Dual Inhibition of Bruton's Tyrosine Kinase and Phosphoinositide-3-Kinase p110 δ as a Therapeutic Approach to Treat Non-Hodgkin's B Cell Malignancies
Alfaro, Jennifer, Pérez de Arce, Felipe, Belmar, Sebastián, Fuentealba, Glenda, Avila, Patricio, Ureta, Gonzalo, Flores, Camila, Acuña, Claudia, Delgado, Luz, Gaete, Diana, Pujala, Brahmam, Barde, Anup, Nayak, Anjan K, Upendra, T V R, Patel, Dhananjay, Chauhan, Shailender, Sharma, Vijay K, Kanno, Stacy, Almirez, Ramona G, Hung, David T, Chakravarty, Sarvajit, Rai, Roopa, Bernales, Sebastián, Quinn, Kevin P, Pham, Son M, McCullagh, Emma
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
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Journal Article
Discovery of Pyrazolopyrimidine Derivatives as Novel Dual Inhibitors of BTK and PI3Kδ
Pujala, Brahmam, Agarwal, Anil K, Middya, Sandip, Banerjee, Monali, Surya, Arjun, Nayak, Anjan K, Gupta, Ashu, Khare, Sweta, Guguloth, Rambabu, Randive, Nitin A, Shinde, Bharat U, Thakur, Anamika, Patel, Dhananjay I, Raja, Mohd, Green, Michael J, Alfaro, Jennifer, Avila, Patricio, Pérez de Arce, Felipe, Almirez, Ramona G, Kanno, Stacy, Bernales, Sebastián, Hung, David T, Chakravarty, Sarvajit, McCullagh, Emma, Quinn, Kevin P, Rai, Roopa, Pham, Son M
Published in ACS medicinal chemistry letters (08.12.2016)
Published in ACS medicinal chemistry letters (08.12.2016)
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Journal Article
Inhibition of p38 Mitogen-Activated Protein Kinase Augments Progression of Remnant Kidney Model by Activating the ERK Pathway
Ohashi, Ryuji, Nakagawa, Takahiko, Watanabe, Susumu, Kanellis, John, Almirez, Ramona G., Schreiner, George F., Johnson, Richard J.
Published in The American journal of pathology (01.02.2004)
Published in The American journal of pathology (01.02.2004)
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Journal Article
SD-208, a novel transforming growth factor β receptor I kinase inhibitor, inhibits growth and invasiveness and enhances immunogenicity of murine and human glioma cells in vitro and in vivo
UHL, Martin, AULWURM, Steffen, MURPHY, Alison, WONG, Darren H, WICK, Wolfgang, HIGGINS, Linda S, WELLER, Michael, WISCHHUSEN, Jörg, WEILER, Markus, JING YING MA, ALMIREZ, Ramona, MANGADU, Ruban, LIU, Yu-Wang, PLATTEN, Michael, HERRLINGER, Ulrich
Published in Cancer research (Chicago, Ill.) (01.11.2004)
Published in Cancer research (Chicago, Ill.) (01.11.2004)
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Journal Article
Human Brain Natriuretic Peptide Reduces Blood Pressure in Normotensive and Acute Norepinephrine-Induced Hypertensive Rabbits
Clemens, L.Edward, Almirez, Ramona G, Baudouin, Karine A, Grossbard, Elliott B, Protter, Andrew A
Published in American journal of hypertension (01.06.1997)
Published in American journal of hypertension (01.06.1997)
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Journal Article
A selective p38 alpha mitogen-activated protein kinase inhibitor reverses cartilage and bone destruction in mice with collagen-induced arthritis
Medicherla, Satyanarayana, Ma, Jing Ying, Mangadu, Ruban, Jiang, Yebin, Zhao, Jenny J, Almirez, Ramona, Kerr, Irene, Stebbins, Elizabeth G, O'Young, Gilbert, Kapoun, Ann M, Luedtke, Gregory, Chakravarty, Sarvajit, Dugar, Sundeep, Genant, Harry K, Protter, Andrew A
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
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Journal Article
Pharmacokinetics and Biological Actions of Subcutaneously Administered Human Brain Natriuretic Peptide
Clemens, L E, Almirez, R G, Baudouin, K A, Mischak, R P, Grossbard, E B, Protter, A A
Published in The Journal of pharmacology and experimental therapeutics (01.10.1998)
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Published in The Journal of pharmacology and experimental therapeutics (01.10.1998)
Journal Article
Transcutaneous Chemical Collection of Caffeine in Normal Subjects: Relationship to Area Under the Plasma Concentration-Time Curve and Sweat Production
Conner, Dale P, Millora, Emily, Zamani, Kaveh, Nix, Darrell, Almirez, Ramona G, Rhyne-Kirsch, Patricia, Peck, Carl C
Published in Journal of investigative dermatology (01.02.1991)
Published in Journal of investigative dermatology (01.02.1991)
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Journal Article
Antinociceptive action of a p38α MAPK inhibitor, SD-282, in a diabetic neuropathy model
Sweitzer, Sarah M., Medicherla, Satyanarayana, Almirez, Ramona, Dugar, Sundeep, Chakravarty, Sarvajit, Shumilla, Jennifer A., Yeomans, David C., Protter, Andrew A.
Published in Pain (Amsterdam) (01.06.2004)
Published in Pain (Amsterdam) (01.06.2004)
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Journal Article
Design and synthesis of piperazine-indole p38α MAP kinase inhibitors with improved pharmacokinetic profiles
Tan, Xuefei, Tester, Richland W., Luedtke, Gregory R., Chakravarty, Sarvajit, Mavunkel, Babu J., Perumattam, John J., Lu, Qing, Nashashibi, Imad, Jung, Joon, Hu, Jie, Liclican, Albert, Almirez, Ramona, Tabora, Jocelyn, Tran, Vinh, Laney, Maureen, Levy, Daniel E., Dugar, Sundeep
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Design and synthesis of piperazine-indole p38a MAP kinase inhibitors with improved pharmacokinetic profiles
Tan, Xuefei, Tester, Richland W, Luedtke, Gregory R, Chakravarty, Sarvajit, Mavunkel, Babu J, Perumattam, John J, Lu, Qing, Nashashibi, Imad, Jung, Joon, Hu, Jie, Liclican, Albert, Almirez, Ramona, Tabora, Jocelyn, Tran, Vinh, Laney, Maureen, Levy, Daniel E, Dugar, Sundeep
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Preventive and therapeutic potential of p38 alpha-selective mitogen-activated protein kinase inhibitor in nonobese diabetic mice with type 1 diabetes
Medicherla, Satyanarayana, Protter, Andrew A, Ma, Jing Ying, Mangadu, Ruban, Almirez, Ramona, Koppelman, Bruce, Kerr, Irene, Navas, Tony A, Movius, Fabiola, Reddy, Mamatha, Liu, Yu-Wang, Luedtke, Gregory, Perumattam, John, Mavunkel, Babu, Dugar, Sundeep, Schreiner, George F
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
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Journal Article
A Selective p38α Mitogen-Activated Protein Kinase Inhibitor Reverses Cartilage and Bone Destruction in Mice with Collagen-Induced Arthritis
Satyanarayana Medicherla, Jing Ying Ma, Ruban Mangadu, Yebin Jiang, Jenny J. Zhao, Ramona Almirez, Irene Kerr, Elizabeth G. Stebbins, Gilbert O'Young, Ann M. Kapoun, Gregory Luedtke, Sarvajit Chakravarty, Sundeep Dugar, Harry K. Genant, Andrew A. Protter
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
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Journal Article
Preventive and Therapeutic Potential of p38α-Selective Mitogen-Activated Protein Kinase Inhibitor in Nonobese Diabetic Mice with Type 1 Diabetes
Satyanarayana Medicherla, Andrew A. Protter, Jing Ying Ma, Ruban Mangadu, Ramona Almirez, Bruce Koppelman, Irene Kerr, Tony A. Navas, Fabiola Movius, Mamatha Reddy, Yu-Wang Liu, Gregory Luedtke, John Perumattam, Babu Mavunkel, Sundeep Dugar, George F. Schreiner
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
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Journal Article
Antinociceptive action of a p38alpha MAPK inhibitor, SD-282, in a diabetic neuropathy model
Sweitzer, Sarah M, Medicherla, Satyanarayana, Almirez, Ramona, Dugar, Sundeep, Chakravarty, Sarvajit, Shumilla, Jennifer A, Yeomans, David C, Protter, Andrew A
Published in Pain (Amsterdam) (01.06.2004)
Published in Pain (Amsterdam) (01.06.2004)
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Journal Article
B-type natriuretic peptide reduces cardiac remodeling and improves cardiac function post myocardial injury induced by L-NAME/Angiotensin II
Li, Zhihe, Mills, Scott, Liang, Faquang, Almirez, Ramona, O'Connell, Maile, Kapoun, Ann, Schreiner, George, Protter, Andy
Published in Journal of cardiac failure (01.08.2004)
Published in Journal of cardiac failure (01.08.2004)
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Journal Article
Pharmacological Properties of SD-282 – An α-Isoform Selective Inhibitor for p38 MAP Kinase
Koppelman, Bruce, Webb, Heather K., Medicherla, Satyanarayana, Almirez, Ramona, Feng, Ying, Chavez, Jose Carlos, Mao, Cheng Ping, Nguyen, Aaron, Liu, Yu-Wang, Kapoun, Ann M., Muiru, Gladys, Huang, Yuanying Anne, Dugar, Sundeep, Mavunkel, Babu J., Lim, Don W., Chakravarty, Sarvajit, Luedtke, Gregory, Protter, Andrew A., Higgins, Linda S.
Published in Pharmacology (01.01.2008)
Published in Pharmacology (01.01.2008)
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Journal Article
Pharmacological Properties of SD-282 - An [alpha]-Isoform Selective Inhibitor for p38 MAP Kinase
Koppelman, Bruce, Webb, Heather K, Medicherla, Satyanarayana, Almirez, Ramona, Feng, Ying, Chavez, Jose Carlos, Mao, Cheng Ping, Nguyen, Aaron, Liu, Yu-wang, Kapoun, Ann M, Muiru, Gladys, Huang, Yuanying Anne, Dugar, Sundeep, Mavunkel, Babu J, Lim, Don W, Chakravarty, Sarvajit, Luedtke, Gregory, Protter, Andrew A, Higgins, Linda S
Published in Pharmacology (01.03.2008)
Published in Pharmacology (01.03.2008)
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Journal Article
The effects of marijuana extract and ∆9-tetrahydrocannabinol on luteal function in the rhesus monkey
Almirez, Ramona G., Smith, Carol Grace, Asch, Ricardo H.
Published in Fertility and sterility (01.02.1983)
Published in Fertility and sterility (01.02.1983)
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