Targeting Mitochondrial Structure Sensitizes Acute Myeloid Leukemia to Venetoclax Treatment
Chen, Xufeng, Glytsou, Christina, Zhou, Hua, Narang, Sonali, Reyna, Denis E, Lopez, Andrea, Sakellaropoulos, Theodore, Gong, Yixiao, Kloetgen, Andreas, Yap, Yoon Sing, Wang, Eric, Gavathiotis, Evripidis, Tsirigos, Aristotelis, Tibes, Raoul, Aifantis, Iannis
Published in Cancer discovery (01.07.2019)
Published in Cancer discovery (01.07.2019)
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Co-targeting of BAX and BCL-XL proteins broadly overcomes resistance to apoptosis in cancer
Lopez, Andrea, Reyna, Denis E, Gitego, Nadege, Kopp, Felix, Zhou, Hua, Miranda-Roman, Miguel A, Nordstrøm, Lars Ulrik, Narayanagari, Swathi-Rao, Chi, Ping, Vilar, Eduardo, Tsirigos, Aristotelis, Gavathiotis, Evripidis
Published in Nature communications (07.03.2022)
Published in Nature communications (07.03.2022)
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Eltrombopag directly inhibits BAX and prevents cell death
Spitz, Adam Z, Zacharioudakis, Emmanouil, Reyna, Denis E, Garner, Thomas P, Gavathiotis, Evripidis
Published in Nature communications (18.02.2021)
Published in Nature communications (18.02.2021)
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An interconnected hierarchical model of cell death regulation by the BCL-2 family
Chen, Hui-Chen, Kanai, Masayuki, Inoue-Yamauchi, Akane, Tu, Ho-Chou, Huang, Yafen, Ren, Decheng, Kim, Hyungjin, Takeda, Shugaku, Reyna, Denis E, Chan, Po M, Ganesan, Yogesh Tengarai, Liao, Chung-Ping, Gavathiotis, Evripidis, Hsieh, James J, Cheng, Emily H
Published in Nature cell biology (01.10.2015)
Published in Nature cell biology (01.10.2015)
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BH3-Triggered Structural Reorganization Drives the Activation of Proapoptotic BAX
Gavathiotis, Evripidis, Reyna, Denis E., Davis, Marguerite L., Bird, Gregory H., Walensky, Loren D.
Published in Molecular cell (12.11.2010)
Published in Molecular cell (12.11.2010)
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An Autoinhibited Dimeric Form of BAX Regulates the BAX Activation Pathway
Garner, Thomas P., Reyna, Denis E., Priyadarshi, Amit, Chen, Hui-Chen, Li, Sheng, Wu, Yang, Ganesan, Yogesh Tengarai, Malashkevich, Vladimir N., Cheng, Emily H., Gavathiotis, Evripidis
Published in Molecular cell (04.08.2016)
Published in Molecular cell (04.08.2016)
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Bax regulates primary necrosis through mitochondrial dynamics
Whelan, Russell S, Konstantinidis, Klitos, Wei, An-Chi, Chen, Yun, Reyna, Denis E, Jha, Saurabh, Yang, Ying, Calvert, John W, Lindsten, Tullia, Thompson, Craig B, Crow, Michael T, Gavathiotis, Evripidis, Dorn, Gerald W. II, O'Rourke, Brian, Kitsis, Richard N
Published in Proceedings of the National Academy of Sciences - PNAS (24.04.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (24.04.2012)
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An Autoinhibited Dimeric Form of BAX Regulates the BAX Activation Pathway
Garner, Thomas P., Reyna, Denis E., Priyadarshi, Amit, Chen, Hui-Chen, Li, Sheng, Wu, Yang, Ganesan, Yogesh Tengarai, Malashkevich, Vladimir N., Cheng, Emily H., Gavathiotis, Evripidis
Published in Molecular cell (20.10.2016)
Published in Molecular cell (20.10.2016)
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Small-molecule allosteric inhibitors of BAX
Garner, Thomas P, Amgalan, Dulguun, Reyna, Denis E, Li, Sheng, Kitsis, Richard N, Gavathiotis, Evripidis
Published in Nature chemical biology (01.04.2019)
Published in Nature chemical biology (01.04.2019)
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Progress in targeting the BCL-2 family of proteins
Garner, Thomas P, Lopez, Andrea, Reyna, Denis E, Spitz, Adam Z, Gavathiotis, Evripidis
Published in Current opinion in chemical biology (01.08.2017)
Published in Current opinion in chemical biology (01.08.2017)
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Direct Activation of BAX by BTSA1 Overcomes Apoptosis Resistance in Acute Myeloid Leukemia
Reyna, Denis E., Garner, Thomas P., Lopez, Andrea, Kopp, Felix, Choudhary, Gaurav S., Sridharan, Ashwin, Narayanagari, Swathi-Rao, Mitchell, Kelly, Dong, Baoxia, Bartholdy, Boris A., Walensky, Loren D., Verma, Amit, Steidl, Ulrich, Gavathiotis, Evripidis
Published in Cancer cell (09.10.2017)
Published in Cancer cell (09.10.2017)
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Apoptosis signaling molecules as treatment targets in head and neck squamous cell carcinoma
Ow, Thomas J, Thomas, Carlos, Fulcher, Cory D, Chen, Jianhong, López, Andrea, Reyna, Denis E, Prystowsky, Michael B, Smith, Richard V, Schiff, Bradley A, Rosenblatt, Gregory, Belbin, Thomas J, Harris, Thomas M, Childs, Geoffrey C, Kawachi, Nicole, Schlecht, Nicolas F, Gavathiotis, Evripidis
Published in The Laryngoscope (01.11.2020)
Published in The Laryngoscope (01.11.2020)
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Optimal targeting of BCL-family proteins in head and neck squamous cell carcinoma requires inhibition of both BCL-xL and MCL-1
Ow, Thomas J, Fulcher, Cory D, Thomas, Carlos, Broin, Pilib Ó, López, Andrea, Reyna, Denis E, Smith, Richard V, Sarta, Catherine, Prystowsky, Michael B, Schlecht, Nicolas F, Schiff, Bradley A, Rosenblatt, Gregory, Belbin, Thomas J, Harris, Thomas M, Childs, Geoffrey C, Kawachi, Nicole, Guha, Chandan, Gavathiotis, Evripidis
Published in Oncotarget (11.01.2019)
Published in Oncotarget (11.01.2019)
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In Response to Regarding: Apoptosis Signaling Molecules as Treatment Targets in Head and Neck Squamous Carcinoma
Ow, Thomas J, Thomas, Carlos, Fulcher, Cory D, Chen, Jianhong, López, Andrea, Reyna, Denis E, Prystowsky, Michael B, Smith, Richard V, Schiff, Bradley A, Rosenblatt, Gregory, Belbin, Thomas J, Harris, Thomas M, Childs, Geoffrey C, Kawachi, Nicole, Schlecht, Nicolas F, Gavathiotis, Evripidis
Published in The Laryngoscope (01.08.2020)
Published in The Laryngoscope (01.08.2020)
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BH3-Triggered Structural Reorganization Drives the Activation of Pro-apoptotic BAX
Gavathiotis, Evripidis, Reyna, Denis E., Davis, Marguerite L., Bird, Gregory H., Walensky, Loren D.
Published in Molecular cell (12.11.2010)
Published in Molecular cell (12.11.2010)
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