Hit and lead criteria in drug discovery for infectious diseases of the developing world
Katsuno, Kei, Burrows, Jeremy N, Duncan, Ken, Hooft van Huijsduijnen, Rob, Kaneko, Takushi, Kita, Kiyoshi, Mowbray, Charles E, Schmatz, Dennis, Warner, Peter, Slingsby, B T
Published in Nature reviews. Drug discovery (01.11.2015)
Published in Nature reviews. Drug discovery (01.11.2015)
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Journal Article
Partnering to fight malaria in India: Past, present and future
Samby, Kirandeep, Ramachandruni, Hanu, Banerji, Jaya, Burrows, Jeremy, Daumerie, Penny, Hooft van Huijsduijnen, Rob, Duparc, Stephan, Wells, Timothy
Published in Journal of vector borne diseases (01.01.2019)
Published in Journal of vector borne diseases (01.01.2019)
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Journal Article
New developments in anti-malarial target candidate and product profiles
Burrows, Jeremy N, Duparc, Stephan, Gutteridge, Winston E, Hooft van Huijsduijnen, Rob, Kaszubska, Wiweka, Macintyre, Fiona, Mazzuri, Sébastien, Möhrle, Jörg J, Wells, Timothy N C
Published in Malaria journal (13.01.2017)
Published in Malaria journal (13.01.2017)
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Journal Article
Antimalarial activity of single-dose DSM265, a novel plasmodium dihydroorotate dehydrogenase inhibitor, in patients with uncomplicated Plasmodium falciparum or Plasmodium vivax malaria infection: a proof-of-concept, open-label, phase 2a study
Llanos-Cuentas, Alejandro, Casapia, Martin, Chuquiyauri, Raúl, Hinojosa, Juan-Carlos, Kerr, Nicola, Rosario, Maria, Toovey, Stephen, Arch, Robert H, Phillips, Margaret A, Rozenberg, Felix D, Bath, Jade, Ng, Caroline L, Cowell, Annie N, Winzeler, Elizabeth A, Fidock, David A, Baker, Mark, Möhrle, Jörg J, Hooft van Huijsduijnen, Rob, Gobeau, Nathalie, Araeipour, Nada, Andenmatten, Nicole, Rückle, Thomas, Duparc, Stephan
Published in The Lancet infectious diseases (01.08.2018)
Published in The Lancet infectious diseases (01.08.2018)
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Journal Article
Multidrug-resistant gonorrhea: A research and development roadmap to discover new medicines
Alirol, Emilie, Wi, Teodora E, Bala, Manju, Bazzo, Maria Luiza, Chen, Xiang-Sheng, Deal, Carolyn, Dillon, Jo-Anne R, Kularatne, Ranmini, Heim, Jutta, Hooft van Huijsduijnen, Rob, Hook, Edward W, Lahra, Monica M, Lewis, David A, Ndowa, Francis, Shafer, William M, Tayler, Liz, Workowski, Kimberly, Unemo, Magnus, Balasegaram, Manica
Published in PLoS medicine (26.07.2017)
Published in PLoS medicine (26.07.2017)
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Journal Article
A Phase II pilot trial to evaluate safety and efficacy of ferroquine against early Plasmodium falciparum in an induced blood-stage malaria infection study
McCarthy, James S, Rückle, Thomas, Djeriou, Elhadj, Cantalloube, Cathy, Ter-Minassian, Daniel, Baker, Mark, O'Rourke, Peter, Griffin, Paul, Marquart, Louise, Hooft van Huijsduijnen, Rob, Möhrle, Jörg J
Published in Malaria journal (13.09.2016)
Published in Malaria journal (13.09.2016)
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Journal Article
Two successful decades of Swiss collaborations to develop new anti-malarials
Hooft van Huijsduijnen, Rob, Wells, Timothy, Tanner, Marcel, Wittlin, Sergio
Published in Malaria journal (22.03.2019)
Published in Malaria journal (22.03.2019)
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Journal Article
Anticancer properties of distinct antimalarial drug classes
Hooft van Huijsduijnen, Rob, Guy, R Kiplin, Chibale, Kelly, Haynes, Richard K, Peitz, Ingmar, Kelter, Gerhard, Phillips, Margaret A, Vennerstrom, Jonathan L, Yuthavong, Yongyuth, Wells, Timothy N C
Published in PloS one (31.12.2013)
Published in PloS one (31.12.2013)
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Journal Article
A discovery and development roadmap for new endectocidal transmission-blocking agents in malaria
Burrows, Jeremy, Slater, Hannah, Macintyre, Fiona, Rees, Sarah, Thomas, Anna, Okumu, Fredros, Hooft van Huijsduijnen, Rob, Duparc, Stephan, Wells, Timothy N C
Published in Malaria journal (10.12.2018)
Published in Malaria journal (10.12.2018)
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Journal Article
Injectable anti-malarials revisited: discovery and development of new agents to protect against malaria
Macintyre, Fiona, Ramachandruni, Hanu, Burrows, Jeremy N, Holm, René, Thomas, Anna, Möhrle, Jörg J, Duparc, Stephan, Hooft van Huijsduijnen, Rob, Greenwood, Brian, Gutteridge, Winston E, Wells, Timothy N C, Kaszubska, Wiweka
Published in Malaria journal (01.11.2018)
Published in Malaria journal (01.11.2018)
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Journal Article
12/15-lipoxygenase–derived lipid peroxides control receptor tyrosine kinase signaling through oxidation of protein tyrosine phosphatases
Conrad, Marcus, Sandin, Åsa, Förster, Heidi, Seiler, Alexander, Frijhoff, Jeroen, Dagnell, Markus, Bornkamm, Georg W., Rådmark, Olof, van Huijsduijnen, Rob Hooft, Aspenström, Pontus, Böhmer, Frank, Östman, Arne, Schlessinger, Joseph
Published in Proceedings of the National Academy of Sciences - PNAS (07.09.2010)
Published in Proceedings of the National Academy of Sciences - PNAS (07.09.2010)
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Journal Article
Reduction of heart failure by pharmacological inhibition or gene deletion of protein tyrosine phosphatase 1B
Gomez, Elodie, Vercauteren, Magali, Kurtz, Baptiste, Ouvrard-Pascaud, Antoine, Mulder, Paul, Henry, Jean-Paul, Besnier, Marie, Waget, Aurélie, Hooft Van Huijsduijnen, Rob, Tremblay, Michel L, Burcelin, Remy, Thuillez, Christian, Richard, Vincent
Published in Journal of molecular and cellular cardiology (01.06.2012)
Published in Journal of molecular and cellular cardiology (01.06.2012)
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Journal Article
Structural Basis for Selective Inhibition of Mycobacterium tuberculosis Protein Tyrosine Phosphatase PtpB
Grundner, Christoph, Perrin, Dominique, Hooft van Huijsduijnen, Rob, Swinnen, Dominique, Gonzalez, Jérome, Gee, Christine L., Wells, Timothy N., Alber, Tom
Published in Structure (London) (01.04.2007)
Published in Structure (London) (01.04.2007)
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Journal Article
Malaria medicines: a glass half full?
Wells, Timothy N C, Hooft van Huijsduijnen, Rob, Van Voorhis, Wesley C
Published in Nature reviews. Drug discovery (01.06.2015)
Published in Nature reviews. Drug discovery (01.06.2015)
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Journal Article
Identification of VHY/Dusp15 as a regulator of oligodendrocyte differentiation through a systematic genomics approach
Schmidt, Fanny, van den Eijnden, Monique, Pescini Gobert, Rosanna, Saborio, Gabriela P, Carboni, Susanna, Alliod, Chantal, Pouly, Sandrine, Staugaitis, Susan M, Dutta, Ranjan, Trapp, Bruce, Hooft van Huijsduijnen, Rob
Published in PloS one (11.07.2012)
Published in PloS one (11.07.2012)
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Journal Article
Improvement of peripheral endothelial dysfunction by protein tyrosine phosphatase inhibitors in heart failure
VERCAUTEREN, Magali, REMY, Elise, RICHARD, Vincent, DEVAUX, Corinne, DAUTREAUX, Brigitte, HENRY, Jean-Paul, BAUER, Fabrice, MULDER, Paul, VAN HUIJSDUIJNEN, Rob Hooft, BOMBRUN, Agnès, THUILLEZ, Christian
Published in Circulation (New York, N.Y.) (05.12.2006)
Published in Circulation (New York, N.Y.) (05.12.2006)
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Journal Article
The antimalarial pipeline
Hooft van Huijsduijnen, Rob, Wells, Timothy NC
Published in Current opinion in pharmacology (01.10.2018)
Published in Current opinion in pharmacology (01.10.2018)
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Journal Article