Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer's disease therapy
Pachón-Angona, Irene, Refouvelet, Bernard, Andrýs, Rudolf, Martin, Helène, Luzet, Vincent, Iriepa, Isabel, Moraleda, Ignacio, Diez-Iriepa, Daniel, Oset-Gasque, María-Jesús, Marco-Contelles, José, Musilek, Kamil, Ismaili, Lhassane
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
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Exploring the Potential of Sulfonamide-Dihydropyridine Hybrids as Multitargeted Ligands for Alzheimer's Disease Treatment
Dakhlaoui, Imen, Bernard, Paul J, Pietrzak, Diana, Simakov, Alexey, Maj, Maciej, Refouvelet, Bernard, Béduneau, Arnaud, Cornu, Raphaël, Jozwiak, Krzysztof, Chabchoub, Fakher, Iriepa, Isabel, Martin, Helene, Marco-Contelles, José, Ismaili, Lhassane
Published in International journal of molecular sciences (04.06.2023)
Published in International journal of molecular sciences (04.06.2023)
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Design, Synthesis and Biological Evaluation of New Antioxidant and Neuroprotective Multitarget Directed Ligands Able to Block Calcium Channels
Pachòn Angona, Irene, Daniel, Solene, Martin, Helene, Bonet, Alexandre, Wnorowski, Artur, Maj, Maciej, Jóźwiak, Krzysztof, Silva, Tiago Barros, Refouvelet, Bernard, Borges, Fernanda, Marco-Contelles, José, Ismaili, Lhassane
Published in Molecules (Basel, Switzerland) (14.03.2020)
Published in Molecules (Basel, Switzerland) (14.03.2020)
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Acetylcholinesterase Inhibition of Diversely Functionalized Quinolinones for Alzheimer's Disease Therapy
Bautista-Aguilera, Óscar M, Ismaili, Lhassane, Chioua, Mourad, Andrys, Rudolf, Schmidt, Monika, Bzonek, Petr, Martínez-Grau, María Ángeles, Beadle, Christopher D, Vetman, Tatiana, López-Muñoz, Francisco, Iriepa, Isabel, Refouvelet, Bernard, Musilek, Kamil, Marco-Contelles, José
Published in International journal of molecular sciences (01.06.2020)
Published in International journal of molecular sciences (01.06.2020)
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Synthesis and biological assessment of KojoTacrines as new agents for Alzheimer's disease therapy
Dgachi, Youssef, Martin, Hélène, Malek, Rim, Jun, Daniel, Janockova, Jana, Sepsova, Vendula, Soukup, Ondrej, Iriepa, Isabel, Moraleda, Ignacio, Maalej, Emna, Carreiras, M. Carmo, Refouvelet, Bernard, Chabchoub, Fakher, Marco-Contelles, José, Ismaili, Lhassane
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
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Pharmacophore Modelling and Synthesis of Quinoline-3-Carbohydrazide as Antioxidants
El Bakkali, Mustapha, Ismaili, Lhassane, Tomassoli, Isabelle, Nicod, Laurence, Pudlo, Marc, Refouvelet, Bernard
Published in International Journal of Medicinal Chemistry (Online) (01.01.2011)
Published in International Journal of Medicinal Chemistry (Online) (01.01.2011)
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Multitarget compounds bearing tacrine- and donepezil-like structural and functional motifs for the potential treatment of Alzheimer's disease
Ismaili, Lhassane, Refouvelet, Bernard, Benchekroun, Mohamed, Brogi, Simone, Brindisi, Margherita, Gemma, Sandra, Campiani, Giuseppe, Filipic, Slavica, Agbaba, Danica, Esteban, Gerard, Unzeta, Mercedes, Nikolic, Katarina, Butini, Stefania, Marco-Contelles, José
Published in Progress in neurobiology (01.04.2017)
Published in Progress in neurobiology (01.04.2017)
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Quinolone–benzylpiperidine derivatives as novel acetylcholinesterase inhibitor and antioxidant hybrids for Alzheimer Disease
Pudlo, Marc, Luzet, Vincent, Ismaïli, Lhassane, Tomassoli, Isabelle, Iutzeler, Anne, Refouvelet, Bernard
Published in Bioorganic & medicinal chemistry (15.04.2014)
Published in Bioorganic & medicinal chemistry (15.04.2014)
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Journal Article
Synthesis and evaluation of lipoic acid – donepezil hybrids for Alzheimer’s disease using a straightforward strategy
Luzet, Vincent, Allemand, Florentin, Richet, Chloé, Dehecq, Barbara, Bonet, Alexandre, Harakat, Dominique, Refouvelet, Bernard, Martin, Hélène, Cardey, Bruno, Pudlo, Marc
Published in Bioorganic & medicinal chemistry letters (01.11.2024)
Published in Bioorganic & medicinal chemistry letters (01.11.2024)
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Journal Article
The Antioxidant Additive Approach for Alzheimer’s Disease Therapy: New Ferulic (Lipoic) Acid Plus Melatonin Modified Tacrines as Cholinesterases Inhibitors, Direct Antioxidants, and Nuclear Factor (Erythroid-Derived 2)-Like 2 Activators
Benchekroun, Mohamed, Romero, Alejandro, Egea, Javier, León, Rafael, Michalska, Patrycja, Buendía, Izaskun, Jimeno, María Luisa, Jun, Daniel, Janockova, Jana, Sepsova, Vendula, Soukup, Ondrej, Bautista-Aguilera, Oscar M, Refouvelet, Bernard, Ouari, Olivier, Marco-Contelles, José, Ismaili, Lhassane
Published in Journal of medicinal chemistry (10.11.2016)
Published in Journal of medicinal chemistry (10.11.2016)
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Pharmacological Profile of 6,12-Dihydro-3-methoxy-1-benzopyrano[3,4-b][1,4]benzothiazin-6-one, a Novel Human Estrogen Receptor Agonist
Jacquot, Yves, Cleeren, Anny, Laios, Ioanna, Ma, Yan, Boulahdour, Athem, Bermont, Laurent, Refouvelet, Bernard, Adessi, Gérard, Leclercq, Guy, Xicluna, Alain
Published in Biological & pharmaceutical bulletin (01.03.2002)
Published in Biological & pharmaceutical bulletin (01.03.2002)
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Journal Article
Donepezil plus chromone plus melatonin hybrids as promising agents for Alzheimer's disease therapy
Pachon-Angona, Irene, Refouvelet, Bernard, Andrys, Rudolf, Martin, Helene, Luzet, Vincent, Iriepa, Isabel, Moraleda, Ignacio, Diez-Iriepa, Daniel, Oset-Gasque, Maria-Jesus, Marco-Contelles, Jose, Musilek, Kamil, Ismaili, Lhassane
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
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Journal Article
Exploring the Potential of Sulfonamide-Dihydropyridine Hybrids as Multitargeted Ligands for Alzheimer’s Disease Treatment
Dakhlaoui, Imen, Bernard, Paul, Pietrzak, Diana, Simakov, Alexey, Maj, Maciej, Refouvelet, Bernard, Béduneau, Arnaud, Cornu, Raphaël, Jozwiak, Krzysztof, Chabchoub, Fakher, Iriepa, Isabel, Martin, Helene, Marco-Contelles, José, Ismaili, Lhassane
Published in International journal of molecular sciences (04.06.2023)
Published in International journal of molecular sciences (04.06.2023)
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Journal Article
Discovery of New Highly Potent Histamine H 3 Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase Inhibitors
Malek, Rim, Sałat, Kinga, Totoson, Perle, Karcz, Tadeusz, Refouvelet, Bernard, Skrzypczak-Wiercioch, Anna, Maj, Maciej, Simakov, Alexey, Martin, Helene, Siwek, Agata, Szałaj, Natalia, Godyń, Justyna, Panek, Dawid, Więckowska, Anna, Jozwiak, Krzysztof, Demougeot, Celine, Kieć-Kononowicz, Katarzyna, Chabchoub, Fakher, Iriepa, Isabel, Marco-Contelles, José, Ismaili, Lhassane
Published in ACS chemical neuroscience (18.09.2024)
Published in ACS chemical neuroscience (18.09.2024)
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5-amino salicylic acid bound nanoparticles for the therapy of inflammatory bowel disease
Pertuit, David, Moulari, Brice, Betz, Thomas, Nadaradjane, Arulraj, Neumann, Dirk, Ismaïli, Lhassane, Refouvelet, Bernard, Pellequer, Yann, Lamprecht, Alf
Published in Journal of controlled release (20.11.2007)
Published in Journal of controlled release (20.11.2007)
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(±)-BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3β Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer’s Disease
Ismaili, Lhassane, Monnin, Julie, Etievant, Adeline, Arribas, Raquel L, Viejo, Lucía, Refouvelet, Bernard, Soukup, Ondrej, Janockova, Jana, Hepnarova, Vendula, Korabecny, Jan, Kucera, Tomas, Jun, Daniel, Andrys, Rudolf, Musilek, Kamil, Baguet, Aurelie, García-Frutos, Eva M, De Simone, Angela, Andrisano, Vincenza, Bartolini, Manuela, de los Ríos, Cristóbal, Marco-Contelles, José, Haffen, Emmanuel
Published in ACS chemical neuroscience (21.04.2021)
Published in ACS chemical neuroscience (21.04.2021)
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