Structure-Guided Identification of Resistance Breaking Antimalarial N‑Myristoyltransferase Inhibitors
Schlott, Anja C, Mayclin, Stephen, Reers, Alexandra R, Coburn-Flynn, Olivia, Bell, Andrew S, Green, Judith, Knuepfer, Ellen, Charter, David, Bonnert, Roger, Campo, Brice, Burrows, Jeremy, Lyons-Abbott, Sally, Staker, Bart L, Chung, Chun-Wa, Myler, Peter J, Fidock, David A, Tate, Edward W, Holder, Anthony A
Published in Cell chemical biology (18.07.2019)
Published in Cell chemical biology (18.07.2019)
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Identification of and Structural Insights into Hit Compounds Targeting N‑Myristoyltransferase for Cryptosporidium Drug Development
Fenwick, Michael K., Reers, Alexandra R., Liu, Yi, Zigweid, Rachael, Sankaran, Banumathi, Shin, Janis, Hulverson, Matthew A., Hammerson, Bradley, Fernández Álvaro, Elena, Myler, Peter J., Kaushansky, Alexis, Van Voorhis, Wesley C., Fan, Erkang, Staker, Bart L.
Published in ACS infectious diseases (13.10.2023)
Published in ACS infectious diseases (13.10.2023)
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The Flame-Retardant Tris(1,3-dichloro-2-propyl) Phosphate Represses Androgen Signaling in Human Prostate Cancer Cell Lines
Reers, Alexandra R., Eng, Margaret L., Williams, Tony D., Elliott, John E., Cox, Michael E., Beischlag, Timothy V.
Published in Journal of biochemical and molecular toxicology (01.05.2016)
Published in Journal of biochemical and molecular toxicology (01.05.2016)
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The Effects of the Organic Flame-Retardant 1,2-Dibromo-4-(1,2-dibromoethyl) Cyclohexane (TBECH) on Androgen Signaling in Human Prostate Cancer Cell Lines
Wong, Lilian I. L., Reers, Alexandra R., Currier, Heidi A., Williams, Tony D., Cox, Michael E., Elliott, John E., Beischlag, Timothy V.
Published in Journal of biochemical and molecular toxicology (01.05.2016)
Published in Journal of biochemical and molecular toxicology (01.05.2016)
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The crystal structure of dihydrodipicolinate reductase from the human-pathogenic bacterium Bartonella henselae strain Houston-1 at 2.3 Å resolution
Cala, Ali R., Nadeau, Maria T., Abendroth, Jan, Staker, Bart L., Reers, Alexandra R., Weatherhead, Anthony W., Dobson, Renwick C. J., Myler, Peter J., Hudson, André O.
Published in Acta crystallographica. Section F, Structural biology communications (01.12.2016)
Published in Acta crystallographica. Section F, Structural biology communications (01.12.2016)
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Identification of Selective Inhibitors of Plasmodium N‑Myristoyltransferase by High-Throughput Screening
Harupa, Anke, De Las Heras, Laura, Colmenarejo, Gonzalo, Lyons-Abbott, Sally, Reers, Alexandra, Caballero Hernandez, Iván, Chung, Chun-Wa, Charter, David, Myler, Peter J, Fernández-Menéndez, Raquel M, Calderón, Félix, Palomo, Sara, Rodríguez, Beatriz, Berlanga, Manuela, Herreros-Avilés, Esperanza, Staker, Bart L, Fernández Álvaro, Elena, Kaushansky, Alexis
Published in Journal of medicinal chemistry (23.01.2020)
Published in Journal of medicinal chemistry (23.01.2020)
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Ternary structure of Plasmodium vivaxN‐myristoyltransferase with myristoyl‐CoA and inhibitor IMP‐0001173
Bolling, Cydni, Mendez, Alex, Taylor, Shane, Makumire, Stanley, Reers, Alexandra, Zigweid, Rachael, Subramanian, Sandhya, Dranow, David M., Staker, Bart, Edwards, Thomas E., Tate, Edward W., Bell, Andrew S., Myler, Peter J., Asojo, Oluwatoyin A., Chakafana, Graham
Published in Acta crystallographica. Section F, Structural biology communications (01.10.2024)
Published in Acta crystallographica. Section F, Structural biology communications (01.10.2024)
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Journal Article
Structural insights on three series of anti-malarial N -myristoyltransferase inhibitors
Mayclin, Stephen, Schlott, Anja, Reers, Alexandra, Coburn-Flynn, Olivia, Holder, Anthony, Bell, Andrew, Fidock, David, Tate, Edward
Published in Acta crystallographica. Section A, Foundations and advances (20.07.2018)
Published in Acta crystallographica. Section A, Foundations and advances (20.07.2018)
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Journal Article
The crystal structure of dihydrodipicolinate reductase from the human-pathogenic bacterium Bartonella henselae strain Houston-1 at 2.3Aa resolution
Cala, Ali R, Nadeau, Maria T, Abendroth, Jan, Staker, Bart L, Reers, Alexandra R, Weatherhead, Anthony W, Dobson, Renwick CJ, Myler, Peter J, Hudson, Andre O
Published in Acta crystallographica. Section F, Structural biology communications (01.12.2016)
Published in Acta crystallographica. Section F, Structural biology communications (01.12.2016)
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Journal Article
The crystal structure of dihydrodipicolinate reductase from the human-pathogenic bacterium Bartonella henselae strain Houston-1 at 2.3Å resolution
Cala, Ali R, Nadeau, Maria T, Abendroth, Jan, Staker, Bart L, Reers, Alexandra R, Weatherhead, Anthony W, Dobson, Renwick C J, Myler, Peter J, Hudson, André O
Published in Acta crystallographica. Section F, Structural biology communications (01.12.2016)
Published in Acta crystallographica. Section F, Structural biology communications (01.12.2016)
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Journal Article