Ursolic acid derivatives as potential antidiabetic agents: In vitro, in vivo, and in silico studies
Guzmán‐Ávila, Ricardo, Flores‐Morales, Virginia, Paoli, Paolo, Camici, Guido, Ramírez‐Espinosa, Juan José, Cerón‐Romero, Litzia, Navarrete‐Vázquez, Gabriel, Hidalgo‐Figueroa, Sergio, Yolanda Rios, Maria, Villalobos‐Molina, Rafael, Estrada‐Soto, Samuel
Published in Drug development research (01.03.2018)
Published in Drug development research (01.03.2018)
Get full text
Journal Article
Synthesis, in vitro, in silico and in vivo hypoglycemic and lipid-lowering effects of 4-benzyloxy-5-benzylidene-1,3-thiazolidine-2,4-diones mediated by dual PPAR α/γ modulation
Madrigal-Angulo, José Luis, Ménez-Guerrero, Carlos, Estrada-Soto, Samuel, Ramírez-Espinosa, Juan José, Almanza-Pérez, Julio César, León-Rivera, Ismael, Hernández-Núñez, Emanuel, Aguirre-Vidal, Yoshajandith, Flores-León, Carlos D., Aguayo-Ortíz, Rodrigo, Navarrete-Vazquez, Gabriel
Published in Bioorganic & medicinal chemistry letters (15.08.2022)
Published in Bioorganic & medicinal chemistry letters (15.08.2022)
Get full text
Journal Article
Antidiabetic activity of some pentacyclic acid triterpenoids, role of PTP–1B: In vitro, in silico, and in vivo approaches
Ramírez-Espinosa, Juan José, Rios, Maria Yolanda, López-Martínez, Sugey, López-Vallejo, Fabian, Medina-Franco, José L., Paoli, Paolo, Camici, Guido, Navarrete-Vázquez, Gabriel, Ortiz-Andrade, Rolffy, Estrada-Soto, Samuel
Published in European journal of medicinal chemistry (01.06.2011)
Published in European journal of medicinal chemistry (01.06.2011)
Get full text
Journal Article
Chrysin Induces Antidiabetic, Antidyslipidemic and Anti-Inflammatory Effects in Athymic Nude Diabetic Mice
Ramírez-Espinosa, Juan José, Saldaña-Ríos, Johann, García-Jiménez, Sara, Villalobos-Molina, Rafael, Ávila-Villarreal, Gabriela, Rodríguez-Ocampo, Angélica Nallelhy, Bernal-Fernández, Germán, Estrada-Soto, Samuel
Published in Molecules (Basel, Switzerland) (28.12.2017)
Published in Molecules (Basel, Switzerland) (28.12.2017)
Get full text
Journal Article
Synthesis and In Vitro AMPK Activation of Cycloalkyl/Alkarylbiguanides with Robust In Vivo Antihyperglycemic Action
Navarrete-Vázquez, Gabriel, Estrada-Soto, Samuel, Carvajal, Karla, Centurión, David, Rivera-Leyva, Julio C., Ramírez-Espinosa, Juan José, Rosales-Ortega, Edgar, Martínez-Conde, Carlos, Gutierrez-Lara, Erika, Ortega-Cuellar, Daniel
Published in Journal of chemistry (2017)
Published in Journal of chemistry (2017)
Get full text
Journal Article
Vasorelaxant effect of Valeriana edulis ssp. procera (Valerianaceae) and its mode of action as calcium channel blocker
Estrada-Soto, Samuel, Rivera-Leyva, Julio, Ramírez-Espinosa, Juan José, Castillo-España, Patricia, Aguirre-Crespo, Francisco, Hernández-Abreu, Oswaldo
Published in Journal of pharmacy and pharmacology (01.09.2010)
Published in Journal of pharmacy and pharmacology (01.09.2010)
Get more information
Journal Article
Synthesis and molecular docking of N′-arylidene-5-(4-chlorophenyl)-1-(3,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carbohydrazides as novel hypoglycemic and antioxidant dual agents
Hernández-Vázquez, Eduardo, Salgado-Barrera, Sandybel, Ramírez-Espinosa, Juan José, Estrada-Soto, Samuel, Hernández-Luis, Francisco
Published in Bioorganic & medicinal chemistry (15.05.2016)
Published in Bioorganic & medicinal chemistry (15.05.2016)
Get full text
Journal Article
Synthesis and evaluation of thiazolidine-2,4-dione/benzazole derivatives as inhibitors of protein tyrosine phosphatase 1B (PTP-1B): Antihyperglycemic activity with molecular docking study
Hidalgo-Figueroa, Sergio, Estrada-Soto, Samuel, Ramírez-Espinosa, Juan José, Paoli, Paolo, Lori, Giulia, León-Rivera, Ismael, Navarrete-Vázquez, Gabriel
Published in Biomedicine & pharmacotherapy (01.11.2018)
Published in Biomedicine & pharmacotherapy (01.11.2018)
Get full text
Journal Article
Synthesis, hypoglycemic activity and molecular modeling studies of pyrazole-3-carbohydrazides designed by a CoMFA model
Hernández-Vázquez, Eduardo, Aguayo-Ortiz, Rodrigo, Ramírez-Espinosa, Juan José, Estrada-Soto, Samuel, Hernández-Luis, Francisco
Published in European journal of medicinal chemistry (01.11.2013)
Published in European journal of medicinal chemistry (01.11.2013)
Get full text
Journal Article
Synthesis of oleanolic acid derivatives: In vitro, in vivo and in silico studies for PTP-1B inhibition
Ramírez-Espinosa, Juan José, Rios, Maria Yolanda, Paoli, Paolo, Flores-Morales, Virginia, Camici, Guido, Rosa-Lugo, Vianey de la, Hidalgo-Figueroa, Sergio, Navarrete-Vázquez, Gabriel, Estrada-Soto, Samuel
Published in European journal of medicinal chemistry (24.11.2014)
Published in European journal of medicinal chemistry (24.11.2014)
Get full text
Journal Article
1,5-Diarylpyrazole and vanillin hybrids: Synthesis, biological activity and DFT studies
Hernández-Vázquez, Eduardo, Castañeda-Arriaga, Romina, Ramírez-Espinosa, Juan José, Medina-Campos, Omar Noel, Hernández-Luis, Francisco, Chaverri, José Pedraza, Estrada-Soto, Samuel
Published in European journal of medicinal chemistry (15.07.2015)
Published in European journal of medicinal chemistry (15.07.2015)
Get full text
Journal Article
Synthesis, in vitro and in silico studies of a PPARγ and GLUT-4 modulator with hypoglycemic effect
Navarrete-Vázquez, Gabriel, Torres-Gómez, Héctor, Hidalgo-Figueroa, Sergio, Ramírez-Espinosa, Juan José, Estrada-Soto, Samuel, Medina-Franco, José L., León-Rivera, Ismael, Alarcón-Aguilar, Francisco Javier, Almanza-Pérez, Julio César
Published in Bioorganic & medicinal chemistry letters (15.09.2014)
Published in Bioorganic & medicinal chemistry letters (15.09.2014)
Get full text
Journal Article
Synthesis of 2-{2-[(α/β-naphthalen-1-ylsulfonyl)amino]-1,3-thiazol-4-yl} acetamides with 11β-hydroxysteroid dehydrogenase inhibition and in combo antidiabetic activities
Navarrete-Vázquez, Gabriel, Morales-Vilchis, Maria Guadalupe, Estrada-Soto, Samuel, Ramírez-Espinosa, Juan José, Hidalgo-Figueroa, Sergio, Nava-Zuazo, Carlos, Tlahuext, Hugo, Leon-Rivera, Ismael, Medina-Franco, José L., López-Vallejo, Fabian, Webster, Scott P., Binnie, Margaret, Ortiz-Andrade, Rolffy, Moreno-Diaz, Hermenegilda
Published in European journal of medicinal chemistry (03.03.2014)
Published in European journal of medicinal chemistry (03.03.2014)
Get full text
Journal Article
Antihyperglycemic and sub-chronic antidiabetic actions of morolic and moronic acids, in vitro and in silico inhibition of 11β-HSD 1
Ramírez-Espinosa, Juan José, García-Jiménez, Sara, Rios, Maria Yolanda, Medina-Franco, José L., López-Vallejo, Fabián, Webster, Scott P., Binnie, Margareth, Ibarra-Barajas, Maximiliano, Ortiz-Andrade, Rolffy, Estrada-Soto, Samuel
Published in Phytomedicine (Stuttgart) (15.05.2013)
Published in Phytomedicine (Stuttgart) (15.05.2013)
Get full text
Journal Article