Orexin receptor agonist Yan 7874 is a weak agonist of orexin/hypocretin receptors and shows orexin receptor-independent cytotoxicity
Turku, Ainoleena, Rinne, Maiju K, Boije Af Gennäs, Gustav, Xhaard, Henri, Lindholm, Dan, Kukkonen, Jyrki P
Published in PloS one (02.06.2017)
Published in PloS one (02.06.2017)
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Journal Article
Characterization of a putative orexin receptor in Ciona intestinalis sheds light on the evolution of the orexin/hypocretin system in chordates
Rinne, Maiju K, Urvas, Lauri, Mandrika, Ilona, Fridmanis, Dāvids, Riddy, Darren M, Langmead, Christopher J, Kukkonen, Jyrki P, Xhaard, Henri
Published in Scientific reports (02.04.2024)
Published in Scientific reports (02.04.2024)
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Journal Article
Cartography of rhodopsin-like G protein-coupled receptors across vertebrate genomes
Rinne, Maiju, Tanoli, Zia-Ur-Rehman, Khan, Asifullah, Xhaard, Henri
Published in Scientific reports (07.05.2019)
Published in Scientific reports (07.05.2019)
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Journal Article
Prolyl oligopeptidase inhibition by KYP-2407 increases alpha-synuclein fibril degradation in neuron-like cells
Rostami, Jinar, Jäntti, Maria, Cui, Hengjing, Rinne, Maiju K., Kukkonen, Jyrki P., Falk, Anna, Erlandsson, Anna, Myöhänen, Timo
Published in Biomedicine & pharmacotherapy (01.11.2020)
Published in Biomedicine & pharmacotherapy (01.11.2020)
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Corrigendum to “Prolyl oligopeptidase inhibition by KYP-2407 increases alpha-synuclein fibril degradation in neuron-like cells” [Biomed. Pharmacother. 131 (2020) 110788]
Rostami, Jinar, Jäntti, Maria, Cui, Hengjing, Rinne, Maiju K., Kukkonen, Jyrki P., Falk, Anna, Erlandsson, Anna, Myöhänen, Timo
Published in Biomedicine & pharmacotherapy (01.01.2021)
Published in Biomedicine & pharmacotherapy (01.01.2021)
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Journal Article
Pharmacological characterization of the orexin/hypocretin receptor agonist Nag 26
Rinne, Maiju K., Leino, Teppo O., Turku, Ainoleena, Turunen, Pauli M., Steynen, Yana, Xhaard, Henri, Wallén, Erik A.A., Kukkonen, Jyrki P.
Published in European journal of pharmacology (15.10.2018)
Published in European journal of pharmacology (15.10.2018)
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Journal Article
Mitoxantrone, pixantrone and mitoxantrone (2-hydroxyethyl)piperazine are toll-like receptor 4 antagonists, inhibit NF-κB activation, and decrease TNF-alpha secretion in primary microglia
Rinne, Maiju, Mätlik, Kert, Ahonen, Tiina, Vedovi, Fabio, Zappia, Giovanni, Moreira, Vânia M., Yli-Kauhaluoma, Jari, Leino, Sakari, Salminen, Outi, Kalso, Eija, Airavaara, Mikko, Xhaard, Henri
Published in European journal of pharmaceutical sciences (01.11.2020)
Published in European journal of pharmaceutical sciences (01.11.2020)
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Journal Article
Orexin/hypocretin receptor agonists: Pharmacological characterization of Nag 26 and discovery of novel agonist/potentiator structures based on the azulene scaffold
Kukkonen, Jyrki P, Rinne, Maiju K, Leino, Teppo O, Turku, Ainoleena, Turunen, Pauli M, Steynen, Yana, Xhaard, Henri, Wallen, Erik A
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
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Journal Article
Synthesis of 7β-hydroxy-8-ketone opioid derivatives with antagonist activity at mu- and delta-opioid receptors
Ahonen, Tiina J., Rinne, Maiju, Grutschreiber, Peter, Mätlik, Kert, Airavaara, Mikko, Schaarschmidt, Dieter, Lang, Heinrich, Reiss, David, Xhaard, Henri, Gaveriaux-Ruff, Claire, Yli-Kauhaluoma, Jari, Moreira, Vânia M.
Published in European journal of medicinal chemistry (10.05.2018)
Published in European journal of medicinal chemistry (10.05.2018)
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Journal Article
Synthesis of 7beta-hydroxy-8-ketone opioid derivatives with antagonist activity at mu- and delta-opioid receptors
Ahonen, Tiina, Rinne, Maiju, Grutschreiber, Peter, Matlik, Kert, Airavaara, Mikko, Schaarschmidt, Dieter, Lang, Heinrich, Reiss, David, Xhaard, Henri, Gaveriaux-Ruff, Claire, Yli-Kauhaluoma, Jari, Moreira, Vânia
Published in European journal of medicinal chemistry (2018)
Published in European journal of medicinal chemistry (2018)
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