The BET Family of Proteins Targets Moloney Murine Leukemia Virus Integration near Transcription Start Sites
De Rijck, Jan, de Kogel, Christine, Demeulemeester, Jonas, Vets, Sofie, El Ashkar, Sara, Malani, Nirav, Bushman, Frederic D., Landuyt, Bart, Husson, Steven J., Busschots, Katrien, Gijsbers, Rik, Debyser, Zeger
Published in Cell reports (Cambridge) (01.11.2013)
Published in Cell reports (Cambridge) (01.11.2013)
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LEDGF/p75-independent HIV-1 replication demonstrates a role for HRP-2 and remains sensitive to inhibition by LEDGINs
Schrijvers, Rik, De Rijck, Jan, Demeulemeester, Jonas, Adachi, Noritaka, Vets, Sofie, Ronen, Keshet, Christ, Frauke, Bushman, Frederic D, Debyser, Zeger, Gijsbers, Rik
Published in PLoS pathogens (01.03.2012)
Published in PLoS pathogens (01.03.2012)
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Correction: LEDGF/p75-Independent HIV-1 Replication Demonstrates a Role for HRP-2 and Remains Sensitive to Inhibition by LEDGINs
Schrijvers, Rik, Rijck, Jan De, Demeulemeester, Jonas, Adachi, Noritaka, Vets, Sofie, Ronen, Keshet, Christ, Frauke, Bushman, Frederic D, Debyser, Zeger, Gijsbers, Rik
Published in PLoS pathogens (01.09.2020)
Published in PLoS pathogens (01.09.2020)
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Virus evolution reveals an exclusive role for LEDGF/p75 in chromosomal tethering of HIV
Hombrouck, Anneleen, De Rijck, Jan, Hendrix, Jelle, Vandekerckhove, Linos, Voet, Arnout, De Maeyer, Marc, Witvrouw, Myriam, Engelborghs, Yves, Christ, Frauke, Gijsbers, Rik, Debyser, Zeger
Published in PLoS pathogens (01.03.2007)
Published in PLoS pathogens (01.03.2007)
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A ubiquitous disordered protein interaction module orchestrates transcription elongation
Cermakova, Katerina, Demeulemeester, Jonas, Lux, Vanda, Nedomova, Monika, Goldman, Seth R, Smith, Eric A, Srb, Pavel, Hexnerova, Rozalie, Fabry, Milan, Madlikova, Marcela, Horejsi, Magdalena, De Rijck, Jan, Debyser, Zeger, Adelman, Karen, Hodges, H Courtney, Veverka, Vaclav
Published in Science (American Association for the Advancement of Science) (26.11.2021)
Published in Science (American Association for the Advancement of Science) (26.11.2021)
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HIV-1 Integrase Variants Retarget Viral Integration and Are Associated with Disease Progression in a Chronic Infection Cohort
Demeulemeester, Jonas, Vets, Sofie, Schrijvers, Rik, Madlala, Paradise, De Maeyer, Marc, De Rijck, Jan, Ndung’u, Thumbi, Debyser, Zeger, Gijsbers, Rik
Published in Cell host & microbe (12.11.2014)
Published in Cell host & microbe (12.11.2014)
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Multiple cellular proteins interact with LEDGF/p75 through a conserved unstructured consensus motif
Tesina, Petr, Čermáková, Kateřina, Hořejší, Magdalena, Procházková, Kateřina, Fábry, Milan, Sharma, Subhalakshmi, Christ, Frauke, Demeulemeester, Jonas, Debyser, Zeger, Rijck, Jan De, Veverka, Václav, Řezáčová, Pavlína
Published in Nature communications (06.08.2015)
Published in Nature communications (06.08.2015)
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LEDGINs inhibit late stage HIV-1 replication by modulating integrase multimerization in the virions
Desimmie, Belete Ayele, Schrijvers, Rik, Demeulemeester, Jonas, Borrenberghs, Doortje, Weydert, Caroline, Thys, Wannes, Vets, Sofie, Van Remoortel, Barbara, Hofkens, Johan, De Rijck, Jan, Hendrix, Jelle, Bannert, Norbert, Gijsbers, Rik, Christ, Frauke, Debyser, Zeger
Published in Retrovirology (30.05.2013)
Published in Retrovirology (30.05.2013)
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Correction: Y-box-binding protein 1 supports the early and late steps of HIV replication
Weydert, Caroline, van Heertum, Bart, Dirix, Lieve, De Houwer, Stéphanie, De Wit, Flore, Mast, Jan, Husson, Steven J, Busschots, Katrien, König, Renate, Gijsbers, Rik, De Rijck, Jan, Debyser, Zeger
Published in PloS one (29.10.2020)
Published in PloS one (29.10.2020)
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Targeting Virus-host Interactions of HIV Replication
Weydert, Caroline, De Rijck, Jan, Christ, Frauke, Debyser, Zeger
Published in Current topics in medicinal chemistry (01.01.2016)
Published in Current topics in medicinal chemistry (01.01.2016)
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Journal Article
Validation and structural characterization of the LEDGF/p75-MLL interface as a new target for the treatment of MLL-dependent leukemia
Cermáková, Kateřina, Tesina, Petr, Demeulemeester, Jonas, El Ashkar, Sara, Méreau, Hélène, Schwaller, Juerg, Rezáčová, Pavlína, Veverka, Vaclav, De Rijck, Jan
Published in Cancer research (Chicago, Ill.) (15.09.2014)
Published in Cancer research (Chicago, Ill.) (15.09.2014)
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Journal Article
Overexpression of the Lens Epithelium-Derived Growth Factor/p75 Integrase Binding Domain Inhibits Human Immunodeficiency Virus Replication
DE RIJCK, Jan, VANDEKERCKHOVE, Linos, GIJSBERS, Rik, HOMBROUCK, Anneleen, HENDRIX, Jelle, VERCAMMEN, Jo, ENGELBORGHS, Yves, CHRIST, Frauke, DEBYSER, Zeger
Published in Journal of Virology (01.12.2006)
Published in Journal of Virology (01.12.2006)
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Journal Article
Y-box-binding protein 1 supports the early and late steps of HIV replication
Weydert, Caroline, van Heertum, Bart, Dirix, Lieve, De Houwer, Stéphanie, De Wit, Flore, Mast, Jan, Husson, Steven J, Busschots, Katrien, König, Renate, Gijsbers, Rik, De Rijck, Jan, Debyser, Zeger
Published in PloS one (11.07.2018)
Published in PloS one (11.07.2018)
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Transient and Stable Knockdown of the Integrase Cofactor LEDGF/p75 Reveals Its Role in the Replication Cycle of Human Immunodeficiency Virus
VANDEKERCKHOVE, Linos, CHRIST, Frauke, VAN MAELE, Bénédicte, DE RIJCK, Jan, GIJSBERS, Rik, VAN DEN HAUTE, Chris, WITVROUW, Myriam, DEBYSER, Zeger
Published in Journal of Virology (01.02.2006)
Published in Journal of Virology (01.02.2006)
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Journal Article
Retroviral integration: Site matters
Demeulemeester, Jonas, De Rijck, Jan, Gijsbers, Rik, Debyser, Zeger
Published in BioEssays (01.11.2015)
Published in BioEssays (01.11.2015)
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Journal Article
HRP-2 determines HIV-1 integration site selection in LEDGF/p75 depleted cells
Schrijvers, Rik, Vets, Sofie, De Rijck, Jan, Malani, Nirav, Bushman, Frederic D, Debyser, Zeger, Gijsbers, Rik
Published in Retrovirology (09.10.2012)
Published in Retrovirology (09.10.2012)
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Toward the Discovery of Novel Anti-HIV Drugs. Second-Generation Inhibitors of the Cellular ATPase DDX3 with Improved Anti-HIV Activity: Synthesis, Structure-Activity Relationship Analysis, Cytotoxicity Studies, and Target Validation
Maga, Giovanni, Falchi, Federico, Radi, Marco, Botta, Lorenzo, Casaluce, Gianni, Bernardini, Martina, Irannejad, Hamid, Manetti, Fabrizio, Garbelli, Anna, Samuele, Alberta, Zanoli, Samantha, Esté, José A., Gonzalez, Emmanuel, Zucca, Elisa, Paolucci, Stefania, Baldanti, Fausto, De Rijck, Jan, Debyser, Zeger, Botta, Maurizio
Published in ChemMedChem (01.08.2011)
Published in ChemMedChem (01.08.2011)
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Correction to: HIV-1 IN/Pol recruits LEDGF/p75 into viral particles
Desimmie, Belete Ayele, Weydert, Caroline, Schrijvers, Rik, Vets, Sofie, Demeulemeester, Jonas, Proost, Paul, Paron, Igor, De Rijck, Jan, Mast, Jan, Bannert, Norbert, Gijsbers, Rik, Christ, Frauke, Debyser, Zeger
Published in Retrovirology (29.07.2020)
Published in Retrovirology (29.07.2020)
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Journal Article
Lens Epithelium-derived Growth Factor/p75 Interacts with the Transposase-derived DDE Domain of PogZ
Bartholomeeusen, Koen, Christ, Frauke, Hendrix, Jelle, Rain, Jean-Christophe, Emiliani, Stéphane, Benarous, Richard, Debyser, Zeger, Gijsbers, Rik, De Rijck, Jan
Published in The Journal of biological chemistry (24.04.2009)
Published in The Journal of biological chemistry (24.04.2009)
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Journal Article
BET-Independent Murine Leukemia Virus Integration Is Retargeted In Vivo and Selects Distinct Genomic Elements for Lymphomagenesis
Nombela, Ivan, Michiels, Martine, Van Looveren, Dominique, Marcelis, Lukas, el Ashkar, Sara, Van Belle, Siska, Bruggemans, Anne, Tousseyn, Thomas, Schwaller, Jürg, Christ, Frauke, Gijsbers, Rik, De Rijck, Jan, Debyser, Zeger
Published in Microbiology spectrum (31.08.2022)
Published in Microbiology spectrum (31.08.2022)
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