Improving oral bioavailability of cyclic peptides by N-methylation
Räder, Andreas F.B., Reichart, Florian, Weinmüller, Michael, Kessler, Horst
Published in Bioorganic & medicinal chemistry (01.06.2018)
Published in Bioorganic & medicinal chemistry (01.06.2018)
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Journal Article
Orally Active Peptides: Is There a Magic Bullet?
Räder, Andreas F. B., Weinmüller, Michael, Reichart, Florian, Schumacher‐Klinger, Adi, Merzbach, Shira, Gilon, Chaim, Hoffman, Amnon, Kessler, Horst
Published in Angewandte Chemie International Edition (26.10.2018)
Published in Angewandte Chemie International Edition (26.10.2018)
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Journal Article
Selective Targeting of Integrin alpha v beta 8 by a Highly Active Cyclic Peptide
Reichart, Florian, Maltsev, Oleg V., Kapp, Tobias G., Raeder, Andreas F. B., Weinmueller, Michael, Marelli, Udaya Kiran, Notni, Johannes, Wurzer, Alexander, Beck, Roswitha, Wester, Hans Juergen, Steiger, Katja, Di Maro, Salvatore, Di Leva, Francesco Saverio, Marinelli, Luciana, Nieberler, Markus, Reuning, Ute, Schwaiger, Markus, Kessler, Horst
Published in Journal of medicinal chemistry (28.02.2019)
Published in Journal of medicinal chemistry (28.02.2019)
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Journal Article
Bioconjugation of Supramolecular Metallacages to Integrin Ligands for Targeted Delivery of Cisplatin
Han, Jiaying, Räder, Andreas F. B, Reichart, Florian, Aikman, Brech, Wenzel, Margot N, Woods, Ben, Weinmüller, Michael, Ludwig, Beatrice S, Stürup, Stefan, Groothuis, Geny M. M, Permentier, Hjalmar P, Bischoff, Rainer, Kessler, Horst, Horvatovich, Peter, Casini, Angela
Published in Bioconjugate chemistry (21.11.2018)
Published in Bioconjugate chemistry (21.11.2018)
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Journal Article
N-Methylation of isoDGR Peptides: Discovery of a Selective alpha 5 beta 1-Integrin Ligand as a Potent Tumor Imaging Agent
Kapp, Tobias G., Di Leva, Francesco Saverio, Notni, Johannes, Raeder, Andreas F. B., Fottner, Maximilian, Reichart, Florian, Reich, Dominik, Wurzer, Alexander, Steiger, Katja, Novellino, Ettore, Marelli, Udaya Kiran, Wester, Hans-Juergen, Marinelli, Luciana, Kessler, Horst
Published in Journal of medicinal chemistry (22.03.2018)
Published in Journal of medicinal chemistry (22.03.2018)
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Journal Article
Enhancing Oral Bioavailability of Cyclic RGD Hexa-peptides by the Lipophilic Prodrug Charge Masking Approach: Redirection of Peptide Intestinal Permeability from a Paracellular to Transcellular Pathway
Schumacher-Klinger, Adi, Fanous, Joseph, Merzbach, Shira, Weinmüller, Michael, Reichart, Florian, Räder, Andreas F. B, Gitlin-Domagalska, Agata, Gilon, Chaim, Kessler, Horst, Hoffman, Amnon
Published in Molecular pharmaceutics (06.08.2018)
Published in Molecular pharmaceutics (06.08.2018)
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Journal Article
Tertiary Alcohols as Substrates for SN2-Like Stereoinversion
Räder, Andreas F. B., Tiefenbacher, Konrad
Published in Angewandte Chemie (International ed.) (27.01.2014)
Published in Angewandte Chemie (International ed.) (27.01.2014)
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Journal Article
Tertiary Alcohols as Substrates for S sub(N)2-Like Stereoinversion
Raeder, Andreas FB, Tiefenbacher, Konrad
Published in Angewandte Chemie International Edition (01.01.2014)
Published in Angewandte Chemie International Edition (01.01.2014)
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Journal Article
Lösung des Problems mangelnder oraler Verfugbarkeit cyclischer Hexapeptide: Entwicklung eines selektiven, oral verfugbaren Liganden fur das Integrin[alpha]v[beta]3
Weinmuller, Michael, Rechenmacher, Florian, KiranMarelli, Udaya, Reichart, Florian, Kapp, Tobias G, Rader, Andreas F B, DiLeva, Francesco Saverio, Marinelli, Luciana, Novellino, Ettore, Munoz-Felix, José M, Hodivala-Dilke, Kairbaan, Schumacher, Adi, Fanous, Joseph, Gilon, Chaim, Hoffman, Amnon, Kessler, Horst
Published in Angewandte Chemie (18.12.2017)
Published in Angewandte Chemie (18.12.2017)
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Journal Article
Oral aktive Peptide: Gibt es ein Patentrezept?
Räder, Andreas F. B., Weinmüller, Michael, Reichart, Florian, Schumacher‐Klinger, Adi, Merzbach, Shira, Gilon, Chaim, Hoffman, Amnon, Kessler, Horst
Published in Angewandte Chemie (26.10.2018)
Published in Angewandte Chemie (26.10.2018)
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Journal Article