11.2011)
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A novel series of arylpiperazines with high affinity and selectivity for the dopamine D3 receptor
John Murray, P., Harrison, Lee A., Johnson, Martin R., Robertson, Graeme M., Scopes, David I.C., Bull, David R., Graham, Elizabeth A., Hayes, Ann G., Kilpatrick, Gavin J., Daas, Izaak Den, Large, Charles, Sheehan, Michael J., Stubbs, Carole M., Turpin, Michael P.
Published in Bioorganic & medicinal chemistry letters (02.02.1995)
Published in Bioorganic & medicinal chemistry letters (02.02.1995)
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Journal Article
A novel series of arylpiperazines with high affinity and selectivity for the dopamine D 3 receptor
John Murray, P., Harrison, Lee A., Johnson, Martin R., Robertson, Graeme M., Scopes, David I.C., Bull, David R., Graham, Elizabeth A., Hayes, Ann G., Kilpatrick, Gavin J., Daas, Izaak Den, Large, Charles, Sheehan, Michael J., Stubbs, Carole M., Turpin, Michael P.
Published in Bioorganic & medicinal chemistry letters (02.02.1995)
Published in Bioorganic & medicinal chemistry letters (02.02.1995)
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ChemInform Abstract: Solution-Phase Synthesis of ICG-001, a β-Turn Peptidomimetic Molecule Inhibitor of β-Catenin-Tcf-Mediated Transcription
Piergentili, Alessandro, Del Bello, Fabio, Gentili, Francesco, Giannella, Mario, Quaglia, Wilma, Vesprini, Cristian, Thomas, Russell J., Robertson, Graeme M.
Published in ChemInform (20.05.2008)
Published in ChemInform (20.05.2008)
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Journal Article
Morpholin-acetamide derivatives for the treatment of inflammatory diseases
HODGSON SIMON T, COOK CAROLINE M, ELDRED COLIN D, JUDD DUNCAN B, ROBERTSON GRAEME M, ANCLIFF RACHAEL A, LEWELL XIAO Q, GORE PAUL M, KEELING SUZANNE E, HARRISON LEE A, SWANSON STEPHEN
Year of Publication 13.04.2006
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Year of Publication 13.04.2006
Patent
Novel compounds
HODGSON SIMON T, MILLS GAIL, ANCLIFF RACHAEL A, HARRISON LEE A, COOK CAROLINE M, ELDRED COLIN D, JUDD DUNCAN B, LEWELL XIAO O, ROBERTSON GRAEME M, GORE PAUL M, KEELING SUZANNE E, WILKINSON MARK, WALKER ANDREW J, HAYES MARTIN A, SWANSON STEPHEN
Year of Publication 23.03.2006
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Year of Publication 23.03.2006
Patent
N-2s-4-3,4-difluorobenzyl morpholin-2yl methyl -2-(3-methylsulphonyl amino!phenyl acetamide as ccr3 antagonist for the treatment of inflammatory conditions
HODGSON SIMON T, MILLS GAIL, ANCLIFF RACHAEL A, LEWELL XIAO Q, HARRISON LEE A, COOK CAROLINE M, ELDRED COLIN D, JUDD DUNCAN B, ROBERTSON GRAEME M, GORE PAUL M, KEELING SUZANNE E, WILKINSON MARK, WALKER ANDREW J, HAYES MARTIN A, SWANSON STEPHEN
Year of Publication 16.03.2006
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Year of Publication 16.03.2006
Patent