Editorial: The boulder peptide symposium 2021 scientific update
Angell, Yvonne, Mayer, John, Nofsinger, Rebecca, Danho, Waleed
Published in Frontiers in drug discovery (25.03.2024)
Published in Frontiers in drug discovery (25.03.2024)
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Journal Article
Design of prodrugs to enhance colonic absorption by increasing lipophilicity and blocking ionization
Nofsinger, Rebecca, Clas, Sophie-Dorothee, Sanchez, Rosa I, Walji, Abbas, Manser, Kimberly, Nissley, Becky, Balsells, Jaume, Nair, Amrithraj, Dang, Qun, Bennett, David Jonathan, Hafey, Michael, Wang, Junying, Higgins, John, Templeton, Allen, Coleman, Paul, Grobler, Jay, Smith, Ronald, Wu, Yunhui
Published in Pharmaceuticals (Basel, Switzerland) (24.02.2014)
Published in Pharmaceuticals (Basel, Switzerland) (24.02.2014)
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Journal Article
Chemistry-enabled drug delivery (prodrugs): recent progress and challenges
Clas, Sophie-Dorothee, Sanchez, Rosa I., Nofsinger, Rebecca
Published in Drug discovery today (01.01.2014)
Published in Drug discovery today (01.01.2014)
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Journal Article
Head-to-Head Comparison of Caco‑2 Transwell and Gut-on-a-Chip Models for Assessing Oral Peptide Formulations
Gleeson, John P., Zhang, Stephanie Y., Subelzu, Natalia, Ling, Jing, Nissley, Becky, Ong, Whitney, Nofsinger, Rebecca, Kesisoglou, Filippos
Published in Molecular pharmaceutics (05.08.2024)
Published in Molecular pharmaceutics (05.08.2024)
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Journal Article
3D printed capsules for quantitative regional absorption studies in the GI tract
Smith, Derrick, Kapoor, Yash, Hermans, Andre, Nofsinger, Rebecca, Kesisoglou, Filippos, Gustafson, Tiffany P., Procopio, Adam
Published in International journal of pharmaceutics (25.10.2018)
Published in International journal of pharmaceutics (25.10.2018)
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Journal Article
A Retrospective Analysis of Preclinical and Clinical Pharmacokinetics from Administration of Long-Acting Aqueous Suspensions
Johnson, Ashley R., Ballard, Jeanine E., Leithead, Andrew, Miller, Corin, Faassen, Fried, Zang, Xiaowei, Nofsinger, Rebecca, Wagner, Angela M.
Published in Pharmaceutical research (01.07.2023)
Published in Pharmaceutical research (01.07.2023)
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Journal Article
Controlled release of etoricoxib from poly(ester urea) films for post-operative pain management
Brigham, Natasha C., Nofsinger, Rebecca, Luo, Xin, Dreger, Nathan Z., Abel, Alexandra K., Gustafson, Tiffany P., Forster, Seth P., Hermans, Andre, Ji, Ru-Rong, Becker, Matthew L.
Published in Journal of controlled release (10.01.2021)
Published in Journal of controlled release (10.01.2021)
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Journal Article
Assessing the Utility of In Vitro Screening Tools for Predicting Bio-Performance of Oral Peptide Delivery
Gadgil, Prajakta, Alleyne, Candice, Feng, Kung-I, Hu, Mengwei, Gindy, Marian, Buevich, Alexei V., Fauty, Scott, Salituro, Gino, Wen, Jianzhong, Li, Ying, Nofsinger, Rebecca, Sawyer, Tomi K., Buist, Nicole
Published in Pharmaceutical research (01.10.2019)
Published in Pharmaceutical research (01.10.2019)
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Journal Article
Comparing Dog and Human Intestinal Fluids: Implications on Solubility and Biopharmaceutical Risk Assessment
Walsh, Paul L., Stellabott, Joyce, Nofsinger, Rebecca, Xu, Wei, Levorse, Dorothy, Galipeau, Kendra, Kesisoglou, Filippos
Published in AAPS PharmSciTech (01.05.2017)
Published in AAPS PharmSciTech (01.05.2017)
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Journal Article
Analyzing the Potential Root Causes of Variability of Pharmacokinetics in Preclinical Species
Daublain, Pierre, Feng, Kung-I, Altman, Michael D, Martin, Iain, Mukherjee, Suman, Nofsinger, Rebecca, Northrup, Alan B, Tschirret-Guth, Richard, Cartwright, Mark, McGregor, Caroline
Published in Molecular pharmaceutics (01.05.2017)
Published in Molecular pharmaceutics (01.05.2017)
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Journal Article
Factors that Restrict the Cell Permeation of Cyclic Prodrugs of an Opioid Peptide, Part 4: Characterization of the Biopharmaceutical and Physicochemical Properties of Two New Cyclic Prodrugs Designed to be Stable to Oxidative Metabolism by Cytochrome P-450 Enzymes in the Intestinal Mucosa
Nofsinger, Rebecca, Borchardt, Ronald T.
Published in Journal of pharmaceutical sciences (01.09.2012)
Published in Journal of pharmaceutical sciences (01.09.2012)
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Journal Article
Factors that Restrict the Cell Permeation of Cyclic Prodrugs of an Opioid Peptide, Part 3: Synthesis of Analogs Designed to have Improved Stability to Oxidative Metabolism
Nofsinger, Rebecca, Fuchs-Knotts, Tarra, Borchardt, Ronald T.
Published in Journal of pharmaceutical sciences (01.09.2012)
Published in Journal of pharmaceutical sciences (01.09.2012)
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Journal Article
A canine biorelevant dissolution method for predicting in vivo performance of orally administered sustained release matrix tablets
Walsh, Paul L., Bothe, Jameson R., Bhardwaj, Sunny, Hu, Mengwei, Nofsinger, Rebecca, Xia, Binfeng, Persak, Steven, Pennington, Justin, Bak, Annette
Published in Drug development and industrial pharmacy (03.05.2016)
Published in Drug development and industrial pharmacy (03.05.2016)
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Journal Article
Discovery of MK-8970: An Acetal Carbonate Prodrug of Raltegravir with Enhanced Colonic Absorption
Walji, Abbas M., Sanchez, Rosa I., Clas, Sophie-Dorothee, Nofsinger, Rebecca, de Lera Ruiz, Manuel, Li, Jing, Bennet, Amrithraj, John, Christopher, Bennett, David Jonathan, Sanders, John M., Di Marco, Christina N., Kim, Somang Hope, Balsells, Jaume, Ceglia, Scott S., Dang, Qun, Manser, Kimberly, Nissley, Becky, Wai, John S., Hafey, Michael, Wang, Junying, Chessen, Gene, Templeton, Allen, Higgins, John, Smith, Ronald, Wu, Yunhui, Grobler, Jay, Coleman, Paul J.
Published in ChemMedChem (01.02.2015)
Published in ChemMedChem (01.02.2015)
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Journal Article
A comparison of the effects of p-glycoprotein inhibitors on the blood–brain barrier permeation of cyclic prodrugs of an opioid peptide (DADLE)
Ouyang, Hui, Andersen, Thomas E., Chen, Weiqing, Nofsinger, Rebecca, Steffansen, Bente, Borchardt, Ronald T.
Published in Journal of pharmaceutical sciences (01.06.2009)
Published in Journal of pharmaceutical sciences (01.06.2009)
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Journal Article
TABLET FORMULATION FOR CGRP ACTIVE COMPOUNDS
CHAD D BROWN, LISA LUPTON, XI HANMI, LEONARDO RESENDE ALLAIN, PARESH B PATEL, REBECCA NOFSINGER, MARY ANN JOHNSON, FRANCIS J FLANAGAN JR, W MARK EICKHOFF, CRAIG B IKEDA, MELANIE MAROTA, XU WEI
Year of Publication 04.07.2019
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Year of Publication 04.07.2019
Patent
Cover Picture: Discovery of MK-8970: An Acetal Carbonate Prodrug of Raltegravir with Enhanced Colonic Absorption (ChemMedChem 2/2015)
Walji, Abbas M., Sanchez, Rosa I., Clas, Sophie-Dorothee, Nofsinger, Rebecca, de Lera Ruiz, Manuel, Li, Jing, Bennet, Amrithraj, John, Christopher, Bennett, David Jonathan, Sanders, John M., Di Marco, Christina N., Kim, Somang Hope, Balsells, Jaume, Ceglia, Scott S., Dang, Qun, Manser, Kimberly, Nissley, Becky, Wai, John S., Hafey, Michael, Wang, Junying, Chessen, Gene, Templeton, Allen, Higgins, John, Smith, Ronald, Wu, Yunhui, Grobler, Jay, Coleman, Paul J.
Published in ChemMedChem (01.02.2015)
Published in ChemMedChem (01.02.2015)
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Journal Article
Formulations for cgrp receptor antagonists
Lupton, Lisa, Xu, Wei, Nofsinger, Rebecca, Allain, Leonardo, Sotthivirat, Sutthilug, Maus, Russell, Flanagan, Francis, Mahjour, Majid
Year of Publication 29.10.2021
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Year of Publication 29.10.2021
Patent
Tablet formulation for CGRP active compounds
Allain, Leonardo Resende, Eickhoff, W. Mark, Lupton, Lisa, Flanagan, Jr., Francis J, Xu, Wei, Nofsinger, Rebecca, Xi, Hanmi, Johnson, Mary Ann, Ikeda, Craig B, Marota, Melanie, Brown, Chad D, Patel, Paresh B
Year of Publication 12.03.2024
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Year of Publication 12.03.2024
Patent