Isoquinoline Kelch-like ECH-Associated Protein 1‑Nuclear Factor (Erythroid-Derived 2)-like 2 (KEAP1-NRF2) Inhibitors with High Metabolic Stability
Lazzara, Phillip R, David, Brian P, Ankireddy, Aparna, Richardson, Benjamin G, Dye, Katherine, Ratia, Kiira M, Reddy, Sekhar P, Moore, Terry W
Published in Journal of medicinal chemistry (25.06.2020)
Published in Journal of medicinal chemistry (25.06.2020)
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Journal Article
Mechanism of Allosteric Modulation of Nicotinamide Phosphoribosyltransferase to Elevate Cellular NAD
Ratia, Kiira M., Shen, Zhengnan, Gordon-Blake, Jesse, Lee, Hyun, Laham, Megan S., Krider, Isabella S., Christie, Nicholas, Ackerman-Berrier, Martha, Penton, Christopher, Knowles, Natalie G., Musku, Soumya Reddy, Fu, Jiqiang, Velma, Ganga Reddy, Xiong, Rui, Thatcher, Gregory R. J.
Published in Biochemistry (Easton) (21.02.2023)
Published in Biochemistry (Easton) (21.02.2023)
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Synthesis and Evaluation of Noncovalent Naphthalene-Based KEAP1-NRF2 Inhibitors
Lazzara, Phillip R, Jain, Atul D, Maldonado, Amanda C, Richardson, Benjamin, Skowron, Kornelia J, David, Brian P, Siddiqui, Zamia, Ratia, Kiira M, Moore, Terry W
Published in ACS medicinal chemistry letters (09.04.2020)
Published in ACS medicinal chemistry letters (09.04.2020)
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Discovery of Nonlipogenic ABCA1 Inducing Compounds with Potential in Alzheimer’s Disease and Type 2 Diabetes
Ben Aissa, Manel, Lewandowski, Cutler T, Ratia, Kiira M, Lee, Sue H, Layden, Brian T, LaDu, Mary Jo, Thatcher, Gregory R. J
Published in ACS pharmacology & translational science (12.02.2021)
Published in ACS pharmacology & translational science (12.02.2021)
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Abstract 1063: G Protein 12 Alpha Subunit Covalent Binding To Alpha-snap And Its Potential Role In Von Willebrand Factor Secretion
Rusu, Luiza, Bloem, Laura J, Chen, Hui, Lee, Hyun, Ratia, Kiira M, Jayathilaka, Lasanthi, Carlier, Paul R, Minshall, Richard D
Published in Arteriosclerosis, thrombosis, and vascular biology (01.05.2024)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.05.2024)
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Journal Article
The mechanism of nicotinamide phosphoribosyltransferase whereby positive allosteric modulation elevates cellular NAD
Ratia, Kiira M, Shen, Zhengnan, Gordon-Blake, Jesse, Lee, Hyun, Laham, Megan S, Krider, Isabella S, Christie, Nicholas, Ackerman-Berrier, Martha S, Penton, Christopher, Knowles, Natalie G, Soumya Reddy Musku, Fu, Jiqiang, Ganga Reddy Musku, Xiong, Rui, Thatcher, Gregory R J
Published in bioRxiv (22.10.2022)
Published in bioRxiv (22.10.2022)
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Paper
COMPOUNDS AND METHODS FOR TREATING RESPIRATORY DISEASES
RATIA KIIRA M, MESECAR ANDREW DAVID, CHAUDHURI RIMA, MULHEARN DEBBIE C, TAKAYAMA JUN, GHOSH ARUN K, JOHNSON MICHAEL E
Year of Publication 03.11.2011
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Year of Publication 03.11.2011
Patent
COMPOUNDS AND METHODS FOR TREATING RESPIRATORY DISEASES
MESECAR, ANDREW DAVID, RATIA, KIIRA M, JOHNSON, MICHAEL E, CHAUDHURI, RIMA, GHOSH, ARUN K, TAKAYAMA, JUN, MULHEARN, DEBBIE C
Year of Publication 25.02.2010
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Year of Publication 25.02.2010
Patent