ChEMBL: towards direct deposition of bioassay data
Mendez, David, Gaulton, Anna, Bento, A Patrícia, Chambers, Jon, De Veij, Marleen, Félix, Eloy, Magariños, María Paula, Mosquera, Juan F, Mutowo, Prudence, Nowotka, Michał, Gordillo-Marañón, María, Hunter, Fiona, Junco, Laura, Mugumbate, Grace, Rodriguez-Lopez, Milagros, Atkinson, Francis, Bosc, Nicolas, Radoux, Chris J, Segura-Cabrera, Aldo, Hersey, Anne, Leach, Andrew R
Published in Nucleic acids research (08.01.2019)
Published in Nucleic acids research (08.01.2019)
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Bispecific repurposed medicines targeting the viral and immunological arms of COVID-19
Redhead, Martin A., Owen, C. David, Brewitz, Lennart, Collette, Amelia H., Lukacik, Petra, Strain-Damerell, Claire, Robinson, Sean W., Collins, Patrick M., Schäfer, Philipp, Swindells, Mark, Radoux, Chris J., Hopkins, Iva Navratilova, Fearon, Daren, Douangamath, Alice, von Delft, Frank, Malla, Tika R., Vangeel, Laura, Vercruysse, Thomas, Thibaut, Jan, Leyssen, Pieter, Nguyen, Tu-Trinh, Hull, Mitchell, Tumber, Anthony, Hallett, David J., Schofield, Christopher J., Stuart, David I., Hopkins, Andrew L., Walsh, Martin A.
Published in Scientific reports (24.06.2021)
Published in Scientific reports (24.06.2021)
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The druggable genome: Twenty years later
Radoux, Chris J., Vianello, Francesca, McGreig, Jake, Desai, Nikita, Bradley, Anthony R.
Published in Frontiers in bioinformatics (30.09.2022)
Published in Frontiers in bioinformatics (30.09.2022)
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Publisher Correction: Bispecific repurposed medicines targeting the viral and immunological arms of COVID-19
Redhead, Martin A., Owen, C. David, Brewitz, Lennart, Collette, Amelia H., Lukacik, Petra, Strain-Damerell, Claire, Robinson, Sean W., Collins, Patrick M., Schäfer, Philipp, Swindells, Mark, Radoux, Chris J., Hopkins, Iva Navratilova, Fearon, Daren, Douangamath, Alice, von Delft, Frank, Malla, Tika R., Vangeel, Laura, Vercruysse, Thomas, Thibaut, Jan, Leyssen, Pieter, Nguyen, Tu-Trinh, Hull, Mitchell, Tumber, Anthony, Hallett, David J., Schofield, Christopher J., Stuart, David I., Hopkins, Andrew L., Walsh, Martin A.
Published in Scientific reports (28.09.2021)
Published in Scientific reports (28.09.2021)
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The PROTACtable genome
Schneider, Melanie, Radoux, Chris J, Hercules, Andrew, Ochoa, David, Dunham, Ian, Zalmas, Lykourgos-Panagiotis, Hessler, Gerhard, Ruf, Sven, Shanmugasundaram, Veerabahu, Hann, Michael M, Thomas, Pam J, Queisser, Markus A, Benowitz, Andrew B, Brown, Kris, Leach, Andrew R
Published in Nature reviews. Drug discovery (01.10.2021)
Published in Nature reviews. Drug discovery (01.10.2021)
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Target-Based Evaluation of “Drug-Like” Properties and Ligand Efficiencies
Leeson, Paul D, Bento, A. Patricia, Gaulton, Anna, Hersey, Anne, Manners, Emma J, Radoux, Chris J, Leach, Andrew R
Published in Journal of medicinal chemistry (10.06.2021)
Published in Journal of medicinal chemistry (10.06.2021)
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Identifying Interactions that Determine Fragment Binding at Protein Hotspots
Radoux, Chris J, Olsson, Tjelvar S. G, Pitt, Will R, Groom, Colin R, Blundell, Tom L
Published in Journal of medicinal chemistry (12.05.2016)
Published in Journal of medicinal chemistry (12.05.2016)
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Fragment Hotspot Mapping to Identify Selectivity-Determining Regions between Related Proteins
Smilova, Mihaela D, Curran, Peter R, Radoux, Chris J, von Delft, Frank, Cole, Jason C, Bradley, Anthony R, Marsden, Brian D
Published in Journal of chemical information and modeling (24.01.2022)
Published in Journal of chemical information and modeling (24.01.2022)
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Hotspots API: A Python Package for the Detection of Small Molecule Binding Hotspots and Application to Structure-Based Drug Design
Curran, Peter R, Radoux, Chris J, Smilova, Mihaela D, Sykes, Richard A, Higueruelo, Alicia P, Bradley, Anthony R, Marsden, Brian D, Spring, David R, Blundell, Tom L, Leach, Andrew R, Pitt, William R, Cole, Jason C
Published in Journal of chemical information and modeling (27.04.2020)
Published in Journal of chemical information and modeling (27.04.2020)
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