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Chamberlain, Philip P, Lopez-Girona, Antonia, Miller, Karen, Carmel, Gilles, Pagarigan, Barbra, Chie-Leon, Barbara, Rychak, Emily, Corral, Laura G, Ren, Yan J, Wang, Maria, Riley, Mariko, Delker, Silvia L, Ito, Takumi, Ando, Hideki, Mori, Tomoyuki, Hirano, Yoshinori, Handa, Hiroshi, Hakoshima, Toshio, Daniel, Thomas O, Cathers, Brian E
Published in Nature structural & molecular biology (01.09.2014)
Published in Nature structural & molecular biology (01.09.2014)
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Novel oxysterols activate the Hedgehog pathway and induce osteogenesis
Stappenbeck, Frank, Xiao, Wei, Epperson, Matt, Riley, Mariko, Priest, Aaron, Huang, Danwen, Nguyen, KhanhLinh, Jung, Michael E., Scott Thies, R., Farouz, Francine
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
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A novel cereblon modulator recruits GSPT1 to the CRL4CRBN ubiquitin ligase
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Published in Nature (London) (22.06.2016)
Published in Nature (London) (22.06.2016)
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A novel cereblon modulator recruits GSPT1 to the CRL4(CRBN) ubiquitin ligase
Matyskiela, Mary E, Lu, Gang, Ito, Takumi, Pagarigan, Barbra, Lu, Chin-Chun, Miller, Karen, Fang, Wei, Wang, Nai-Yu, Nguyen, Derek, Houston, Jack, Carmel, Gilles, Tran, Tam, Riley, Mariko, Nosaka, Lyn'Al, Lander, Gabriel C, Gaidarova, Svetlana, Xu, Shuichan, Ruchelman, Alexander L, Handa, Hiroshi, Carmichael, James, Daniel, Thomas O, Cathers, Brian E, Lopez-Girona, Antonia, Chamberlain, Philip P
Published in Nature (London) (14.07.2016)
Published in Nature (London) (14.07.2016)
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A Cereblon Modulator (CC-220) with Improved Degradation of Ikaros and Aiolos
Matyskiela, Mary E, Zhang, Weihong, Man, Hon-Wah, Muller, George, Khambatta, Godrej, Baculi, Frans, Hickman, Matthew, LeBrun, Laurie, Pagarigan, Barbra, Carmel, Gilles, Lu, Chin-Chun, Lu, Gang, Riley, Mariko, Satoh, Yoshitaka, Schafer, Peter, Daniel, Thomas O, Carmichael, James, Cathers, Brian E, Chamberlain, Philip P
Published in Journal of medicinal chemistry (25.01.2018)
Published in Journal of medicinal chemistry (25.01.2018)
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SALL4 mediates teratogenicity as a thalidomide-dependent cereblon substrate
Matyskiela, Mary E, Couto, Suzana, Zheng, Xinde, Lu, Gang, Hui, Julia, Stamp, Katie, Drew, Clifton, Ren, Yan, Wang, Maria, Carpenter, Aaron, Lee, Chung-Wein, Clayton, Thomas, Fang, Wei, Lu, Chin-Chun, Riley, Mariko, Abdubek, Polat, Blease, Kate, Hartke, James, Kumar, Gondi, Vessey, Rupert, Rolfe, Mark, Hamann, Lawrence G, Chamberlain, Philip P
Published in Nature chemical biology (01.10.2018)
Published in Nature chemical biology (01.10.2018)
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Abstract SY37-02: Ligand-directed degradation of GSPT1 by a novel cereblon modulator drives potent antitumor effects
Matyskiela, Mary, Lu, Gang, Ito, Takumi, Pagarigan, Barbra, Lu, Chin-Chu, Miller, Karen, Fang, Wei, Wang, Nai-Yu, Nguyen, Derek, Houston, Jack, Carmel, Gilles, Tran, Tam, Riley, Mariko, Nosaka, Lyn'Al, Lander, Gabriel, Gaidarova, Svetlana, Xu, Shuichan, Ruchelman, Alexander, Handa, Hiroshi, Carmichale, James, Daniel, Thomas O., Cathers, Brian E., Lopez-Girona, Antonia, Chamberlain, Philip
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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A novel cereblon modulator recruits GSPT1 to the [CRL4.sup.CRBN] ubiquitin ligase
Matyskiela, Mary E, Lu, Gang, Ito, Takumi, Pagarigan, Barbra, Lu, Chin-Chun, Miller, Karen, Fang, Wei, Wang, Nai-Yu, Nguyen, Derek, Houston, Jack, Carmel, Gilles, Tran, Tam, Riley, Mariko, Nosaka, Lyn'Al, Lander, Gabriel C, Gaidarova, Svetlana, Xu, Shuichan, Ruchelman, Alexander L, Handa, Hiroshi, Carmichael, James, Daniel, Thomas O, Cathers, Brian E, Lopez-Girona, Antonia, chamberlain, Philip P
Published in Nature (London) (14.07.2016)
Published in Nature (London) (14.07.2016)
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A novel cereblon modulator recruits GSPT1 to the CRL4 ^sup CRBN^ ubiquitin ligase
Matyskiela, Mary E, Lu, Gang, Ito, Takumi, Pagarigan, Barbra, Lu, Chin-Chun, Miller, Karen, Fang, Wei, Wang, Nai-Yu, Nguyen, Derek, Houston, Jack, Carmel, Gilles, Tran, Tam, Riley, Mariko, Nosaka, Lyn'Al, Lander, Gabriel C, Gaidarova, Svetlana, Xu, Shuichan, Ruchelman, Alexander L, Handa, Hiroshi, Carmichael, James, Daniel, Thomas O, Cathers, Brian E, Lopez-Girona, Antonia, Chamberlain, Philip P
Published in Nature (London) (14.07.2016)
Published in Nature (London) (14.07.2016)
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Developing targets for drug discovery using genome-wide gene trapping and ultra-sensitive beta-lactamase reporters
Liyanage, M, Zamiara, E M, Mandurrago, B, Riley, M, Sanders, P, Welchlin, H L, Xanthopoulos, K G
Published in Proceedings of the Western Pharmacology Society (1999)
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Published in Proceedings of the Western Pharmacology Society (1999)
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