Structure-activity and structure-property relationship studies of spirocyclic chromanes with antimalarial activity
Iyamu, Iredia D., Zhao, Yingzhao, Parvatkar, Prakash T., Roberts, Bracken F., Casandra, Debora R., Wojtas, Lukasz, Kyle, Dennis E., Chakrabarti, Debopam, Manetsch, Roman
Published in Bioorganic & medicinal chemistry (01.03.2022)
Published in Bioorganic & medicinal chemistry (01.03.2022)
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Journal Article
Parallel Synthesis of Piperazine Tethered Thiazole Compounds with Antiplasmodial Activity
Rayala, Ramanjaneyulu, Chaudhari, Prakash, Bunnell, Ashley, Roberts, Bracken, Chakrabarti, Debopam, Nefzi, Adel
Published in International journal of molecular sciences (12.12.2023)
Published in International journal of molecular sciences (12.12.2023)
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Journal Article
Identification of Bis-Cyclic Guanidines as Antiplasmodial Compounds from Positional Scanning Mixture-Based Libraries
Perry, Jr, David L, Roberts, Bracken F, Debevec, Ginamarie, Michaels, Heather A, Chakrabarti, Debopam, Nefzi, Adel
Published in Molecules (Basel, Switzerland) (20.03.2019)
Published in Molecules (Basel, Switzerland) (20.03.2019)
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Journal Article
Dragmacidin G, a Bioactive Bis-Indole Alkaloid from a Deep-Water Sponge of the Genus Spongosorites
Wright, Amy E, Killday, K Brian, Chakrabarti, Debopam, Guzmán, Esther A, Harmody, Dedra, McCarthy, Peter J, Pitts, Tara, Pomponi, Shirley A, Reed, John K, Roberts, Bracken F, Rodrigues Felix, Carolina, Rohde, Kyle H
Published in Marine drugs (11.01.2017)
Published in Marine drugs (11.01.2017)
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Journal Article
4-Nitro styrylquinoline is an antimalarial inhibiting multiple stages of Plasmodium falciparum asexual life cycle
Roberts, Bracken F., Zheng, Yongsheng, Cleaveleand, Jacob, Lee, Sukjun, Lee, Eunyoung, Ayong, Lawrence, Yuan, Yu, Chakrabarti, Debopam
Published in International journal for parasitology -- drugs and drug resistance (01.04.2017)
Published in International journal for parasitology -- drugs and drug resistance (01.04.2017)
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Journal Article
Characterization of Plasmodium falciparum Atypical Kinase PfPK7– Dependent Phosphoproteome
Pease, Brittany N, Huttlin, Edward L, Jedrychowski, Mark P, Dorin-Semblat, Dominique, Sebastiani, Daniela, Segarra, Daniel T, Roberts, Bracken F, Chakrabarti, Ratna, Doerig, Christian, Gygi, Steven P, Chakrabarti, Debopam
Published in Journal of proteome research (01.06.2018)
Published in Journal of proteome research (01.06.2018)
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Journal Article
Antiplasmodial Compounds from Deep-Water Marine Invertebrates
Wright, Amy E, Collins, Jennifer E, Roberts, Bracken, Roberts, Jill C, Winder, Priscilla L, Reed, John K, Diaz, Maria Cristina, Pomponi, Shirley A, Chakrabarti, Debopam
Published in Marine drugs (25.03.2021)
Published in Marine drugs (25.03.2021)
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Journal Article
Marine microbiome as a source of antimalarials
McCarthy, Peter J, Roberts, Bracken F, Carbonell, Abigail, Roberts, Jill, Wright, Amy E, Chakrabarti, Debopam
Published in Tropical medicine and infectious disease (13.07.2019)
Published in Tropical medicine and infectious disease (13.07.2019)
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Journal Article
Spirocyclic chromanes exhibit antiplasmodial activities and inhibit all intraerythrocytic life cycle stages
Roberts, Bracken F., Iyamu, Iredia D., Lee, Sukjun, Lee, Eunyoung, Ayong, Lawrence, Kyle, Dennis E., Yuan, Yu, Manetsch, Roman, Chakrabarti, Debopam
Published in International journal for parasitology -- drugs and drug resistance (01.04.2016)
Published in International journal for parasitology -- drugs and drug resistance (01.04.2016)
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Journal Article
Anti-parasitic compounds and uses thereof
Verano, Alyssa, McKerrow, James, Tan, Derek Shieh, Foley, Corinne N, Chakrabarti, Debopam, Roberts, Bracken, Dandapani, Sivaraman, Edwankar, Rahul, Moura-Letts, Gustavo
Year of Publication 27.08.2024
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Year of Publication 27.08.2024
Patent
ANTI-PARASITIC COMPOUNDS AND USES THEREOF
Verano, Alyssa, McKerrow, James, Tan, Derek Shieh, Foley, Corinne N, Chakrabarti, Debopam, Roberts, Bracken, Dandapani, Sivaraman, Edwankar, Rahul, Moura-Letts, Gustavo
Year of Publication 27.10.2022
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Year of Publication 27.10.2022
Patent
Anti-parasitic compounds and uses thereof
Verano, Alyssa, McKerrow, James, Tan, Derek Shieh, Foley, Corinne N, Chakrabarti, Debopam, Roberts, Bracken, Dandapani, Sivaraman, Edwankar, Rahul, Moura-Letts, Gustavo
Year of Publication 23.11.2021
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Year of Publication 23.11.2021
Patent
ANTI-PARASITIC COMPOUNDS AND USES THEREOF
MCKERROW, James, ROBERTS, Bracken, TAN, Derek, Shieh, VERANO, Alyssa, EDWANKAR, Rahul, FOLEY, Corinne, N, DANDAPANI, Sivaraman, MOURA-LETTS, Gustavo, CHAKRABARTI, Debopam
Year of Publication 20.07.2017
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Year of Publication 20.07.2017
Patent