Small Molecule Mimetics of α-Helical Domain of IRAK2 Attenuate the Proinflammatory Effects of IL-33 in Asthma-like Mouse Models
Li, Jinghong, Saruta, Kunio, Dumouchel, Justin P, Magat, Jenna M, Thomas, Joanna L, Ajami, Dariush, Rebek, Mitra, Rebek, Jr, Julius, Bigby, Timothy D
Published in The Journal of immunology (1950) (15.06.2018)
Published in The Journal of immunology (1950) (15.06.2018)
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MyD88-dependent and -independent signaling by IL-1 in neurons probed by bifunctional Toll/IL-1 receptor domain/BB-loop mimetics
Christopher N. Davis, Enrique Mann, M. Margarita Behrens, Svetlana Gaidarova, Mitra Rebek, Julius Rebek, Jr, Tamas Bartfai
Published in Proceedings of the National Academy of Sciences - PNAS (21.02.2006)
Published in Proceedings of the National Academy of Sciences - PNAS (21.02.2006)
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Therapeutic inhibition of pro-inflammatory signaling and toxicity to staphylococcal enterotoxin B by a synthetic dimeric BB-loop mimetic of MyD88
Kissner, Teri L, Ruthel, Gordon, Alam, Shahabuddin, Mann, Enrique, Ajami, Dariush, Rebek, Mitra, Larkin, Eileen, Fernandez, Stefan, Ulrich, Robert G, Ping, Sun, Waugh, David S, Rebek, Jr, Julius, Saikh, Kamal U
Published in PloS one (27.07.2012)
Published in PloS one (27.07.2012)
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Synthesis and Biological Activity of DNA Damaging Agents that Form Decoy Binding Sites for the Estrogen Receptor
Rink, Stacia M., Yarema, Kevin J., Solomon, Marjorie S., Paige, Lisa A., Tadayoni-Rebek, B. Mitra, Essigmann, John M., Croy, Robert G.
Published in Proceedings of the National Academy of Sciences - PNAS (24.12.1996)
Published in Proceedings of the National Academy of Sciences - PNAS (24.12.1996)
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Small molecule mimetics of α-helical domain of IRAK2 attenuate the pro-inflammatory effects of IL-33 in asthma-like mouse models
Li, Jinghong, Saruta, Kunio, Dumouchel, Justin P., Magat, Jenna M., Thomas, Joanna L., Ajami, Dariush, Rebek, Mitra, Rebek, Julius, Bigby, Timothy D.
Published in The Journal of immunology (1950) (04.05.2018)
Published in The Journal of immunology (1950) (04.05.2018)
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Rational design of peptide derivatives for inhibition of MyD88‐mediated toll‐like receptor signaling in human peripheral blood mononuclear cells and epithelial cells exposed to Francisella tularensis
Ryan, Daniel A., Degardin, Melissa, Alam, Shahabuddin, Kissner, Teri L., Hale, Martha, Cameron, Michael D., Rebek, Mitra, Ajami, Dariush, Saikh, Kamal U., Rebek, Julius
Published in Chemical biology & drug design (01.12.2017)
Published in Chemical biology & drug design (01.12.2017)
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A Small Molecule That Mimics the BB-loop in the Toll Interleukin-1 (IL-1) Receptor Domain of MyD88 Attenuates Staphylococcal Enterotoxin B-induced Pro-inflammatory Cytokine Production and Toxicity in Mice
Kissner, Teri L., Moisan, Lionel, Mann, Enrique, Alam, Shahabuddin, Ruthel, Gordon, Ulrich, Robert G., Rebek, Mitra, Rebek, Julius, Saikh, Kamal U.
Published in The Journal of biological chemistry (09.09.2011)
Published in The Journal of biological chemistry (09.09.2011)
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Structure-Based Design and Synthesis of a Small Molecule that Exhibits Anti-inflammatory Activity by Inhibition of MyD88-mediated Signaling to Bacterial Toxin Exposure
Alam, Shahabuddin, Javor, Sacha, Degardin, Melissa, Ajami, Dariush, Rebek, Mitra, Kissner, Teri L., Waag, David M., Rebek Jr, Julius, Saikh, Kamal U.
Published in Chemical biology & drug design (01.08.2015)
Published in Chemical biology & drug design (01.08.2015)
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Formylated polyamines as peptidomimetics
Javor, Sacha, Janowsky, Aaron, Johnson, Robert, Wolfrum, Katherine, Tadayoni-Rebek, Mitra, Rebek, Julius
Published in Bioorganic & medicinal chemistry letters (01.11.2012)
Published in Bioorganic & medicinal chemistry letters (01.11.2012)
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MyD88-Dependent and -Independent Signaling by IL-1 in Neurons Probed by Bifunctional Toll/IL-1 Receptor Domain/BB-Ioop Mimetics
Davis, Christopher N., Mann, Enrique, Behrens, M. Margarita, Gaidarova, Svetlana, Rebek, Mitra, Rebek, Julius, Bartfai, Tamas
Published in Proceedings of the National Academy of Sciences - PNAS (21.02.2006)
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Published in Proceedings of the National Academy of Sciences - PNAS (21.02.2006)
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