A peripherally acting alpha-2 adrenoceptor antagonist: L-659,066
CLINESCHMIDT, B. V, PETTIBONE, D. J, LOTTI, V. J, HUCKER, H. B, SWEENEY, B. M, REISS, D. R, LIS, E. V, HUFF, J. R, VACCA, J
Published in The Journal of pharmacology and experimental therapeutics (01.04.1988)
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Published in The Journal of pharmacology and experimental therapeutics (01.04.1988)
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Characterization of 5-hydroxytryptamine receptors in rat stomach fundus
CLINESCHMIDT, B. V, REISS, D. R, PETTIBONE, D. J, ROBINSON, J. L
Published in The Journal of pharmacology and experimental therapeutics (01.12.1985)
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Published in The Journal of pharmacology and experimental therapeutics (01.12.1985)
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Identification of an orally active, nonpeptidyl oxytocin antagonist
PETTIBONE, D. J, CLINESCHMIDT, B. V, HALUSKA, G. J, NOVY, M. J, LOWENSOHN, R. I, KISHEL, M. T, LIS, E. V, REISS, D. R, WOYDEN, C. J, EVANS, B. E, FREIDINGER, R. M, VEBER, D. F, COOK, M. J
Published in The Journal of pharmacology and experimental therapeutics (01.01.1993)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.1993)
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Nonpeptide oxytocin antagonists: Analogs of L-371,257 with improved potency
Williams, Peter D., Bock, Mark G., Evans, Ben E., Freidinger, Roger M., Gallicchio, Steven N., Guidotti, Maribeth T., Jacobson, Marlene A., Kuo, Michelle S., Levy, Michelle R., Lis, Edward V., Michelson, Stuart R., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Salvatore, Christopher, Stauffer, Kenneth J., Woyden, Carla J.
Published in Bioorganic & medicinal chemistry letters (03.05.1999)
Published in Bioorganic & medicinal chemistry letters (03.05.1999)
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Journal Article
In vitro pharmacological profile of a novel structural class of oxytocin antagonists
PETTIBONE, D. J, CLINESCHMIDT, B. V, WILLIAMS, P. D, LOWENSOHN, R. I, LIS, E. V, REISS, D. R, TOTARO, J. A, WOYDEN, C. J, BOCK, M. G, FREIDINGER, R. M, TUNG, R. D, VEBER, D. F
Published in The Journal of pharmacology and experimental therapeutics (01.01.1991)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.1991)
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Strong convergence of multivariate point processes of exceedances
KAUFMANN, E, REISS, R.-D
Published in Annals of the Institute of Statistical Mathematics (01.09.1993)
Published in Annals of the Institute of Statistical Mathematics (01.09.1993)
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Nonpeptide oxytocin antagonists: Potent, orally bioavailable analogs of L-371,257 containing A 1- R-(pyridyl)ethyl ether terminus
Kuo, Michelle S., Bock, Mark G., Freidinger, Roger M., Guidotti, Maribeth T., Lis, Edward V., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Williams, Peter D., Woyden, Carla J.
Published in Bioorganic & medicinal chemistry letters (03.11.1998)
Published in Bioorganic & medicinal chemistry letters (03.11.1998)
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Journal Article
Antagonism of oxytocin in rats and pregnant rhesus monkeys by the novel cyclic hexapeptides, L-366,682 and L-366,948
CLINESCHMIDT, B. V, PETTIBONE, D. J, FREIDINGER, R. M, VEBER, D. F, WILLIAMS, P. D, REISS, D. R, LIS, E. V, HALUSKA, G. J, NOVY, M. J, COOK, M. J, CUKIERSKI, M. A, KAUFMAN, M. J, BOCK, M. G
Published in The Journal of pharmacology and experimental therapeutics (01.03.1991)
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Published in The Journal of pharmacology and experimental therapeutics (01.03.1991)
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