Research modular tool system influence on the dynamic characteristics of the boring machines
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Conference Proceeding
To the problem of computer-aided design of gear-and-leverage mechanisms
Rivkin, Alexey, Sobolev, Alexandr, Nekrasov, Alexey, Arbuzov, Michael
Published in MATEC Web of Conferences (2020)
Published in MATEC Web of Conferences (2020)
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Journal Article
Conference Proceeding
Structural basis for therapeutic inhibition of influenza A polymerase PB2 subunit
Ma, Xiaolei, Xie, Lili, Wartchow, Charles, Warne, Robert, Xu, Yongjin, Rivkin, Alexey, Tully, David, Shia, Steven, Uehara, Kyoko, Baldwin, Dianna M., Muiru, Gladys, Zhong, Weidong, Zaror, Isabel, Bussiere, Dirksen E., Leonard, Vincent H. J.
Published in Scientific reports (24.08.2017)
Published in Scientific reports (24.08.2017)
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A novel strategy for the synthesis of uracil derivatives using bis(pentafluorophenyl)imidodicarbonate
Chichetti, Stephanie M., Ahearn, Sean P., Rivkin, Alexey
Published in Tetrahedron letters (13.10.2008)
Published in Tetrahedron letters (13.10.2008)
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Journal Article
Complex Target-Oriented Total Synthesis in the Drug Discovery Process: The Discovery of a Highly Promising Family of Second Generation Epothilones
Rivkin, Alexey, Yoshimura, Fumihiko, Gabarda, Ana E, Chou, Ting-Chao, Dong, Huajin, Tong, William P, Danishefsky, Samuel J
Published in Journal of the American Chemical Society (12.03.2003)
Published in Journal of the American Chemical Society (12.03.2003)
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Journal Article
On the Introduction of a Trifluoromethyl Substituent in the Epothilone Setting: Chemical Issues Related to Ring Forming Olefin Metathesis and Earliest Biological Findings
Rivkin, Alexey, Biswas, Kaustav, Chou, Ting-Chao, Danishefsky, Samuel J
Published in Organic letters (14.11.2002)
Published in Organic letters (14.11.2002)
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Journal Article
Beyond Rule of Five and PROTACs in Modern Drug Discovery: Polarity Reducers, Chameleonicity, and the Evolving Physicochemical Landscape
Price, Edward, Weinheimer, Manuel, Rivkin, Alexey, Jenkins, Gary, Nijsen, Marjoleen, Cox, Philip B., DeGoey, David
Published in Journal of medicinal chemistry (11.04.2024)
Published in Journal of medicinal chemistry (11.04.2024)
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Journal Article
Use of allylic triflones for allylation of C-H bonds
Xiang, Jason, Evarts, Jerry, Rivkin, Alexey, Curran, Dennis P., Fuchs, P.L.
Published in Tetrahedron letters (01.06.1998)
Published in Tetrahedron letters (01.06.1998)
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Journal Article
Determination of the Optimal Temperature for Processing Styrofoam with a Thermo-Tool
Sobolev, Alexandr N., Rivkin, Alexey V., Arbuzov, Michael O., Nekrasov, Alexey Ja
Published in Key engineering materials (15.02.2022)
Published in Key engineering materials (15.02.2022)
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Journal Article
Abbv-101, a Highly Potent and Selective Clinical Stage Bruton Tyrosine Kinase Degrader for the Treatment of B-Cell Malignancies
Pan, Chin, Gururaja, Tarikere L, Li, Haiyan, Nguyen, Henry, Zhai, Yongjiao, Xie, Xiaoping, Ding, Rong-Xian, Mathew, Rebecca, Hoh, Hana Y, Jia, Zhaozhong J, Liu, Bo, Shu, Cassandra, Assaily, Wissam, Lam, Lloyd T, Riehm, Jacob J, Stevenson, Claudina, Will, Christine, Innocenti, Federico, Rivkin, Alexey
Published in Blood (02.11.2023)
Published in Blood (02.11.2023)
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Journal Article
In Vitro and In Vivo Properties of CUO246, a Novel Bacterial DNA Gyrase/Topoisomerase IV Inhibitor
Blais, Johanne, Dean, Charles R, Lapointe, Guillaume, Leeds, Jennifer A, Ma, Sylvia, Morris, Laura, Moser, Heinz E, Osborne, Colin S, Prosen, Katherine R, Richie, Daryl, Skepper, Colin, Thompson, Katherine, Vo, Jason, Yue, Qin, Rivkin, Alexey
Published in Antimicrobial agents and chemotherapy (20.12.2022)
Published in Antimicrobial agents and chemotherapy (20.12.2022)
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Journal Article
Rationalization of load distribution in multi-pair gearing based on a discrete contact model
Rivkin, Alexey, Nekrasov, Alexey, Sobolev, Alexandr, Arbusov, Michael
Published in Materials today : proceedings (01.01.2021)
Published in Materials today : proceedings (01.01.2021)
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Journal Article
The features of the gears profile forming by the electrical discharge machining
Rivkin, Alexey, Nekrasov, Alexey, Sobolev, Alexandr, Arbusov, Michael
Published in Materials today : proceedings (01.01.2021)
Published in Materials today : proceedings (01.01.2021)
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Journal Article
Topoisomerase Inhibitors Addressing Fluoroquinolone Resistance in Gram-Negative Bacteria
Skepper, Colin K, Armstrong, Duncan, Balibar, Carl J, Bauer, Daniel, Bellamacina, Cornelia, Benton, Bret M, Bussiere, Dirksen, De Pascale, Gianfranco, De Vicente, Javier, Dean, Charles R, Dhumale, Bhavesh, Fisher, L. Mark, Fuller, John, Fulsunder, Mangesh, Holder, Lauren M, Hu, Cheng, Kantariya, Bhavin, Lapointe, Guillaume, Leeds, Jennifer A, Li, Xiaolin, Lu, Peichao, Lvov, Anatoli, Ma, Sylvia, Madhavan, Shravanthi, Malekar, Swapnil, McKenney, David, Mergo, Wosenu, Metzger, Louis, Moser, Heinz E, Mutnick, Daniel, Noeske, Jonas, Osborne, Colin, Patel, Ashish, Patel, Darshit, Patel, Tushar, Prajapati, Krunal, Prosen, Katherine R, Reck, Folkert, Richie, Daryl L, Rico, Alice, Sanderson, Mark R, Satasia, Shailesh, Sawyer, William S, Selvarajah, Jogitha, Shah, Nirav, Shanghavi, Kartik, Shu, Wei, Thompson, Katherine V, Traebert, Martin, Vala, Anand, Vala, Lakhan, Veselkov, Dennis A, Vo, Jason, Wang, Michael, Widya, Marcella, Williams, Sarah L, Xu, Yongjin, Yue, Qin, Zang, Richard, Zhou, Bo, Rivkin, Alexey
Published in Journal of medicinal chemistry (23.07.2020)
Published in Journal of medicinal chemistry (23.07.2020)
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Journal Article
Targeting IRAK3 for Degradation to Enhance IL-12 Pro-inflammatory Cytokine Production
Rowley, Ann, Brown, Brian S., Stofega, Mary, Hoh, Hana, Mathew, Rebecca, Marin, Violeta, Ding, Rong-Xian, McClure, Ryan A., Bittencourt, Fabiola M., Chen, Jun, Gururaja, Tarikere, Kinoshita, Taisei, Wang, Xueqing, Rivkin, Alexey, Woller, Kevin R.
Published in ACS chemical biology (17.06.2022)
Published in ACS chemical biology (17.06.2022)
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Journal Article
Discovery and Optimization of DNA Gyrase and Topoisomerase IV Inhibitors with Potent Activity against Fluoroquinolone-Resistant Gram-Positive Bacteria
Lapointe, Guillaume, Skepper, Colin K, Holder, Lauren M, Armstrong, Duncan, Bellamacina, Cornelia, Blais, Johanne, Bussiere, Dirksen, Bian, Jianwei, Cepura, Cody, Chan, Helen, Dean, Charles R, De Pascale, Gianfranco, Dhumale, Bhavesh, Fisher, L. Mark, Fulsunder, Mangesh, Kantariya, Bhavin, Kim, Julie, King, Sean, Kossy, Lauren, Kulkarni, Upendra, Lakshman, Jay, Leeds, Jennifer A, Ling, Xiaolan, Lvov, Anatoli, Ma, Sylvia, Malekar, Swapnil, McKenney, David, Mergo, Wosenu, Metzger, Louis, Mhaske, Keshav, Moser, Heinz E, Mostafavi, Mina, Namballa, Sunil, Noeske, Jonas, Osborne, Colin, Patel, Ashish, Patel, Darshit, Patel, Tushar, Piechon, Philippe, Polyakov, Valery, Prajapati, Krunal, Prosen, Katherine R, Reck, Folkert, Richie, Daryl L, Sanderson, Mark R, Satasia, Shailesh, Savani, Bhautik, Selvarajah, Jogitha, Sethuraman, Vijay, Shu, Wei, Tashiro, Kyuto, Thompson, Katherine V, Vaarla, Krishniah, Vala, Lakhan, Veselkov, Dennis A, Vo, Jason, Vora, Bhavesh, Wagner, Trixie, Wedel, Laura, Williams, Sarah L, Yendluri, Satya, Yue, Qin, Yifru, Aregahegn, Zhang, Yong, Rivkin, Alexey
Published in Journal of medicinal chemistry (13.05.2021)
Published in Journal of medicinal chemistry (13.05.2021)
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Journal Article
Evaluation of JAK3 Biology in Autoimmune Disease Using a Highly Selective, Irreversible JAK3 Inhibitor
Elwood, Fiona, Witter, David J, Piesvaux, Jennifer, Kraybill, Brian, Bays, Nathan, Alpert, Carla, Goldenblatt, Peter, Qu, Yujie, Ivanovska, Irena, Lee, Hyun-Hee, Chiu, Chi-Sung, Tang, Hao, Scott, Mark E, Deshmukh, Sujal V, Zielstorff, Mark, Byford, Alan, Chakravarthy, Kalyan, Dorosh, Lauren, Rivkin, Alexey, Klappenbach, Joel, Pan, Bo-Sheng, Kariv, Ilona, Dinsmore, Christopher, Slipetz, Deborah, Dandliker, Peter J
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
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