Thrombin active site inhibitors: chemical synthesis, in vitro and in vivo pharmacological profile of a novel and selective agent BMS-189090 and analogues
Das, Jagabandhu, Kimball, S.David, Reid, Joyce A., Wang, Tammy C., Lau, Wan F., Roberts, Daniel G.M., Seiler, Steven M., Schumacher, William A., Ogletree, Martin L.
Published in Bioorganic & medicinal chemistry letters (07.01.2002)
Published in Bioorganic & medicinal chemistry letters (07.01.2002)
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Molecular design and structure–Activity relationships leading to the potent, selective, and orally active thrombin active site inhibitor BMS-189664
Das, Jagabandhu, Kimball, S.David, Hall, Steven E., Han, Wen-Ching, Iwanowicz, Edwin, Lin, James, Moquin, Robert V., Reid, Joyce A., Sack, John S., Malley, Mary F., Chang, Chiehying Y., Chong, Saeho, Wang-Iverson, David B., Roberts, Daniel G.M., Seiler, Steven M., Schumacher, William A., Ogletree, Martin L.
Published in Bioorganic & medicinal chemistry letters (07.01.2002)
Published in Bioorganic & medicinal chemistry letters (07.01.2002)
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7-Oxabicyclo[2.2.1]heptyl carboxylic acids as thromboxane A2 antagonists: aza .omega.-chain analogs
Nakane, Masami, Reid, Joyce A, Han, Wen Ching, Das, Jagabandhu, Vu Chi Truc, Vu Chi, Haslanger, Martin F, Garber, Dianne, Harris, Don N, Hedberg, Anders, Ogletree, Martin L, Hall, Steven E
Published in Journal of medicinal chemistry (01.09.1990)
Published in Journal of medicinal chemistry (01.09.1990)
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9,11-Epoxy-9-homoprosta-5-enoic acid analogs as thromboxane A2 receptor antagonists
Das, Jagabandhu, Hall, Steven E, Nakane, Masami, Haslanger, Martin F, Reid, Joyce A, Garber, Dianne, Vu Chi Truc, Harris, Don N, Hedberg, Anders, Ogletree, Martin L
Published in Journal of medicinal chemistry (01.06.1990)
Published in Journal of medicinal chemistry (01.06.1990)
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Angiotensin-converting enzyme inhibitors: importance of the amide carbonyl of mercaptoacyl amino acids for hydrogen bonding to the enzyme
Condon, Michael E, Petrillo, Edward W, Ryono, Denis E, Reid, Joyce A, Neubeck, Richard, Puar, Mohindar, Heikes, James E, Sabo, Emily F, Losee, Kathryn A
Published in Journal of medicinal chemistry (01.03.1982)
Published in Journal of medicinal chemistry (01.03.1982)
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Dual metalloprotease inhibitors. IV. Utilization of thiazepines and thiazines as constrained peptidomimetic surrogates in mercaptoacyl dipeptides
Das, Jagabandhu, Robl, Jeffrey A., Reid, Joyce A., Sun, Chong-Qing, Misra, Raj N., Brown, Baerbel R., Ryono, Denis E., Asaad, Magdi M., Bird, J.Eileen, Trippodo, Nick C., Petrillo, Edward W., Karanewsky, Donald S.
Published in Bioorganic & medicinal chemistry letters (22.09.1994)
Published in Bioorganic & medicinal chemistry letters (22.09.1994)
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NOVEL METHODS FOR SYNTHESES OF SUBSTITUTED OXAZOLES BY CYCLIZATION OF VINYL BROMIDES
DAS, J, REID, JA, KRONENTHAL, DR, SINGH, J, PANSEGRAU, PD, MUELLER, RH
Published in Tetrahedron letters (15.12.1992)
Published in Tetrahedron letters (15.12.1992)
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Thoromboxane A2/endoperoxide receptor antagonists: 1,3-Dioxane and 1,3-dioxolane analogs
Das, Jagabandhu, Reid, Joyce A., Harris, Don N., Goldenberg, Harold, Michel, Inge M., Monshizadegan, Hossain, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (01.06.1993)
Published in Bioorganic & medicinal chemistry letters (01.06.1993)
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Thoromboxane A 2/endoperoxide receptor antagonists: 1,3-Dioxane and 1,3-dioxolane analogs
Das, Jagabandhu, Reid, Joyce A., Harris, Don N., Goldenberg, Harold, Michel, Inge M., Monshizadegan, Hossain, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (1993)
Published in Bioorganic & medicinal chemistry letters (1993)
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1,4-substituted indoles: a potent and selective class of angiostensin II receptor antagonists
Poss, Michael A., Gu, Zhengxiang, Ryono, Denis E., Reid, Joyce A., Sieber-McMaster, Ellen, Spitzmiller, Ervin R., Dejneka, Tamara, Dickinson, Kenneth E.J., Williams, Sharon B., Moreland, Suzanne, Delaney, Carol L., Bird, J.Eileen, Waldron, Thomas L., Schaeffer, Thomas R., Hedberg, S.Anders, Petrillo, Edward W.
Published in Bioorganic & medicinal chemistry letters (1994)
Published in Bioorganic & medicinal chemistry letters (1994)
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Syntheses of Cyclopentane, Cyclohexene and Olefin Oxazoles as Thromboxane A2/Endoperoxide Receptor Antagonists
Das, Jagabandhu, Hall, Steven E., Reid, Joyce A., Han, Wen-Ching, Harris, Don N., Goldenberg, Harold, Michel, Inge M., Monshizadegan, Hossain, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (01.06.1993)
Published in Bioorganic & medicinal chemistry letters (01.06.1993)
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Syntheses of Cyclopentane, Cyclohexene and Olefin Oxazoles as Thromboxane A 2/Endoperoxide Receptor Antagonists
Das, Jagabandhu, Hall, Steven E., Reid, Joyce A., Han, Wen-Ching, Harris, Don N., Goldenberg, Harold, Michel, Inge M., Monshizadegan, Hossain, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (1993)
Published in Bioorganic & medicinal chemistry letters (1993)
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Diol sulfonamides: A potent and novel class of inhibitors of human renin
Poss, Michael A., Reid, Joyce A., Free, Charles A., Rogers, W.Lynn, Weber, Helen, Ryono, Denis E., Dejneka, Tamara, DeForrest, Jack M., Waldron, Thomas L., Brittain, Russell J., Weller, Harold N., Cimarusti, Maria P., Petrillo, Edward W.
Published in Bioorganic & medicinal chemistry letters (01.12.1993)
Published in Bioorganic & medicinal chemistry letters (01.12.1993)
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