Molecular hybridization yields triazole bronchodilators for the treatment of COPD
Jones, Lyn H., Burrows, Jane, Feeder, Neil, Glossop, Paul, James, Kim, Jones, Rhys M., Kenyon, Amy S., Patel, Sheena, Roberts, Dannielle F., Selby, Matthew D., Strang, Ross S., Stuart, Emilio F., Trevethick, Michael A., Watson, Jessica, Wright, Karen N., Clarke, Nick
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
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Development of a Scaleable Synthesis of a Geminal Dimethyl Tertiary Amine as an Inhaled Muscarinic Antagonist for the Treatment of COPD
Dillon, Barry R, Roberts, Dannielle F, Entwistle, David A, Glossop, Paul A, Knight, Craig J, Laity, Daniel A, James, Kim, Praquin, Celine F, Strang, Ross S, Watson, Christine A. L
Published in Organic process research & development (17.02.2012)
Published in Organic process research & development (17.02.2012)
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A perspective on synthetic and solid-form enablement of inhalation candidates
Selby, Matthew D, de Koning, Pieter D, Roberts, Dannielle F
Published in Future medicinal chemistry (01.10.2011)
Published in Future medicinal chemistry (01.10.2011)
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A highly selective method for 11 beta-OH protection of steroidal 11 beta, 17 alpha-diols
Glossop, Paul A., Hoogenraad, Marcel, Peakman, Torren M., Roberts, Dannielle F.
Published in Steroids (01.05.2008)
Published in Steroids (01.05.2008)
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A highly selective method for 11β-OH protection of steroidal 11β, 17α-diols
Glossop, Paul A., Hoogenraad, Marcel, Peakman, Torren M., Roberts, Dannielle F.
Published in Steroids (01.05.2008)
Published in Steroids (01.05.2008)
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Discovery of a Selective TRPM8 Antagonist with Clinical Efficacy in Cold-Related Pain
Andrews, Mark D, af Forselles, Kerry, Beaumont, Kevin, Galan, Sébastien R. G, Glossop, Paul A, Grenie, Mathilde, Jessiman, Alan, Kenyon, Amy S, Lunn, Graham, Maw, Graham, Owen, Robert M, Pryde, David C, Roberts, Dannielle, Tran, Thien Duc
Published in ACS medicinal chemistry letters (09.04.2015)
Published in ACS medicinal chemistry letters (09.04.2015)
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Inhalation by Design: Novel Tertiary Amine Muscarinic M-3 Receptor Antagonists with Slow Off-Rate Binding Kinetics for Inhaled Once-Daily Treatment of Chronic Obstructive Pulmonary Disease
Glossop, Paul A., Watson, Christine A. L., Price, David A., Bunnage, Mark E., Middleton, Donald S., Wood, Anthony, James, Kim, Roberts, Dannielle, Strang, Ross S., Yeadon, Michael, Perros-Huguet, Christelle, Clarke, Nicholas P., Trevethick, Michael A., Machin, Ian, Stuart, Emilio F., Evans, Steven M., Harrison, Anthony C., Fairman, David A., Agoram, Balaji, Burrows, Jane L., Feeder, Neil, Fulton, Craig K., Dillon, Barry R., Entwistle, David A., Spence, Fiona J.
Published in Journal of medicinal chemistry (13.10.2011)
Published in Journal of medicinal chemistry (13.10.2011)
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Journal Article
Inhalation by Design: Novel Tertiary Amine Muscarinic M3 Receptor Antagonists with Slow Off-Rate Binding Kinetics for Inhaled Once-Daily Treatment of Chronic Obstructive Pulmonary Disease
Glossop, Paul A, Watson, Christine A. L, Price, David A, Bunnage, Mark E, Middleton, Donald S, Wood, Anthony, James, Kim, Roberts, Dannielle, Strang, Ross S, Yeadon, Michael, Perros-Huguet, Christelle, Clarke, Nicholas P, Trevethick, Michael A, Machin, Ian, Stuart, Emilio F, Evans, Steven M, Harrison, Anthony C, Fairman, David A, Agoram, Balaji, Burrows, Jane L, Feeder, Neil, Fulton, Craig K, Dillon, Barry R, Entwistle, David A, Spence, Fiona J
Published in Journal of medicinal chemistry (13.10.2011)
Published in Journal of medicinal chemistry (13.10.2011)
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