Functionalization of Carbon Nanoparticles Modulates Inflammatory Cell Recruitment and NLRP3 Inflammasome Activation
Yang, Marie, Flavin, Kevin, Kopf, Ilona, Radics, Gabor, Hearnden, Claire H. A., McManus, Gavin J., Moran, Barry, Villalta-Cerdas, Adrian, Echegoyen, Luis A., Giordani, Silvia, Lavelle, Ed C.
Published in Small (Weinheim an der Bergstrasse, Germany) (20.12.2013)
Published in Small (Weinheim an der Bergstrasse, Germany) (20.12.2013)
Get full text
Journal Article
Structure-Guided Discovery of a Selective Mcl‑1 Inhibitor with Cellular Activity
Szlávik, Zoltan, Ondi, Levente, Csékei, Márton, Paczal, Attila, Szabó, Zoltán B, Radics, Gábor, Murray, James, Davidson, James, Chen, Ijen, Davis, Ben, Hubbard, Roderick E, Pedder, Christopher, Dokurno, Pawel, Surgenor, Allan, Smith, Julia, Robertson, Alan, LeToumelin-Braizat, Gaetane, Cauquil, Nicolas, Zarka, Marion, Demarles, Didier, Perron-Sierra, Francoise, Claperon, Audrey, Colland, Frederic, Geneste, Olivier, Kotschy, András
Published in Journal of medicinal chemistry (08.08.2019)
Published in Journal of medicinal chemistry (08.08.2019)
Get full text
Journal Article
New highly toxic bile acids derived from deoxycholic acid, chenodeoxycholic acid and lithocholic acid
Májer, Ferenc, Sharma, Ruchika, Mullins, Claire, Keogh, Luke, Phipps, Sinead, Duggan, Shane, Kelleher, Dermot, Keely, Stephen, Long, Aideen, Radics, Gábor, Wang, Jun, Gilmer, John F.
Published in Bioorganic & medicinal chemistry (01.01.2014)
Published in Bioorganic & medicinal chemistry (01.01.2014)
Get full text
Journal Article
The MCL1 inhibitor S63845 is tolerable and effective in diverse cancer models
Kotschy, András, Szlavik, Zoltán, Murray, James, Davidson, James, Maragno, Ana Leticia, Le Toumelin-Braizat, Gaëtane, Chanrion, Maïa, Kelly, Gemma L., Gong, Jia-Nan, Moujalled, Donia M., Bruno, Alain, Csekei, Márton, Paczal, Attila, Szabo, Zoltán B., Sipos, Szabolcs, Radics, Gábor, Proszenyak, Agnes, Balint, Balázs, Ondi, Levente, Blasko, Gábor, Robertson, Alan, Surgenor, Allan, Dokurno, Pawel, Chen, Ijen, Matassova, Natalia, Smith, Julia, Pedder, Christopher, Graham, Christopher, Studeny, Aurélie, Lysiak-Auvity, Gaëlle, Girard, Anne-Marie, Gravé, Fabienne, Segal, David, Riffkin, Chris D., Pomilio, Giovanna, Galbraith, Laura C. A., Aubrey, Brandon J., Brennan, Margs S., Herold, Marco J., Chang, Catherine, Guasconi, Ghislaine, Cauquil, Nicolas, Melchiore, Fabien, Guigal-Stephan, Nolwen, Lockhart, Brian, Colland, Frédéric, Hickman, John A., Roberts, Andrew W., Huang, David C. S., Wei, Andrew H., Strasser, Andreas, Lessene, Guillaume, Geneste, Olivier
Published in Nature (London) (27.10.2016)
Published in Nature (London) (27.10.2016)
Get full text
Journal Article
Discovery of S64315, a Potent and Selective Mcl‑1 Inhibitor
Szlavik, Zoltan, Csekei, Marton, Paczal, Attila, Szabo, Zoltan B, Sipos, Szabolcs, Radics, Gabor, Proszenyak, Agnes, Balint, Balazs, Murray, James, Davidson, James, Chen, Ijen, Dokurno, Pawel, Surgenor, Allan E, Daniels, Zoe Marie, Hubbard, Roderick E, Le Toumelin-Braizat, Gaëtane, Claperon, Audrey, Lysiak-Auvity, Gaëlle, Girard, Anne-Marie, Bruno, Alain, Chanrion, Maia, Colland, Frédéric, Maragno, Ana-Leticia, Demarles, Didier, Geneste, Olivier, Kotschy, Andras
Published in Journal of medicinal chemistry (25.11.2020)
Published in Journal of medicinal chemistry (25.11.2020)
Get full text
Journal Article
Orthogonally protected, carboxy-activated L-homoisoserine, 2-methyl-L-homoisoserine, and homoisocysteine derivatives. New building blocks for peptide and depsipeptide modification
Burger, K, Radics, G, Hennig, L, Bottcher, C, Spengler, J, Albericio, F
Published in Monatshefte für Chemie (01.05.2005)
Published in Monatshefte für Chemie (01.05.2005)
Get full text
Journal Article
A fluorescent analogue of tauroursodeoxycholic acid reduces ER stress and is cytoprotective
Gavin, Jason, Quilty, Fran, Majer, Ferenc, Gilsenan, Georgina, Byrne, Anne Marie, Long, Aideen, Radics, Gabor, Gilmer, John F.
Published in Bioorganic & medicinal chemistry letters (01.11.2016)
Published in Bioorganic & medicinal chemistry letters (01.11.2016)
Get full text
Journal Article
Novel Iron-Whey Protein Microspheres Protect Gut Epithelial Cells from Iron-Related Oxidative Stress and Damage and Improve Iron Absorption in Fasting Adults
Wang, Jun, Radics, Gabor, Whelehan, Michael, OʼDriscoll, Aoibhe, Healy, Anne Marie, Gilmer, John F, Ledwidge, Mark
Published in Acta haematologica (01.01.2017)
Published in Acta haematologica (01.01.2017)
Get more information
Journal Article
Design, Synthesis, and Pharmacological Effects of a Cyclization-Activated Steroid Prodrug for Colon Targeting in Inflammatory Bowel Disease
Ruiz, Juan F. Márquez, Radics, Gabor, Windle, Henry, Serra, Hugo O, Simplício, Ana Luísa, Kedziora, Kinga, Fallon, Padraic G, Kelleher, Dermot P, Gilmer, John F
Published in Journal of medicinal chemistry (28.05.2009)
Published in Journal of medicinal chemistry (28.05.2009)
Get full text
Journal Article
Carbon Nanotubes: Functionalization of Carbon Nanoparticles Modulates Inflammatory Cell Recruitment and NLRP3 Inflammasome Activation (Small 24/2013)
Yang, Marie, Flavin, Kevin, Kopf, Ilona, Radics, Gabor, Hearnden, Claire H. A., McManus, Gavin J., Moran, Barry, Villalta-Cerdas, Adrian, Echegoyen, Luis A., Giordani, Silvia, Lavelle, Ed C.
Published in Small (Weinheim an der Bergstrasse, Germany) (20.12.2013)
Published in Small (Weinheim an der Bergstrasse, Germany) (20.12.2013)
Get full text
Journal Article
신규한 아미노산 유도체, 이의 제조방법, 및 이를 함유한 약제 조성물
SZLAVIK ZOLTAN, CHEN I JEN, CSEKEI MARTON, ONDI LEVENTE, RADICS GABOR, KOTSCHY ANDRAS, PACZAL ATTILA, PROSZENYAK AGNES, SZABO ZOLTAN, GENESTE OLIVIER, BALINT BALAZS, SIPOS SZABOLCS, MURRAY JAMES BROOKE, BRUNO ALAIN, DAVIDSON JAMES EDWARD PAUL, PERRON SIERRA FRANCOISE
Year of Publication 12.02.2018
Get full text
Year of Publication 12.02.2018
Patent
NEW THIENOPYRIMIDINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
SZLAVIK ZOLTAN, CHEN I JEN, CSEKEI MARTON, RADICS GABOR, KOTSCHY ANDRAS, PACZAL ATTILA, PROSZENYAK AGNES, SZABO ZOLTAN, BALINT BALAZS, GENESTE OLIVIER, SIPOS SZABOLCS, MURRAY JAMES BROOKE, BRUNO ALAIN, DAVIDSON JAMES EDWARD PAUL, PERRON SIERRA FRANCOISE
Year of Publication 01.07.2015
Get full text
Year of Publication 01.07.2015
Patent
Hexafluoroacetone as a protecting and activating reagent: 5,5-difluoro- and trans-5-fluoropipecolic acids from glutamic acid
Golubev, AS, Schedel, H, Radics, G, Fioroni, M, Thust, S, Burger, K
Published in Tetrahedron letters (09.02.2004)
Published in Tetrahedron letters (09.02.2004)
Get full text
Journal Article
COMPOSITIONS AND METHODS FOR INCREASING IRON INTAKE IN A MAMMAL
GILMER, JOHN, WANG, JUN, GABOR, RADICS, O'FLYNN, PAT, LEDWIDGE, MARK, WHELEHAN, MICHAEL
Year of Publication 05.12.2023
Get full text
Year of Publication 05.12.2023
Patent
COMPOSITIONS AND METHODS FOR INCREASING IRON INTAKE IN A MAMMAL
GILMER, JOHN, WANG, JUN, GABOR, RADICS, O'FLYNN, PAT, WHELEHAN, MICHAEL, LEDWIDGE, PAT
Year of Publication 19.04.2023
Get full text
Year of Publication 19.04.2023
Patent
Stereoselective syntheses of 4-fluoro- and 4,4-difluoropipecolic acids
Golubev, Alexander S, Schedel, Hartmut, Radics, Gabor, Sieler, Joachim, Burger, Klaus
Published in Tetrahedron letters (05.11.2001)
Published in Tetrahedron letters (05.11.2001)
Get full text
Journal Article
COMPOSITIONS AND METHODS FOR INCREASING IRON INTAKE IN MAMMAL
O'FLYNN, Pat, WHELEHAN, Michael, WANG, Jun, LEDWIDGE, Mark, GABOR, Radics, GILMER, John
Year of Publication 12.12.2022
Get full text
Year of Publication 12.12.2022
Patent
Compositions and methods for increasing iron intake in a mammal
Gilmer, John, Wang, Jun, Gabor, Radics, Ledwidge, Mark, O'flynn, Pat, Whelehan, Michael
Year of Publication 25.11.2022
Get full text
Year of Publication 25.11.2022
Patent
Compositions and methods for increasing iron intake in a mammal
Gilmer, John, Gabor, Radics, Wang, Jun, Ledwidge, Mark, Whelehan, Michael, O'Flynn, Pat
Year of Publication 06.10.2022
Get full text
Year of Publication 06.10.2022
Patent