A Molecular-Wide and Electron Density-Based Approach in Exploring Chemical Reactivity and Explicit Dimethyl Sulfoxide (DMSO) Solvent Molecule Effects in the Proline Catalyzed Aldol Reaction
Cukrowski, Ignacy, Dhimba, George, Riley, Darren L
Published in Molecules (Basel, Switzerland) (31.01.2022)
Published in Molecules (Basel, Switzerland) (31.01.2022)
Get full text
Journal Article
New syntheses of (±)-tashiromine and (±)-epitashiromine via enaminone intermediates
Riley, Darren L, Michael, Joseph P, de Koning, Charles B
Published in Beilstein journal of organic chemistry (02.12.2016)
Published in Beilstein journal of organic chemistry (02.12.2016)
Get full text
Journal Article
A reaction energy profile and fragment attributed molecular system energy change (FAMSEC)-based protocol designed to uncover reaction mechanisms: a case study of the proline-catalysed aldol reaction
Cukrowski, Ignacy, Dhimba, George, Riley, Darren L
Published in Physical chemistry chemical physics : PCCP (14.08.2019)
Published in Physical chemistry chemical physics : PCCP (14.08.2019)
Get full text
Journal Article
Discovery of Novel Acetylcholinesterase Inhibitors by Virtual Screening, In Vitro Screening, and Molecular Dynamics Simulations
van der Westhuizen, C. Johan, Stander, André, Riley, Darren L, Panayides, Jenny-Lee
Published in Journal of chemical information and modeling (28.03.2022)
Published in Journal of chemical information and modeling (28.03.2022)
Get full text
Journal Article
Targeting Alzheimer's disease by investigating previously unexplored chemical space surrounding the cholinesterase inhibitor donepezil
van Greunen, Divan G., Cordier, Werner, Nell, Margo, van der Westhuyzen, Chris, Steenkamp, Vanessa, Panayides, Jenny-Lee, Riley, Darren L.
Published in European journal of medicinal chemistry (15.02.2017)
Published in European journal of medicinal chemistry (15.02.2017)
Get full text
Journal Article
Novel N-benzylpiperidine carboxamide derivatives as potential cholinesterase inhibitors for the treatment of Alzheimer's disease
van Greunen, Divan G., Johan van der Westhuizen, C., Cordier, Werner, Nell, Margo, Stander, Andre, Steenkamp, Vanessa, Panayides, Jenny-Lee, Riley, Darren L.
Published in European journal of medicinal chemistry (01.10.2019)
Published in European journal of medicinal chemistry (01.10.2019)
Get full text
Journal Article
Anticancer Agents from Diverse Natural Sources
Khazir, Jabeena, Riley, Darren L., Pilcher, Lynne A., De-Maayer, Pieter, Mir, Bilal Ahmad
Published in Natural product communications (01.11.2014)
Published in Natural product communications (01.11.2014)
Get full text
Journal Article
The in silico and in vitro analysis of donepezil derivatives for Anopheles acetylcholinesterase inhibition
Rants'o, Thankhoe A, van Greunen, Divan G, van der Westhuizen, C. Johan, Riley, Darren L, Panayides, Jenny-Lee, Koekemoer, Lizette L, van Zyl, Robyn L
Published in PloS one (09.11.2022)
Published in PloS one (09.11.2022)
Get full text
Journal Article
An Improved Process for the Preparation of Tenofovir Disoproxil Fumarate
Riley, Darren L, Walwyn, David R, Edlin, Chris D
Published in Organic process research & development (15.04.2016)
Published in Organic process research & development (15.04.2016)
Get full text
Journal Article
Design, synthesis and anticancer activity of Michael-type thiol adducts of α-santonin analogue with exocyclic methylene
Khazir, Jabeena, Riley, Darren L., Chashoo, Gousia, Mir, Bilal Ahmad, Liles, David, Islam, Md. Ataul, Singh, Shashank K., Vishwakarma, Ram A., Pilcher, Lynne A.
Published in European journal of medicinal chemistry (28.08.2015)
Published in European journal of medicinal chemistry (28.08.2015)
Get full text
Journal Article
Assessing a sustainable manufacturing route to lapatinib
Stark, Roderick T, Pye, Dominic R, Chen, Wenyi, Newton, Oliver J, Deadman, Benjamin J, Miller, Philip W, Panayides, Jenny-Lee, Riley, Darren L, Hellgardt, Klaus, Hii, King Kuok (Mimi)
Published in Reaction chemistry & engineering (25.10.2022)
Published in Reaction chemistry & engineering (25.10.2022)
Get full text
Journal Article
Design and synthesis of ring C opened analogues of α-santonin as potential anticancer agents
Khazir, Jabeena, Mir, Bilal Ahmad, Pilcher, Lynne A., Riley, Darren L., Chashoo, Gousia, Islam, Md. Ataul, Saxena, Ajit K., Kumar, H. M. Sampath
Published in Medicinal chemistry research (01.09.2016)
Published in Medicinal chemistry research (01.09.2016)
Get full text
Journal Article
A concise, rapid and high yielding flow synthesis of aryldiazonium tetrafluoroborates
Scholtz, Chantal, Riley, Darren L.
Published in ARKIVOC free online journal of organic chemistry (01.01.2020)
Published in ARKIVOC free online journal of organic chemistry (01.01.2020)
Get full text
Journal Article