Microwave-Assisted Paal-Knorr Reaction - Three-Step Regiocontrolled Synthesis of Polysubstituted Furans, Pyrroles and Thiophenes
Minetto, Giacomo, Raveglia, Luca F., Sega, Alessandro, Taddei, Maurizio
Published in European Journal of Organic Chemistry (01.12.2005)
Published in European Journal of Organic Chemistry (01.12.2005)
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Synthesis and biological activity of flurbiprofen analogues as selective inhibitors beta-amyloid(1-42) secretion
Peretto, Radaelli, S, Parini, C, Zandi, M, Raveglia, LF, Dondio, G, Fontanella, L, Misiano, P, Bigogno, C, Rizzi, A, Riccardi, B, Biscaioli, M, Marchetti, S, Puccini, P, Catinella, S, Rondelli, Cenacchi, Bolzoni, PT, Caruso, P, Villetti, G, Facchinetti, F, Del Giudice, E, Moretto, N, Imbimbo, BP
Published in Journal of medicinal chemistry (08.09.2005)
Published in Journal of medicinal chemistry (08.09.2005)
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Nonpeptide Tachykinin Receptor Antagonists. III. SB 235375, a Low Central Nervous System-Penetrant, Potent and Selective Neurokinin-3 Receptor Antagonist, Inhibits Citric Acid-Induced Cough and Airways Hyper-reactivity in Guinea Pigs
Hay, Douglas W P, Giardina, Giuseppe A M, Griswold, Don E, Underwood, David C, Kotzer, Charles J, Bush, Brian, Potts, William, Sandhu, Punam, Lundberg, Dave, Foley, James J, Schmidt, Dulcie B, Martin, Lenox D, Kilian, David, Legos, Jeffrey J, Barone, Frank C, Luttmann, Mark A, Grugni, Mario, Raveglia, Luca F, Sarau, Henry M
Published in The Journal of pharmacology and experimental therapeutics (01.01.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2002)
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Journal Article
Solid Phase Synthesis of Diamino-Substituted Pyrimidines
Barillari, Caterina, Barlocco, Daniela, Raveglia, Luca F.
Published in European journal of organic chemistry (01.12.2001)
Published in European journal of organic chemistry (01.12.2001)
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Journal Article
Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 2. Identification of (S)-N-(1-Phenylpropyl)-3-hydroxy-2- phenylquinoline-4-carboxamide (SB 223412)
Giardina, Giuseppe A. M, Raveglia, Luca F, Grugni, Mario, Sarau, Henry M, Farina, Carlo, Medhurst, Andrew D, Graziani, Davide, Schmidt, Dulcie B, Rigolio, Roberto, Luttmann, Mark, Cavagnera, Stefano, Foley, James J, Vecchietti, Vittorio, Hay, Douglas W. P
Published in Journal of medicinal chemistry (25.03.1999)
Published in Journal of medicinal chemistry (25.03.1999)
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Journal Article
Stepwise Modulation of Neurokinin-3 and Neurokinin-2 Receptor Affinity and Selectivity in Quinoline Tachykinin Receptor Antagonists
Blaney, Frank E, Raveglia, Luca F, Artico, Marco, Cavagnera, Stefano, Dartois, Catherine, Farina, Carlo, Grugni, Mario, Gagliardi, Stefania, Luttmann, Mark A, Martinelli, Marisa, Nadler, Guy M. M. G, Parini, Carlo, Petrillo, Paola, Sarau, Henry M, Scheideler, Mark A, Hay, Douglas W. P, Giardina, Giuseppe A. M
Published in Journal of medicinal chemistry (24.05.2001)
Published in Journal of medicinal chemistry (24.05.2001)
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Journal Article
Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 1. Identification of the 4-Quinolinecarboxamide Framework
Giardina, Giuseppe A. M, Sarau, Henry M, Farina, Carlo, Medhurst, Andrew D, Grugni, Mario, Raveglia, Luca F, Schmidt, Dulcie B, Rigolio, Roberto, Luttmann, Mark, Vecchietti, Vittorio, Hay, Douglas W. P
Published in Journal of medicinal chemistry (06.06.1997)
Published in Journal of medicinal chemistry (06.06.1997)
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Determination of the amino acid residue involved in [3H]beta-funaltrexamine covalent binding in the cloned rat mu-opioid receptor
Chen, C, Yin, J, Riel, J K, DesJarlais, R L, Raveglia, L F, Zhu, J, Liu-Chen, L Y
Published in The Journal of biological chemistry (30.08.1996)
Published in The Journal of biological chemistry (30.08.1996)
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Journal Article
2-Phenyl-4-quinolinecarboxamides: A Novel Class of Potent and Selective Non-Peptide Competitive Antagonists for the Human Neurokinin-3 Receptor
Giardina, Giuseppe A. M, Sarau, Henry M, Farina, Carlo, Medhurst, Andrew D, Grugni, Mario, Foley, James J, Raveglia, Luca F, Schmidt, Dulcie B, Rigolio, Roberto, Vassallo, Marco, Vecchietti, Vittorio, Hay, Douglas W. P
Published in Journal of medicinal chemistry (07.06.1996)
Published in Journal of medicinal chemistry (07.06.1996)
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Journal Article
Synthesis and NMR Characterization of a Novel Class of Thienomorphinans
Ronzoni, Silvano, Cerri, Alberto, Dondio, Giulio, Fronza, Giovanni, Petrillo, Paola, Raveglia, Luca F, Gatti, Pier Andrea
Published in Organic letters (12.08.1999)
Published in Organic letters (12.08.1999)
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Journal Article
Investigation of SAR requirements of SR 142801 through an indexed combinatorial library in solution
Raveglia, Luca F, Vitali, Mauro, Artico, Marco, Graziani, Davide, Hay, Douglas W.P, Luttmann, Mark A, Mena, Renzo, Pifferi, Giorgio, Giardina, Giuseppe A.M
Published in European journal of medicinal chemistry (01.10.1999)
Published in European journal of medicinal chemistry (01.10.1999)
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Journal Article
A novel synthesis of 3-halo-2-phenylquinoline-4-carboxylic acids
Raveglia, LF, Giardina, GAM, Grugni, M, Rigolio, R, Farina, C
Published in Journal of heterocyclic chemistry (01.03.1997)
Published in Journal of heterocyclic chemistry (01.03.1997)
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Journal Article
Replacement of the quinoline system in 2-phenyl-4-quinolinecarboxamide NK-3 receptor antagonists
Giardina, G.A.M, Artico, M, Cavagnera, S, Cerri, A, Consolandi, E, Gagliardi, S, Graziani, D, Grugni, M, Hay, D.W.P, Luttmann, M.A, Mena, R, Raveglia, L.F, Rigolio, R, Sarau, H.M, Schmidt, D.B, Zanoni, G, Farina, C
Published in Farmaco (Società chimica italiana : 1989) (30.06.1999)
Published in Farmaco (Società chimica italiana : 1989) (30.06.1999)
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Journal Article
Solid-Phase Convergent Synthesis of a Benzimidazolone Library via the Combination of Two Smaller Arrays of Carboxylic Acids and Secondary Amines
Bianchi, Ivana, La Porta, Elena, Barlocco, Daniela, Raveglia, Luca F
Published in Journal of combinatorial chemistry (01.09.2004)
Published in Journal of combinatorial chemistry (01.09.2004)
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