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Szczurowska, Ewa, Szánti-Pintér, Eszter, Chetverikov, Nikolai, Randáková, Alena, Kudová, Eva, Jakubík, Jan
Published in International journal of molecular sciences (28.12.2022)
Published in International journal of molecular sciences (28.12.2022)
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Analysis of equilibrium binding of an orthosteric tracer and two allosteric modulators
Dolezal, Vladimír, Jakubík, Jan, El-Fakahany, Esam E, Randáková, Alena
Published in PloS one (27.03.2019)
Published in PloS one (27.03.2019)
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Agonist-Specific Conformations of the M 2 Muscarinic Acetylcholine Receptor Assessed by Molecular Dynamics
Randáková, Alena, Nelic, Dominik, Doležal, Vladimír, El-Fakahany, Esam E, Boulos, John, Jakubík, Jan
Published in Journal of chemical information and modeling (27.04.2020)
Published in Journal of chemical information and modeling (27.04.2020)
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Novel long‐acting antagonists of muscarinic ACh receptors
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Published in British journal of pharmacology (01.05.2018)
Published in British journal of pharmacology (01.05.2018)
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Neuroactive steroids, WIN-compounds and cholesterol share a common binding site on muscarinic acetylcholine receptors
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Published in Biochemical pharmacology (01.10.2021)
Published in Biochemical pharmacology (01.10.2021)
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Novel M2‐selective, Gi‐biased agonists of muscarinic acetylcholine receptors
Randáková, Alena, Nelic, Dominik, Ungerová, Dana, Nwokoye, Peter, Su, Qiwen, Doležal, Vladimír, El‐Fakahany, Esam E., Boulos, John, Jakubík, Jan
Published in British journal of pharmacology (01.05.2020)
Published in British journal of pharmacology (01.05.2020)
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Role of membrane cholesterol in differential sensitivity of muscarinic receptor subtypes to persistently bound xanomeline
Randáková, Alena, Dolejší, Eva, Rudajev, Vladimír, Zimčík, Pavel, Doležal, Vladimír, El-Fakahany, Esam E., Jakubík, Jan
Published in Neuropharmacology (01.05.2018)
Published in Neuropharmacology (01.05.2018)
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Binding of N-methylscopolamine to the extracellular domain of muscarinic acetylcholine receptors
Jakubík, Jan, Randáková, Alena, Zimčík, Pavel, El-Fakahany, Esam E, Doležal, Vladimír
Published in Scientific reports (16.01.2017)
Published in Scientific reports (16.01.2017)
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Synthesis and In Vitro Evaluation of Novel Dopamine Receptor D2 3,4-dihydroquinolin-2(1H)-one Derivatives Related to Aripiprazole
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Published in Biomolecules (Basel, Switzerland) (24.08.2021)
Published in Biomolecules (Basel, Switzerland) (24.08.2021)
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Subtype differences in pre-coupling of muscarinic acetylcholine receptors
Dolezal, Vladimír, Jakubík, Jan, El-Fakahany, Esam E, Janícková, Helena, Randáková, Alena
Published in PloS one (16.11.2011)
Published in PloS one (16.11.2011)
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The operational model of allosteric modulation of pharmacological agonism
Jakubík, Jan, Randáková, Alena, Chetverikov, Nikolai, El-Fakahany, Esam E, Doležal, Vladimír
Published in Scientific reports (02.09.2020)
Published in Scientific reports (02.09.2020)
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Agonist-selective activation of individual G-proteins by muscarinic receptors
Nelic, Dominik, Chetverikov, Nikolai, Hochmalová, Martina, Diaz, Christina, Doležal, Vladimír, Boulos, John, Jakubík, Jan, Martemyanov, Kirill, Janoušková-Randáková, Alena
Published in Scientific reports (26.04.2024)
Published in Scientific reports (26.04.2024)
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Agonist-Specific Conformations of the M2 Muscarinic Acetylcholine Receptor Assessed by Molecular Dynamics
Randáková, Alena, Nelic, Dominik, Doležal, Vladimír, El-Fakahany, Esam E, Boulos, John, Jakubík, Jan
Published in Journal of chemical information and modeling (27.04.2020)
Published in Journal of chemical information and modeling (27.04.2020)
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Fusion with Promiscuous Gα16 Subunit Reveals Signaling Bias at Muscarinic Receptors
Randáková, Alena, Nelic, Dominik, Hochmalová, Martina, Zimčík, Pavel, Mulenga, Mutale Jane, Boulos, John, Jakubík, Jan
Published in International journal of molecular sciences (18.09.2021)
Published in International journal of molecular sciences (18.09.2021)
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