Interspecies variability in expression of hepatobiliary transporters across human, dog, monkey, and rat as determined by quantitative proteomics
Wang, Li, Prasad, Bhagwat, Salphati, Laurent, Chu, Xiaoyan, Gupta, Anshul, Hop, Cornelis E C A, Evers, Raymond, Unadkat, Jashvant D
Published in Drug metabolism and disposition (01.03.2015)
Published in Drug metabolism and disposition (01.03.2015)
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Journal Article
Interindividual variability in hepatic organic anion-transporting polypeptides and P-glycoprotein (ABCB1) protein expression: quantification by liquid chromatography tandem mass spectroscopy and influence of genotype, age, and sex
Prasad, Bhagwat, Evers, Raymond, Gupta, Anshul, Hop, Cornelis E C A, Salphati, Laurent, Shukla, Suneet, Ambudkar, Suresh V, Unadkat, Jashvant D
Published in Drug metabolism and disposition (01.01.2014)
Published in Drug metabolism and disposition (01.01.2014)
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Journal Article
Disease-Associated Changes in Drug Transporters May Impact the Pharmacokinetics and/or Toxicity of Drugs: A White Paper From the International Transporter Consortium
Evers, Raymond, Piquette-Miller, Micheline, Polli, Joseph W, Russel, Frans G M, Sprowl, Jason A, Tohyama, Kimio, Ware, Joseph A, de Wildt, Saskia N, Xie, Wen, Brouwer, Kim L R
Published in Clinical pharmacology and therapeutics (01.11.2018)
Published in Clinical pharmacology and therapeutics (01.11.2018)
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Journal Article
Interindividual and Regional Variability in Drug Transporter Abundance at the Human Blood-Brain Barrier Measured by Quantitative Targeted Proteomics
Billington, Sarah, Salphati, Laurent, Hop, Cornelis E C A, Chu, Xiaoyan, Evers, Raymond, Burdette, Doug, Rowbottom, Christopher, Lai, Yurong, Xiao, Guangqing, Humphreys, W Griffith, Nguyen, Tot Bui, Prasad, Bhagwat, Unadkat, Jashvant D
Published in Clinical pharmacology and therapeutics (01.07.2019)
Published in Clinical pharmacology and therapeutics (01.07.2019)
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Journal Article
Establishment of a hepatocyte-kupffer cell coculture model for assessment of proinflammatory cytokine effects on metabolizing enzymes and drug transporters
Nguyen, Theresa V, Ukairo, Okechukwu, Khetani, Salman R, McVay, Michael, Kanchagar, Chitra, Seghezzi, Wolfgang, Ayanoglu, Gulesi, Irrechukwu, Onyi, Evers, Raymond
Published in Drug metabolism and disposition (01.05.2015)
Published in Drug metabolism and disposition (01.05.2015)
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Journal Article
Pitavastatin is a more sensitive and selective organic anion‐transporting polypeptide 1B clinical probe than rosuvastatin
Prueksaritanont, Thomayant, Chu, Xiaoyan, Evers, Raymond, Klopfer, Stephanie O., Caro, Luzelena, Kothare, Prajakti A., Dempsey, Cynthia, Rasmussen, Scott, Houle, Robert, Chan, Grace, Cai, Xiaoxin, Valesky, Robert, Fraser, Iain P., Stoch, S. Aubrey
Published in British journal of clinical pharmacology (01.09.2014)
Published in British journal of clinical pharmacology (01.09.2014)
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Journal Article
Physiologically‐based pharmacokinetic modeling for primary metabolites of CYP3A and P‐glycoprotein inhibitors in drug–drug interactions: Should we assume the free drug hypothesis?
Yamazaki, Shinji, Evers, Raymond, De Zwart, Loeckie
Published in CPT: pharmacometrics and systems pharmacology (01.01.2023)
Published in CPT: pharmacometrics and systems pharmacology (01.01.2023)
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Journal Article
Corrigendum to: Physiologically‐based pharmacokinetic modeling to evaluate in vitro‐to‐in vivo extrapolation for intestinal P‐glycoprotein inhibition
Yamazaki, Shinji, Evers, Raymond, De Zwart, Loeckie
Published in CPT: pharmacometrics and systems pharmacology (01.10.2022)
Published in CPT: pharmacometrics and systems pharmacology (01.10.2022)
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Journal Article
The hurdle of human PK Predictions for hepatic oatp substrates: lessons learned from rat allometry
Mei, Hong, Evers, Raymond, Miller, Randall
Published in Drug metabolism and pharmacokinetics (01.01.2019)
Published in Drug metabolism and pharmacokinetics (01.01.2019)
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Journal Article
In Vitro and in Vivo Induction of Cytochrome P450: A Survey of the Current Practices and Recommendations: A Pharmaceutical Research and Manufacturers of America Perspective
Chu, Valeria, Einolf, Heidi J, Evers, Raymond, Kumar, Gondi, Moore, David, Ripp, Sharon, Silva, Jose, Sinha, Vikram, Sinz, Michael, Skerjanec, Andrej
Published in Drug metabolism and disposition (01.07.2009)
Published in Drug metabolism and disposition (01.07.2009)
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Journal Article
Toward improved predictions of pharmacokinetics of transported drugs in hepatic impairment: Insights from the extended clearance model
Storelli, Flavia, Ladumor, Mayur K., Liang, Xiaomin, Lai, Yurong, Chothe, Paresh P., Enogieru, Osatohanmwen J., Evers, Raymond, Unadkat, Jashvant D.
Published in CPT: pharmacometrics and systems pharmacology (01.01.2024)
Published in CPT: pharmacometrics and systems pharmacology (01.01.2024)
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Journal Article
Predicting changes in the pharmacokinetics of CYP3A‐metabolized drugs in hepatic impairment and insights into factors driving these changes
Ladumor, Mayur K., Storelli, Flavia, Liang, Xiaomin, Lai, Yurong, Enogieru, Osatohanmwen J., Chothe, Paresh P., Evers, Raymond, Unadkat, Jashvant D.
Published in CPT: pharmacometrics and systems pharmacology (01.02.2023)
Published in CPT: pharmacometrics and systems pharmacology (01.02.2023)
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Journal Article
Transport of the Dipeptidyl Peptidase-4 Inhibitor Sitagliptin by Human Organic Anion Transporter 3, Organic Anion Transporting Polypeptide 4C1, and Multidrug Resistance P-glycoprotein
Chu, Xiao-Yan, Bleasby, Kelly, Yabut, Jocelyn, Cai, Xiaoxin, Chan, Grace Hoyee, Hafey, Michael J, Xu, Shiyao, Bergman, Arthur J, Braun, Matthew P, Dean, Dennis C, Evers, Raymond
Published in The Journal of pharmacology and experimental therapeutics (01.05.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2007)
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Journal Article
Assessment of the Effect of Pyrimethamine, a Potent Inhibitor of Multidrug and Toxin Extrusion Protein 1/2K, on the Pharmacokinetics of Gefapixant (MK‐7264), a P2X3 Receptor Antagonist
Nussbaum, Jesse C., Hussain, Azher, Ma, Bennett, Min, K. Chris, Evers, Raymond, Li, Yun, Garrett, Graigory, Stoch, S. Aubrey, Iwamoto, Marian
Published in Clinical pharmacology in drug development (01.01.2022)
Published in Clinical pharmacology in drug development (01.01.2022)
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Journal Article
Assessment of Pharmacokinetic Interaction Between Gefapixant (MK‐7264), a P2X3 Receptor Antagonist, and the OATP1B1 Drug Transporter Substrate Pitavastatin
McCrea, Jacqueline B., Hussain, Azher, Ma, Bennett, Garrett, Graigory C., Evers, Raymond, Laabs, John E., Stoch, S. Aubrey, Iwamoto, Marian
Published in Clinical pharmacology in drug development (01.03.2022)
Published in Clinical pharmacology in drug development (01.03.2022)
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Journal Article