Evaluation of Anti-Inflammatory Properties of Isoorientin Isolated from Tubers of Pueraria tuberosa
Pallu, Reddanna, Srivastava, Anand, Dharmapuri, Gangappa, Yarla, Nagendra Sastry, Azad, Rajaram, Reddy, Gorla V., Anilkumar, Kotha, Kamal, Mohammad Amjad
Published in Oxidative medicine and cellular longevity (01.01.2017)
Published in Oxidative medicine and cellular longevity (01.01.2017)
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Design, synthesis, biological evaluation and in silico studies of EGFR inhibitors based on 4-oxo-chromane scaffold targeting resistance in non-small cell lung cancer (NSCLC)
Karnik, Kshipra S., Sarkate, Aniket P., Tiwari, Shailee V., Azad, Rajaram, Wakte, Pravin S.
Published in Medicinal chemistry research (01.09.2022)
Published in Medicinal chemistry research (01.09.2022)
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Efficient Synthesis of Densely Functionalized Pyrido[2,3-d]Pyrimidines via Three-component One-pot Domino Knoevenagel aza-Diels Alder Reaction and Induces Apoptosis in Human Cancer Cell Lines via Inhibiting Aurora A and B Kinases
Bhosle, Manisha R., Palke, Amruta, Bondle, Giribala M., Sarkate, Aniket P., Azad, Rajaram, Burra, Prasad V. L. S.
Published in Polycyclic aromatic compounds (21.10.2023)
Published in Polycyclic aromatic compounds (21.10.2023)
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N-Benzylation of 6-aminoflavone by reductive amination and efficient access to some novel anticancer agents via topoisomerase II inhibition
Thorat, Nitin M., Sarkate, Aniket P., Lokwani, Deepak K., Tiwari, Shailee V., Azad, Rajaram, Thopate, Shankar R.
Published in Molecular diversity (01.05.2021)
Published in Molecular diversity (01.05.2021)
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Green synthesis and inhibitory effect of novel quinoline based thiazolidinones on the growth of MCF-7 human breast cancer cell line by G2/M cell cycle arrest
Dofe, Vidya S., Sarkate, Aniket P., Azad, Rajaram, Gill, Charansingh H.
Published in Research on chemical intermediates (01.02.2018)
Published in Research on chemical intermediates (01.02.2018)
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5-Lipoxygenase and cyclooxygenase inhibitory dammarane triterpenoid 1 from Borassus flabellifer seed coat inhibits tumor necrosis factor-α secretion in LPSInduced THP-1 human monocytes and induces apoptosis in MIA PaCa-2 pancreatic cancer cells
Yarla, Nagendra Sastry, Azad, Rajaram, Basha, Mahaboob, Rajack, Abdul, Kaladhar, D S V G K, Allam, Bharat Kumar, Pragada, Rajeswara Rao, Singh, Krishna Nand, K, Sunanda Kumari, Pallu, Reddanna, Parimi, Umadevi, Bishayee, Anupam, Duddukuri, Govinda Rao
Published in Anti-cancer agents in medicinal chemistry (01.08.2015)
Published in Anti-cancer agents in medicinal chemistry (01.08.2015)
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Anti-inflammatory profile of Aegle marmelos (L) Correa (Bilva) with special reference to young roots grown in different parts of India
Rajaram, Azad, Vanaja, G.R., Vyakaranam, Preeti, Rachamallu, Aparna, Reddy, Gorla V., Anilkumar, Kotha, Arunasree, Kalle M., Dhyani, Anurag, Prasad, Narapureddy Krishna, Sharma, Sakshee, Chandra Joshi, Mahesh, Kimothi, Gaya Prasad, Brindavanam, N.B., Reddanna, Pallu
Published in Journal of ayurveda and integrative medicine (01.04.2018)
Published in Journal of ayurveda and integrative medicine (01.04.2018)
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Design, synthesis, and biological evaluation of novel quinoline derivatives as small molecule mutant EGFR inhibitors targeting resistance in NSCLC: In vitro screening and ADME predictions
Kardile, Ramakant A., Sarkate, Aniket P., Lokwani, Deepak K., Tiwari, Shailee V., Azad, Rajaram, Thopate, Shankar R.
Published in European journal of medicinal chemistry (05.01.2023)
Published in European journal of medicinal chemistry (05.01.2023)
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Free energy perturbation guided Synthesis with Biological Evaluation of Substituted Quinoline derivatives as small molecule L858R/T790M/C797S mutant EGFR inhibitors targeting resistance in Non-Small Cell Lung Cancer (NSCLC)
Karnik, Kshipra S., Sarkate, Aniket P., Tiwari, Shailee V., Azad, Rajaram, Wakte, Pravin S.
Published in Bioorganic chemistry (01.10.2021)
Published in Bioorganic chemistry (01.10.2021)
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Design and synthesis of novel conformationally constrained 7,12-dihydro- dibenzo[b,h][1,6] naphthyridine and 7H-Chromeno[3,2-c] quinoline derivatives as topoisomerase I inhibitors: In vitro screening, molecular docking and ADME predictions
Kardile, Ramakant A., Sarkate, Aniket P., Borude, Avinash S., Mane, Rajendra S., Lokwani, Deepak K., Tiwari, Shailee, Azad, Rajaram, Burra, Prasad V. L. S., Thopate, Shankar R.
Published in Bioorganic chemistry (01.10.2021)
Published in Bioorganic chemistry (01.10.2021)
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New amide linked dimeric 1,2,3-triazoles bearing aryloxy scaffolds as a potent antiproliferative agents and EGFR tyrosine kinase phosphorylation inhibitors
Deshmukh, Tejshri R., Sarkate, Aniket P., Lokwani, Deepak K., Tiwari, Shailee V., Azad, Rajaram, Shingate, Bapurao B.
Published in Bioorganic & medicinal chemistry letters (01.10.2019)
Published in Bioorganic & medicinal chemistry letters (01.10.2019)
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Computational and Synthetic approach with Biological Evaluation of Substituted Quinoline derivatives as small molecule L858R/T790M/C797S triple mutant EGFR inhibitors targeting resistance in Non-Small Cell Lung Cancer (NSCLC)
Karnik, Kshipra S., Sarkate, Aniket P., Tiwari, Shailee V., Azad, Rajaram, Burra, Prasad V.L.S., Wakte, Pravin S.
Published in Bioorganic chemistry (01.02.2021)
Published in Bioorganic chemistry (01.02.2021)
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Molecular dynamic simulations based discovery and development of thiazolidin-4-one derivatives as EGFR inhibitors targeting resistance in non-small cell lung cancer (NSCLC)
Karnik, Kshipra S., Sarkate, Aniket P., Lokwani, Deepak K., Tiwari, Shailee V., Azad, Rajaram, Wakte, Pravin S.
Published in Journal of biomolecular structure & dynamics (03.07.2023)
Published in Journal of biomolecular structure & dynamics (03.07.2023)
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Betulinic acid derivatives: a new class of α-glucosidase inhibitors and LPS-stimulated nitric oxide production inhibition on mouse macrophage RAW 264.7 cells
Gundoju, Narayanarao, Bokam, Ramesh, Yalavarthi, Nageswara Rao, Azad, Rajaram, Ponnapalli, Mangala Gowri
Published in Natural product research (17.09.2019)
Published in Natural product research (17.09.2019)
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Synthesis and evaluation of novel sulfonamide analogues of 6/7-aminoflavones as anticancer agents via topoisomerase II inhibition
Shelke, Rohini N., Pansare, Dattatraya N., Sarkate, Aniket P., Narula, Ishudeep K., Lokwani, Deepak K., Tiwari, Shailee V., Azad, Rajaram, Thopate, Shankar R.
Published in Bioorganic & medicinal chemistry letters (15.07.2020)
Published in Bioorganic & medicinal chemistry letters (15.07.2020)
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Synthesis and pharmacological evaluation of pyrazolo[4,3-c]cinnoline derivatives as potential anti-inflammatory and antibacterial agents
Tonk, Rajiv Kumar, Bawa, Sandhya, Chawla, Gita, Deora, Girdhar Singh, Kumar, Suresh, Rathore, Vandana, Mulakayala, Naveen, Rajaram, Azad, Kalle, Arunasree M., Afzal, Obaid
Published in European journal of medicinal chemistry (01.11.2012)
Published in European journal of medicinal chemistry (01.11.2012)
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