Chiral recognition of the angiotensin II (AT 1) receptor by a highly potent phenoxyproline octanoamide
Steinberg, M.I., Palkowitz, A.D., Thrasher, K.J., Reel, J.K., Zimmerman, K.M., Whitesitt, C.A., Simon, R.L., Hauser, K.L., Lifer, S.L., Pfeifer, W., Takeuchi, K., Wiest, S.A., Vasudevan, V., Bermis, K.G., Deeter, J.B, Barnett, C.J., Wilson, T.M., Marshall, W.S., Boyd, D.B.
Published in Bioorganic & medicinal chemistry letters (06.01.1994)
Published in Bioorganic & medicinal chemistry letters (06.01.1994)
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Structure-activity relationships of trans-3,4-dimethyl-4-(3-hydroxyphenyl)piperidine antagonists for .mu.- and .kappa.-opioid receptors
Zimmerman, Dennis M, Leander, J. David, Cantrell, Buddy E, Reel, Jon K, Snoddy, John, Mendelsohn, Laurane G, Johnson, Bryan G, Mitch, Charles H
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
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Functional gamma‐secretase inhibitors reduce beta‐amyloid peptide levels in brain
Dovey, H. F., John, V., Anderson, J. P., Chen, L. Z., De Saint Andrieu, P., Fang, L. Y., Freedman, S. B., Folmer, B., Goldbach, E., Holsztynska, E. J., Hu, K. L., Johnson‐Wood, K. L., Kennedy, S. L., Kholodenko, D., Knops, J. E., Latimer, L. H., Lee, M., Liao, Z., Lieberburg, I. M., Motter, R. N., Mutter, L. C., Nietz, J., Quinn, K. P., Sacchi, K. L., Seubert, P. A., Shopp, G. M., Thorsett, E. D., Tung, J. S., Wu, J., Yang, S., Yin, C. T., Schenk, D. B., May, P. C., Altstiel, L. D., Bender, M. H., Boggs, L. N., Britton, T. C., Clemens, J. C., Czilli, D. L., Dieckman‐McGinty, D. K., Droste, J. J., Fuson, K. S., Gitter, B. D., Hyslop, P. A., Johnstone, E. M., Li, W‐Y., Little, S. P., Mabry, T. E., Miller, F. D., Ni, B., Nissen, J. S., Porter, W. J., Potts, B. D., Reel, J. K., Stephenson, D., Su, Y., Shipley, L. A., Whitesitt, C. A., Yin, T., Audia, J. E.
Published in Journal of neurochemistry (01.01.2001)
Published in Journal of neurochemistry (01.01.2001)
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Structural Evolution and Pharmacology of a Novel Series of Triacid Angiotensin II Receptor Antagonists
Palkowitz, Alan D, Steinberg, Mitchell I, Thrasher, K. Jeff, Reel, Jon K, Hauser, Kenneth L, Zimmerman, Karen M, Wiest, Sally A, Whitesitt, Celia A, Simon, Richard L
Published in Journal of medicinal chemistry (01.12.1994)
Published in Journal of medicinal chemistry (01.12.1994)
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3,4-Dimethyl-4-(3-hydroxyphenyl)piperidines: opioid antagonists with potent anorectant activity
Mitch, Charles H, Leander, J. David, Mendelsohn, Laurane G, Shaw, Walter N, Wong, David T, Cantrell, Buddy E, Johnson, Bryan G, Reel, John K, Snoddy, John D
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
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Characterization of the neurotoxic potential of m-methoxy-MPTP and the use of its N-ethyl analogue as a means of avoiding exposure to a possible Parkinsonism-causing agent
ZIMMERMAN, D. M, CANTRELL, B. E, REEL, J. K, HEMRICK-LUECKE, S. K, FULLER, R. W
Published in Journal of medicinal chemistry (01.08.1986)
Published in Journal of medicinal chemistry (01.08.1986)
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The development of potent and selective bisarylmaleimide GSK3 inhibitors
Engler, Thomas A., Malhotra, Sushant, Burkholder, Timothy P., Henry, James R., Mendel, David, Porter, Warren J., Furness, Kelly, Diefenbacher, Clive, Marquart, Angela, Reel, Jon K., Li, Yihong, Clayton, Joshua, Cunningham, Brian, McLean, Johnathan, O’Toole, John C., Brozinick, Joseph, Hawkins, Eric, Misener, Elizabeth, Briere, Daniel, Brier, Richard A., Wagner, Jill R., Campbell, Robert M., Anderson, Bryan D., Vaughn, Renee, Bennett, Donald B., Meier, Timothy I., Cook, James A.
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
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Journal Article
Synthesis and absolute configuration of LY25582, a potent opioid antagonist
MITCH, C. H, ZIMMERMAN, D. M, SNODDY, J. D, REEL, J. K, CANTRELL, B. E
Published in Journal of organic chemistry (1991)
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Published in Journal of organic chemistry (1991)
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3,4-dimentyl-4-(3-hydroxyphenyl)piperidines : opioid angatonists with potent anorectant activity
MITCH, C. H, LEANDER, J. D, ZIMMERMAN, D. M, MENDELSOHN, L. G, SHAW, W. N, WONG, D. T, CANTRELL, B. E, JOHNSON, B. G, REEL, J. K, SNODDY, J. D, TAKEMORI, A. E
Published in Journal of medicinal chemistry (1993)
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Published in Journal of medicinal chemistry (1993)
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STRUCTURE-ACTIVITY-RELATIONSHIPS OF TRANS-3,4-DIMETHYL-4-(3-HYDROXYPHENYL)PIPERIDINE ANTAGONISTS FOR MU-OPIOID AND KAPPA-OPIOID RECEPTORS
ZIMMERMAN, DM, LEANDER, JD, CANTRELL, BE, REEL, JK, SNODDY, J, MENDELSOHN, LG, JOHNSON, BG, MITCH, CH
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
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Journal Article
Synthesis and structure-activity relationships of benzophenones as inhibitors of cathepsin D
Whitesitt, Celia A., Simon, Richard L., Reel, Jon K., Sigmund, Sandra K., Phillips, Michael L., Kevin Shadle, J., Heinz, Lawrence J., Koppel, Gary A., Hunden, David C., Lifer, Sherryl L., Berry, Dennis, Ray, Judy, Little, Sheila P, Xiadong Liu, Marshall, Winston S., Panetta, Jill A.
Published in Bioorganic & medicinal chemistry letters (17.09.1996)
Published in Bioorganic & medicinal chemistry letters (17.09.1996)
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CHARACTERIZATION OF THE NEUROTOXIC POTENTIAL OF META-METHOXY-MPTP AND THE USE OF ITS N-ETHYL ANALOG AS A MEANS OF AVOIDING EXPOSURE TO A POSSIBLE PARKINSONISM-CAUSING AGENT
ZIMMERMAN, DM, CANTRELL, BE, REEL, JK, HEMRICKLUECKE, SK, FULLER, RW
Published in Journal of medicinal chemistry (01.08.1986)
Published in Journal of medicinal chemistry (01.08.1986)
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Synthesis and absolute configuration of LY255582, a potent opioid antagonist
Mitch, Charles H, Zimmerman, Dennis M, Snoddy, John D, Reel, Jon K, Cantrell, Buddy E
Published in Journal of organic chemistry (01.02.1991)
Published in Journal of organic chemistry (01.02.1991)
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