Nonsteroidal Selective Glucocorticoid Modulators: The Effect of C-10 Substitution on Receptor Selectivity and Functional Potency of 5-Allyl-2,5-dihydro-2,2,4-trimethyl-1H-[1]benzopyrano[3,4-f]quinolines
Kym, Philip R, Kort, Michael E, Coghlan, Michael J, Moore, Jimmie L, Tang, Rui, Ratajczyk, James D, Larson, Daniel P, Elmore, Steven W, Pratt, John K, Stashko, Michael A, Falls, H. Douglass, Lin, Chun W, Nakane, Masake, Miller, Loan, Tyree, Curtis M, Miner, Jeffery N, Jacobson, Peer B, Wilcox, Denise M, Nguyen, Phong, Lane, Benjamin C
Published in Journal of medicinal chemistry (13.03.2003)
Published in Journal of medicinal chemistry (13.03.2003)
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Structural requirements for the inhibition of 5-lipoxygenase by 15-hydroxyeicosa-5,8,11,13-tetraenoic acid analogs
Haviv, Fortuna, Ratajczyk, James D, DeNet, Robert W, Martin, Yvonne C, Dyer, Richard D, Carter, George W
Published in Journal of medicinal chemistry (01.02.1987)
Published in Journal of medicinal chemistry (01.02.1987)
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Structure−Activity Relationships of N-Hydroxyurea 5-Lipoxygenase Inhibitors
Stewart, Andrew O, Bhatia, Pramila A, Martin, Jonathan G, Summers, James B, Rodriques, Karen E, Martin, Michael B, Holms, James H, Moore, Jimmie L, Craig, Richard A, Kolasa, Teodozyj, Ratajczyk, James D, Mazdiyasni, Hormoz, Kerdesky, Francis A. J, DeNinno, Shari L, Maki, Robert G, Bouska, Jennifer B, Young, Patrick R, Lanni, Carmine, Bell, Randy L, Carter, George W, Brooks, Clint D. W
Published in Journal of medicinal chemistry (20.06.1997)
Published in Journal of medicinal chemistry (20.06.1997)
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3-[1-(2-Benzoxazolyl)hydrazino]propanenitrile derivatives: inhibitors of immune complex induced inflammation
Haviv, Fortuna, Ratajczyk, James D, DeNet, Robert W, Kerdesky, Francis A, Walters, Roland L, Schmidt, Steven P, Holms, James H, Young, Patrick R, Carter, George W
Published in Journal of medicinal chemistry (01.09.1988)
Published in Journal of medicinal chemistry (01.09.1988)
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5-Lipoxygenase Inhibitors: Synthesis and Structure−Activity Relationships of a Series of 1-Aryl-2H,4H-tetrahydro-1,2,4-triazin-3-ones
Bhatia, Pramila A, Brooks, Clint D. W, Basha, Anwer, Ratajczyk, James D, Gunn, Bruce P, Bouska, Jennifer B, Lanni, Carmine, Young, Patrick R, Bell, Randy L, Carter, George W
Published in Journal of medicinal chemistry (27.09.1996)
Published in Journal of medicinal chemistry (27.09.1996)
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Hydroxamic acid inhibitors of 5-lipoxygenase
Summers, James B, Mazdiyasni, Hormoz, Holms, James H, Ratajczyk, James D, Dyer, Richard D, Carter, George W
Published in Journal of medicinal chemistry (01.03.1987)
Published in Journal of medicinal chemistry (01.03.1987)
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Hydroxamic acid inhibitors of 5-lipoxygenase: quantitative structure-activity relationships
Summers, James B, Kim, Ki H, Mazdiyasni, Hormoz, Holms, James H, Ratajczyk, James D, Stewart, Andrew O, Dyer, Richard D, Carter, George W
Published in Journal of medicinal chemistry (01.03.1990)
Published in Journal of medicinal chemistry (01.03.1990)
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Preparation of (R)-(+)-N-[3-[5-[(4-Fluorophenyl)methyl]-2-thienyl]-1-methyl-2-propynyl]-N-hydroxyurea (ABT-761), a second-generation 5-lipoxygenase inhibitor
Brooks, Clint D. W, Stewart, Andrew O, Basha, Anwer, Bhatia, Pramila, Ratajczyk, James D, Martin, Jonathan G, Craig, Richard A, Kolasa, Teodozyj, Bouska, Jennifer B, Lanni, Carmine, Harris, Richard R, Malo, Peter E, Carter, George W, Bell, Randy L
Published in Journal of medicinal chemistry (01.11.1995)
Published in Journal of medicinal chemistry (01.11.1995)
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2-[(Phenylthio)methyl]pyridine derivatives: new antiinflammatory agents
Haviv, Fortuna, DeNet, Robert W, Michaels, Raymond J, Ratajczyk, James D, Carter, George W, Young, Patrick R
Published in Journal of medicinal chemistry (01.02.1983)
Published in Journal of medicinal chemistry (01.02.1983)
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(R)-(+)-N-[3-[5-[(4-FLUOROPHENYL)METHYL]-2-THIENYL]-1-METHYL-2-PROPYNYL]-N-HYDROXYUREA (ABT-761), A 2ND-GENERATION 5-LIPOXYGENASE INHIBITOR
BROOKS, CDW, STEWART, AO, BASHA, A, BHATIA, P, RATAJCZYK, JD, MARTIN, JG, CRAIG, RA, KOLASA, T, BOUSKA, JB, LANNI, C, HARRIS, RR, MALO, PE, CARTER, GW, BELL, RL
Published in Journal of medicinal chemistry (24.11.1995)
Published in Journal of medicinal chemistry (24.11.1995)
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5-Lipoxygenase Inhibitors: Synthesis and Structure−Activity Relationships of a Series of 1-Aryl-2 H ,4 H -tetrahydro-1,2,4-triazin-3-ones
Bhatia, Pramila A., Brooks, Clint D. W., Basha, Anwer, Ratajczyk, James D., Gunn, Bruce P., Bouska, Jennifer B., Lanni, Carmine, Young, Patrick R., Bell, Randy L., Carter, George W.
Published in Journal of medicinal chemistry (01.01.1996)
Published in Journal of medicinal chemistry (01.01.1996)
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Design of inhibitors of leukotriene biosynthesis and their therapeutic potential
Brooks, C. D. W., Stewart, A. O., Kolasa, Teodozyj, Basha, A., Bhatia, Pramila, Ratajczyk, J. D., Craig, R. A., Gunn, David, Harris, R. R., Bouska, J. B., Malo, P. E., Bell, R. L., Carter, G. W.
Published in Pure and applied chemistry (28.02.1998)
Published in Pure and applied chemistry (28.02.1998)
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