Global target profile of the kinase inhibitor bosutinib in primary chronic myeloid leukemia cells
REMSING RIX, L. L, RIX, U, TILL, J. H, SUPERTI-FURGA, G, COLINGE, J, HANTSCHEL, O, BENNETT, K. L, STRANZL, T, MÜLLER, A, BAUMGARTNER, C, VALENT, P, AUGUSTIN, M
Published in Leukemia (01.03.2009)
Published in Leukemia (01.03.2009)
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Journal Article
IGF-binding proteins secreted by cancer-associated fibroblasts induce context-dependent drug sensitization of lung cancer cells
Remsing Rix, Lily L, Sumi, Natalia J, Hu, Qianqian, Desai, Bina, Bryant, Annamarie T, Li, Xueli, Welsh, Eric A, Fang, Bin, Kinose, Fumi, Kuenzi, Brent M, Chen, Y Ann, Antonia, Scott J, Lovly, Christine M, Koomen, John M, Haura, Eric B, Marusyk, Andriy, Rix, Uwe
Published in Science signaling (16.08.2022)
Published in Science signaling (16.08.2022)
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Chemical proteomic profiles of the BCR-ABL inhibitors imatinib, nilotinib, and dasatinib reveal novel kinase and nonkinase targets
Rix, Uwe, Hantschel, Oliver, Dürnberger, Gerhard, Remsing Rix, Lily L., Planyavsky, Melanie, Fernbach, Nora V., Kaupe, Ines, Bennett, Keiryn L., Valent, Peter, Colinge, Jacques, Köcher, Thomas, Superti-Furga, Giulio
Published in Blood (01.12.2007)
Published in Blood (01.12.2007)
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Journal Article
Off-target based drug repurposing opportunities for tivantinib in acute myeloid leukemia
Kuenzi, Brent M, Remsing Rix, Lily L, Kinose, Fumi, Kroeger, Jodi L, Lancet, Jeffrey E, Padron, Eric, Rix, Uwe
Published in Scientific reports (24.01.2019)
Published in Scientific reports (24.01.2019)
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Journal Article
Proteome-wide Profiling of Clinical PARP Inhibitors Reveals Compound-Specific Secondary Targets
Knezevic, Claire E., Wright, Gabriela, Remsing Rix, Lily L., Kim, Woosuk, Kuenzi, Brent M., Luo, Yunting, Watters, January M., Koomen, John M., Haura, Eric B., Monteiro, Alvaro N., Radu, Caius, Lawrence, Harshani R., Rix, Uwe
Published in Cell chemical biology (22.12.2016)
Published in Cell chemical biology (22.12.2016)
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Journal Article
Lowering Sample Requirements to Study Tyrosine Kinase Signaling Using Phosphoproteomics with the TMT Calibrator Approach
Fang, Bin, Izumi, Victoria, Rix, Lily L. Remsing, Welsh, Eric, Pike, Ian, Reuther, Gary W., Haura, Eric B., Rix, Uwe, Koomen, John M.
Published in Proteomics (Weinheim) (01.12.2020)
Published in Proteomics (Weinheim) (01.12.2020)
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Journal Article
Polypharmacology-based ceritinib repurposing using integrated functional proteomics
Kuenzi, Brent M, Remsing Rix, Lily L, Stewart, Paul A, Fang, Bin, Kinose, Fumi, Bryant, Annamarie T, Boyle, Theresa A, Koomen, John M, Haura, Eric B, Rix, Uwe
Published in Nature chemical biology (01.12.2017)
Published in Nature chemical biology (01.12.2017)
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Journal Article
Dissection of TBK1 signaling via phosphoproteomics in lung cancer cells
Kim, Jae-Young, Welsh, Eric A., Oguz, Umut, Fang, Bin, Bai, Yun, Kinose, Fumi, Bronk, Crystina, Rix, Lily L. Remsing, Beg, Amer A., Rix, Uwe, Eschrich, Steven A., Koomen, John M., Haura, Eric B.
Published in Proceedings of the National Academy of Sciences - PNAS (23.07.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (23.07.2013)
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Journal Article
Dual Targeting of WEE1 and PLK1 by AZD1775 Elicits Single Agent Cellular Anticancer Activity
Wright, Gabriela, Golubeva, Volha, Remsing Rix, Lily L, Berndt, Norbert, Luo, Yunting, Ward, Grace A, Gray, Jhanelle E, Schonbrunn, Ernst, Lawrence, Harshani R, Monteiro, Alvaro N.A, Rix, Uwe
Published in ACS chemical biology (21.07.2017)
Published in ACS chemical biology (21.07.2017)
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Journal Article
Differential network analysis of ROS1 inhibitors reveals lorlatinib polypharmacology through co-targeting PYK2
Liao, Yi, Remsing Rix, Lily L., Li, Xueli, Fang, Bin, Izumi, Victoria, Welsh, Eric A., Monastyrskyi, Andrii, Haura, Eric B., Koomen, John M., Doebele, Robert C., Rix, Uwe
Published in Cell chemical biology (15.02.2024)
Published in Cell chemical biology (15.02.2024)
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Journal Article
GSK3 Alpha and Beta Are New Functionally Relevant Targets of Tivantinib in Lung Cancer Cells
Remsing Rix, Lily L, Kuenzi, Brent M, Luo, Yunting, Remily-Wood, Elizabeth, Kinose, Fumi, Wright, Gabriela, Li, Jiannong, Koomen, John M, Haura, Eric B, Lawrence, Harshani R, Rix, Uwe
Published in ACS chemical biology (21.02.2014)
Published in ACS chemical biology (21.02.2014)
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Journal Article
Divergent Polypharmacology-Driven Cellular Activity of Structurally Similar Multi-Kinase Inhibitors through Cumulative Effects on Individual Targets
Sumi, Natalia J, Ctortecka, Claudia, Hu, Qianqian, Bryant, Annamarie T, Fang, Bin, Remsing Rix, Lily L, Ayaz, Muhammad, Kinose, Fumi, Welsh, Eric A, Eschrich, Steven A, Lawrence, Harshani R, Koomen, John M, Haura, Eric B, Rix, Uwe
Published in Cell chemical biology (19.09.2019)
Published in Cell chemical biology (19.09.2019)
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Journal Article
Functional Proteomics and Deep Network Interrogation Reveal a Complex Mechanism of Action of Midostaurin in Lung Cancer Cells
Ctortecka, Claudia, Palve, Vinayak, Kuenzi, Brent M., Fang, Bin, Sumi, Natalia J., Izumi, Victoria, Novakova, Silvia, Kinose, Fumi, Remsing Rix, Lily L., Haura, Eric B., Koomen, John Matthew, Rix, Uwe
Published in Molecular & cellular proteomics (01.12.2018)
Published in Molecular & cellular proteomics (01.12.2018)
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Journal Article
A comprehensive target selectivity survey of the BCR-ABL kinase inhibitor INNO-406 by kinase profiling and chemical proteomics in chronic myeloid leukemia cells
RIX, U, REMSING RIX, L. L, AUGUSTIN, M, TILL, J. H, HEINRICH, M. C, VALENT, P, SUPERTI-FURGA, G, TERKER, A. S, FERNBACH, N. V, HANTSCHEL, O, PLANYAVSKY, M, BREITWIESER, F. P, HERRMANN, H, COLINGE, J, BENNETT, K. L
Published in Leukemia (01.01.2010)
Published in Leukemia (01.01.2010)
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Dabrafenib inhibits the growth of BRAF‐WT cancers through CDK16 and NEK9 inhibition
Phadke, Manali, Remsing Rix, Lily L., Smalley, Inna, Bryant, Annamarie T., Luo, Yunting, Lawrence, Harshani R., Schaible, Braydon J., Chen, Yian A., Rix, Uwe, Smalley, Keiran S. M.
Published in Molecular oncology (01.01.2018)
Published in Molecular oncology (01.01.2018)
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Journal Article
Characterization of epidermal growth factor receptor (EGFR) P848L, an unusual EGFR variant present in lung cancer patients, in a murine Ba/F3 model
Sarcar, Bhaswati, Gimbrone, Nicholas T., Wright, Gabriela, Remsing Rix, Lily L., Gordian, Edna R., Rix, Uwe, Chiappori, Alberto A., Reuther, Gary W., Santiago‐Cardona, Pedro G., Muñoz‐Antonia, Teresita, Cress, William Douglas
Published in FEBS open bio (01.10.2019)
Published in FEBS open bio (01.10.2019)
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Turning liabilities into opportunities: Off-target based drug repurposing in cancer
Palve, Vinayak, Liao, Yi, Remsing Rix, Lily L., Rix, Uwe
Published in Seminars in cancer biology (01.01.2021)
Published in Seminars in cancer biology (01.01.2021)
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