The Alpha Keto Amide Moiety as a Privileged Motif in Medicinal Chemistry: Current Insights and Emerging Opportunities
Robello, Marco, Barresi, Elisabetta, Baglini, Emma, Salerno, Silvia, Taliani, Sabrina, Settimo, Federico Da
Published in Journal of medicinal chemistry (08.04.2021)
Published in Journal of medicinal chemistry (08.04.2021)
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Journal Article
Indol-3-ylglyoxylamide as Privileged Scaffold in Medicinal Chemistry
Barresi, Elisabetta, Robello, Marco, Baglini, Emma, Poggetti, Valeria, Viviano, Monica, Salerno, Silvia, Da Settimo, Federico, Taliani, Sabrina
Published in Pharmaceuticals (Basel, Switzerland) (01.07.2023)
Published in Pharmaceuticals (Basel, Switzerland) (01.07.2023)
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Journal Article
An update into the medicinal chemistry of translocator protein (TSPO) ligands
Barresi, Elisabetta, Robello, Marco, Costa, Barbara, Da Pozzo, Eleonora, Baglini, Emma, Salerno, Silvia, Da Settimo, Federico, Martini, Claudia, Taliani, Sabrina
Published in European journal of medicinal chemistry (01.01.2021)
Published in European journal of medicinal chemistry (01.01.2021)
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Journal Article
Multiple Topoisomerase I (TopoI), Topoisomerase II (TopoII) and Tyrosyl-DNA Phosphodiesterase (TDP) inhibitors in the development of anticancer drugs
Baglini, Emma, Salerno, Silvia, Barresi, Elisabetta, Robello, Marco, Da Settimo, Federico, Taliani, Sabrina, Marini, Anna Maria
Published in European journal of pharmaceutical sciences (01.01.2021)
Published in European journal of pharmaceutical sciences (01.01.2021)
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Journal Article
New antiproliferative agents derived from tricyclic 3,4‐dihydrobenzo[4,5]imidazo[1,2‐a][1,3,5]triazine scaffold: Synthesis and pharmacological effects
Robello, Marco, Salerno, Silvia, Barresi, Elisabetta, Orlandi, Paola, Vaglini, Francesca, Banchi, Marta, Simorini, Francesca, Baglini, Emma, Poggetti, Valeria, Taliani, Sabrina, Da Settimo, Federico, Bocci, Guido
Published in Archiv der Pharmazie (Weinheim) (01.11.2022)
Published in Archiv der Pharmazie (Weinheim) (01.11.2022)
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Journal Article
New antiproliferative agents derived from tricyclic 3,4‐dihydrobenzoimidazotriazine scaffold: Synthesis and pharmacological effects
Robello, Marco, Salerno, Silvia, Barresi, Elisabetta, Orlandi, Paola, Vaglini, Francesca, Banchi, Marta, Simorini, Francesca, Baglini, Emma, Poggetti, Valeria, Taliani, Sabrina, Federico Da Settimo, Bocci, Guido
Published in Archiv der Pharmazie (Weinheim) (01.11.2022)
Published in Archiv der Pharmazie (Weinheim) (01.11.2022)
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Journal Article
Novel fluorescent triazinobenzimidazole derivatives as probes for labelling human A(1) and A(2B) adenosine receptor subtypes
Barresi, Elisabetta, Giacomelli, Chiara, Daniele, Simona, Tonazzini, Ilaria, Robello, Marco, Salerno, Silvia, Piano, Ilaria, Cosimelli, Barbara, Greco, Giovanni, Da Settimo, Federico, Martini, Claudia, Trincavelli, Maria Letizia, Taliani, Sabrina
Published in Bioorganic & medicinal chemistry (01.12.2018)
Published in Bioorganic & medicinal chemistry (01.12.2018)
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Journal Article
Alkyl-substituted N-methylaryl-N′-aryl-4-aminobenzamides: A new series of small molecule inhibitors for Wip1 phosphatase
Robello, Marco, Zheng, Hongchao, Saha, Mrinmoy, George Rosenker, Kara M., Debnath, Subrata, Kumar, Jay Prakash, Tagad, Harichandra D., Mazur, Sharlyn J., Appella, Ettore, Appella, Daniel H.
Published in European journal of medicinal chemistry (05.12.2022)
Published in European journal of medicinal chemistry (05.12.2022)
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Journal Article
Novel fluorescent triazinobenzimidazole derivatives as probes for labelling human A1 and A2B adenosine receptor subtypes
Barresi, Elisabetta, Giacomelli, Chiara, Daniele, Simona, Tonazzini, Ilaria, Robello, Marco, Salerno, Silvia, Piano, Ilaria, Cosimelli, Barbara, Greco, Giovanni, Da Settimo, Federico, Martini, Claudia, Trincavelli, Maria Letizia, Taliani, Sabrina
Published in Bioorganic & medicinal chemistry (01.12.2018)
Published in Bioorganic & medicinal chemistry (01.12.2018)
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Journal Article
Lead Optimization of 2‑Phenylindolylglyoxylyldipeptide Murine Double Minute (MDM)2/Translocator Protein (TSPO) Dual Inhibitors for the Treatment of Gliomas
Daniele, Simona, La Pietra, Valeria, Barresi, Elisabetta, Di Maro, Salvatore, Da Pozzo, Eleonora, Robello, Marco, La Motta, Concettina, Cosconati, Sandro, Taliani, Sabrina, Marinelli, Luciana, Novellino, Ettore, Martini, Claudia, Da Settimo, Federico
Published in Journal of medicinal chemistry (26.05.2016)
Published in Journal of medicinal chemistry (26.05.2016)
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Journal Article
Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases
Salerno, Silvia, La Pietra, Valeria, Hyeraci, Mariafrancesca, Taliani, Sabrina, Robello, Marco, Barresi, Elisabetta, Milite, Ciro, Simorini, Francesca, García-Argáez, Aída Nelly, Marinelli, Luciana, Novellino, Ettore, Da Settimo, Federico, Marini, Anna Maria, Dalla Via, Lisa
Published in European journal of medicinal chemistry (01.03.2019)
Published in European journal of medicinal chemistry (01.03.2019)
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Journal Article
Prodrug Strategy Extends the Use of Anti-HIV Sulfanylbenzamides for Application In Vivo
Robello, Marco, Nikolayevskiy, Herman, Scerba, Michael T., Nahui Palomino, Rogers Alberto, Mercurio, Vincenzo, Appella, Daniel H.
Published in ACS pharmacology & translational science (12.01.2024)
Published in ACS pharmacology & translational science (12.01.2024)
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Journal Article
The structure-activity profile of mercaptobenzamides’ anti-HIV activity suggests that thermodynamics of metabolism is more important than binding affinity to the target
Nikolayevskiy, Herman, Robello, Marco, Scerba, Michael T., Pasternak, Evan H., Saha, Mrinmoy, Hartman, Tracy L., Buchholz, Caitlin A., Buckheit, Robert W., Durell, Stewart R., Appella, Daniel H.
Published in European journal of medicinal chemistry (15.09.2019)
Published in European journal of medicinal chemistry (15.09.2019)
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Journal Article
Residence Time, a New parameter to Predict Neurosteroidogenic Efficacy of Translocator Protein (TSPO) Ligands: the Case Study of N,N‐Dialkyl‐2‐arylindol‐3‐ylglyoxylamides
Costa, Barbara, Taliani, Sabrina, Da Pozzo, Eleonora, Barresi, Elisabetta, Robello, Marco, Cavallini, Chiara, Cosconati, Sandro, Da Settimo, Federico, Novellino, Ettore, Martini, Claudia
Published in ChemMedChem (22.08.2017)
Published in ChemMedChem (22.08.2017)
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Abstract A103: Targeting mutant p53-R248W reactivates WT p53 function and alters the onco-metabolic profile
Brown, Kate, Jenkins, Lisa, Crooks, Dan, Surman, Deborah, Mazur, Sharlyn, Xu, Yuan, Arimilli, Bhargav, Yang, Ye, Lane, Andrew, Durell, Stewart, Fan, Teresa, Schrump, David, Marston, Marston, Ripley, Taylor, Appella, Ettore, Lyons, Gaelyn, Perciaccante, Andrew, Dinan, Jerry, Robello, Marco, Nikolayevskiy, Herman, O’Connor, Robert, Appella, Daniel
Published in Molecular cancer therapeutics (01.12.2023)
Published in Molecular cancer therapeutics (01.12.2023)
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Journal Article
Toward PET imaging of A2B adenosine receptors: a carbon-11 labeled triazinobenzimidazole tracer: Synthesis and imaging of a new A2B PET tracer
Petroni, Debora, Giacomelli, Chiara, Taliani, Sabrina, Barresi, Elisabetta, Robello, Marco, Daniele, Simona, Bartoli, Antonietta, Burchielli, Silvia, Pardini, Silvia, Salvadori, Piero A, Da Settimo, Federico, Martini, Claudia, Trincavelli, Maria Letizia, Menichetti, Luca
Published in Nuclear medicine and biology (01.05.2016)
Published in Nuclear medicine and biology (01.05.2016)
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Journal Article
Toward PET imaging of A2B adenosine receptors: a carbon-11 labeled triazinobenzimidazole tracer
Petroni, Debora, Giacomelli, Chiara, Taliani, Sabrina, Barresi, Elisabetta, Robello, Marco, Daniele, Simona, Bartoli, Antonietta, Burchielli, Silvia, Pardini, Silvia, Salvadori, Piero A., Da Settimo, Federico, Martini, Claudia, Trincavelli, Maria Letizia, Menichetti, Luca
Published in Nuclear medicine and biology (01.05.2016)
Published in Nuclear medicine and biology (01.05.2016)
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Journal Article
Towards PET imaging of A2B Adenosine Receptors: a carbon-11 labeled triazinobenzimidazole tracer
Petroni, Debora, Giacomelli, Chiara, Taliani, Sabrina, Barresi, Elisabetta, Robello, Marco, Daniele, Simona, Bartoli, Antonietta, Burchielli, Silvia, Pardini, Silvia, Salvadori, Piero A, Da Settimo, Federico, Martini, Claudia, Trincavelli, Maria Letizia, Menichetti, Luca
Published in Nuclear medicine and biology (2016)
Published in Nuclear medicine and biology (2016)
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Journal Article
Novel fluorescent triazinobenzimidazole derivatives as probes for labelling human A 1 and A 2B adenosine receptor subtypes
Barresi, Elisabetta, Giacomelli, Chiara, Daniele, Simona, Tonazzini, Ilaria, Robello, Marco, Salerno, Silvia, Piano, Ilaria, Cosimelli, Barbara, Greco, Giovanni, Da Settimo, Federico, Martini, Claudia, Trincavelli, Maria Letizia, Taliani, Sabrina
Published in Bioorganic & medicinal chemistry (01.12.2018)
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Published in Bioorganic & medicinal chemistry (01.12.2018)
Journal Article