Hamamelitannin Analogues that Modulate Quorum Sensing as Potentiators of Antibiotics against Staphylococcus aureus
Vermote, Arno, Brackman, Gilles, Risseeuw, Martijn D. P., Vanhoutte, Bieke, Cos, Paul, Van Hecke, Kristof, Breyne, Koen, Meyer, Evelyne, Coenye, Tom, Van Calenbergh, Serge
Published in Angewandte Chemie International Edition (23.05.2016)
Published in Angewandte Chemie International Edition (23.05.2016)
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Journal Article
Identification of a new tert -leucinate class synthetic cannabinoid in powder and “spice-like” herbal incenses: methyl 2-[[1-(5-fluoropentyl)indole-3-carbonyl]amino]-3,3-dimethyl-butanoate (5F-MDMB-PICA)
Risseeuw, Martijn D.P, Blankaert, Peter, Coopman, Vera, Quekelberghe, Stijn Van, Calenbergh, Serge Van, Cordonnier, Jan
Published in Forensic science international (01.04.2017)
Published in Forensic science international (01.04.2017)
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Journal Article
Structure Guided Lead Generation toward Nonchiral M. tuberculosis Thymidylate Kinase Inhibitors
Song, Lijun, Merceron, Romain, Gracia, Begoña, Quintana, Ainhoa Lucía, Risseeuw, Martijn D. P, Hulpia, Fabian, Cos, Paul, Aínsa, José A, Munier-Lehmann, Hélène, Savvides, Savvas N, Van Calenbergh, Serge
Published in Journal of medicinal chemistry (12.04.2018)
Published in Journal of medicinal chemistry (12.04.2018)
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Journal Article
pH-Degradable Mannosylated Nanogels for Dendritic Cell Targeting
De Coen, Ruben, Vanparijs, Nane, Risseeuw, Martijn D. P, Lybaert, Lien, Louage, Benoit, De Koker, Stefaan, Kumar, Vimal, Grooten, Johan, Taylor, Leeanne, Ayres, Neil, Van Calenbergh, Serge, Nuhn, Lutz, De Geest, Bruno G
Published in Biomacromolecules (11.07.2016)
Published in Biomacromolecules (11.07.2016)
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Journal Article
Well-Defined Polymer-Paclitaxel Prodrugs by a Grafting-from-Drug Approach
Louage, Benoit, Nuhn, Lutz, Risseeuw, Martijn D. P., Vanparijs, Nane, De Coen, Ruben, Karalic, Izet, Van Calenbergh, Serge, De Geest, Bruno G.
Published in Angewandte Chemie International Edition (19.09.2016)
Published in Angewandte Chemie International Edition (19.09.2016)
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Journal Article
Synthetic Rhamnose Glycopolymer Cell-Surface Receptor for Endogenous Antibody Recruitment
De Coen, Ruben, Nuhn, Lutz, Perera, Chamani, Arista-Romero, Maria, Risseeuw, Martijn D. P, Freyn, Alec, Nachbagauer, Raffael, Albertazzi, Lorenzo, Van Calenbergh, Serge, Spiegel, David A, Peterson, Blake R, De Geest, Bruno G
Published in Biomacromolecules (10.02.2020)
Published in Biomacromolecules (10.02.2020)
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Journal Article
RUNX2 regulates leukemic cell metabolism and chemotaxis in high-risk T cell acute lymphoblastic leukemia
Matthijssens, Filip, Sharma, Nitesh D, Nysus, Monique, Nickl, Christian K, Kang, Huining, Perez, Dominique R, Lintermans, Beatrice, Van Loocke, Wouter, Roels, Juliette, Peirs, Sofie, Demoen, Lisa, Pieters, Tim, Reunes, Lindy, Lammens, Tim, De Moerloose, Barbara, Van Nieuwerburgh, Filip, Deforce, Dieter L, Cheung, Laurence C, Kotecha, Rishi S, Risseeuw, Martijn Dp, Van Calenbergh, Serge, Takarada, Takeshi, Yoneda, Yukio, van Delft, Frederik W, Lock, Richard B, Merkley, Seth D, Chigaev, Alexandre, Sklar, Larry A, Mullighan, Charles G, Loh, Mignon L, Winter, Stuart S, Hunger, Stephen P, Goossens, Steven, Castillo, Eliseo F, Ornatowski, Wojciech, Van Vlierberghe, Pieter, Matlawska-Wasowska, Ksenia
Published in The Journal of clinical investigation (15.03.2021)
Published in The Journal of clinical investigation (15.03.2021)
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Journal Article
1-(1-Arylethylpiperidin-4-yl)thymine Analogs as Antimycobacterial TMPK Inhibitors
Jian, Yanlin, Hulpia, Fabian, D P Risseeuw, Martijn, Forbes, He Eun, Caljon, Guy, Munier-Lehmann, Hélène, I M Boshoff, Helena, Van Calenbergh, Serge
Published in Molecules (Basel, Switzerland) (17.06.2020)
Published in Molecules (Basel, Switzerland) (17.06.2020)
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Journal Article
2-((3,5-Dinitrobenzyl)thio)quinazolinones: Potent Antimycobacterial Agents Activated by Deazaflavin (F-420)-Dependent Nitroreductase (Ddn)
Jian, Yanlin, Forbes, He Eun, Hulpia, Fabian, Risseeuw, Martijn D. P., Caljon, Guy, Munier-Lehmann, Helene, Boshoff, Helena I. M., Van Calenbergh, Serge
Published in Journal of medicinal chemistry (14.01.2021)
Published in Journal of medicinal chemistry (14.01.2021)
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Journal Article
Synthesis and Bioactivity of β‑Substituted Fosmidomycin Analogues Targeting 1‑Deoxy‑d‑xylulose-5-phosphate Reductoisomerase
Chofor, René, Sooriyaarachchi, Sanjeewani, Risseeuw, Martijn D. P, Bergfors, Terese, Pouyez, Jenny, Johny, Chinchu, Haymond, Amanda, Everaert, Annelien, Dowd, Cynthia S, Maes, Louis, Coenye, Tom, Alex, Alexander, Couch, Robin D, Jones, T. Alwyn, Wouters, Johan, Mowbray, Sherry L, Van Calenbergh, Serge
Published in Journal of medicinal chemistry (09.04.2015)
Published in Journal of medicinal chemistry (09.04.2015)
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Journal Article
Design, synthesis and biological evaluation of novel hamamelitannin analogues as potentiators for vancomycin in the treatment of biofilm related Staphylococcus aureus infections
Vermote, Arno, Brackman, Gilles, Risseeuw, Martijn D.P., Coenye, Tom, Van Calenbergh, Serge
Published in Bioorganic & medicinal chemistry (01.10.2016)
Published in Bioorganic & medicinal chemistry (01.10.2016)
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Journal Article
Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors
Song, Lijun, Merceron, Romain, Hulpia, Fabian, Lucía, Ainhoa, Gracia, Begoña, Jian, Yanlin, Risseeuw, Martijn D.P., Verstraelen, Toon, Cos, Paul, Aínsa, José A., Boshoff, Helena I., Munier-Lehmann, Hélène, Savvides, Savvas N., Van Calenbergh, Serge
Published in European journal of medicinal chemistry (05.12.2021)
Published in European journal of medicinal chemistry (05.12.2021)
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Journal Article
Identification and characterization of 4-chloromethamphetamine (4-CMA) in seized ecstacy — a risk to public health
Blanckaert, Peter, Vanquekelberghe, Stijn, Coopman, Vera, Risseeuw, Martijn D.P., Van Calenbergh, Serge, Cordonnier, Jan
Published in Forensic science international (01.07.2018)
Published in Forensic science international (01.07.2018)
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Journal Article
Synthesis toward Bivalent Ligands for the Dopamine D2 and Metabotropic Glutamate 5 Receptors
Qian, Mingcheng, Wouters, Elise, Dalton, James A. R, Risseeuw, Martijn D. P, Crans, René A. J, Stove, Christophe, Giraldo, Jesús, Van Craenenbroeck, Kathleen, Van Calenbergh, Serge
Published in Journal of medicinal chemistry (27.09.2018)
Published in Journal of medicinal chemistry (27.09.2018)
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Journal Article
Micellar Paclitaxel-Initiated RAFT Polymer Conjugates with Acid-Sensitive Behavior
Louage, Benoit, van Steenbergen, Mies J, Nuhn, Lutz, Risseeuw, Martijn D. P, Karalic, Izet, Winne, Johan, Van Calenbergh, Serge, Hennink, Wim E, De Geest, Bruno G
Published in ACS macro letters (21.03.2017)
Published in ACS macro letters (21.03.2017)
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Journal Article
Endeavors towards transformation of M. tuberculosis thymidylate kinase (MtbTMPK) inhibitors into potential antimycobacterial agents
Jian, Yanlin, Merceron, Romain, De Munck, Steven, Forbes, He Eun, Hulpia, Fabian, Risseeuw, Martijn D.P., Van Hecke, Kristof, Savvides, Savvas N., Munier-Lehmann, Hélène, Boshoff, Helena.I.M., Van Calenbergh, Serge
Published in European journal of medicinal chemistry (15.11.2020)
Published in European journal of medicinal chemistry (15.11.2020)
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Journal Article
Synthesis and structure activity relationships of cyanopyridone based anti-tuberculosis agents
Jian, Yanlin, Hulpia, Fabian, Risseeuw, Martijn D.P., Forbes, He Eun, Munier-Lehmann, Hélène, Caljon, Guy, Boshoff, Helena I.M., Van Calenbergh, Serge
Published in European journal of medicinal chemistry (01.09.2020)
Published in European journal of medicinal chemistry (01.09.2020)
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Journal Article
Design, Synthesis and Characterization of a New Series of Fluorescent Metabotropic Glutamate Receptor Type 5 Negative Allosteric Modulators
Fernández-Dueñas, Víctor, Qian, Mingcheng, Argerich, Josep, Amaral, Carolina, Risseeuw, Martijn D P, Van Calenbergh, Serge, Ciruela, Francisco
Published in Molecules (Basel, Switzerland) (27.03.2020)
Published in Molecules (Basel, Switzerland) (27.03.2020)
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Journal Article