Practical Asymmetric Synthesis of Efavirenz (DMP 266), an HIV-1 Reverse Transcriptase Inhibitor
Pierce, Michael E, Parsons, Rodney L, Radesca, Lilian A, Lo, Young S, Silverman, Stuart, Moore, James R, Islam, Qamrul, Choudhury, Anusuya, Fortunak, Joseph M. D, Nguyen, Dieu, Luo, Chi, Morgan, Susan J, Davis, Wayne P, Confalone, Pat N, Chen, Cheng-yi, Tillyer, Richard D, Frey, Lisa, Tan, Lushi, Xu, Feng, Zhao, Dalian, Thompson, Andrew S, Corley, Edward G, Grabowski, Edward J. J, Reamer, Robert, Reider, Paul J
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Published in Journal of organic chemistry (13.11.1998)
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Stereoselective Process for a CCR3 Antagonist
Yue, Tai-Yuen, McLeod, Douglas D, Albertson, Kevin B, Beck, Steven R, Deerberg, Joerg, Fortunak, Joseph M, Nugent, William A, Radesca, Lilian A, Tang, Liya, Xiang, Cathie Dong
Published in Organic process research & development (01.03.2006)
Published in Organic process research & development (01.03.2006)
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Stereoselective Synthesis of HIV-1 Protease Inhibitor, DMP 323
Pierce, Michael E, Harris, Gregory D, Islam, Qamrul, Radesca, Lilian A, Storace, Louis, Waltermire, Robert E, Wat, Ed, Jadhav, Prabhakar K, Emmett, George C
Published in Journal of organic chemistry (26.01.1996)
Published in Journal of organic chemistry (26.01.1996)
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Synthesis, characterization, and biological evaluation of a novel class of N-(arylethyl)-N-alkyl-2-(1-pyrrolidinyl)ethylamines: structural requirements and binding affinity at the .sigma. receptor
De Costa, Brian R, Radesca, Lilian, Di Paolo, Lisa, Bowen, Wayne D
Published in Journal of medicinal chemistry (01.01.1992)
Published in Journal of medicinal chemistry (01.01.1992)
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Synthesis and receptor binding of enantiomeric N-substituted cis-N-[2-(3,4-dichlorophenyl)ethyl]-2-(1-pyrrolidinyl)cyclohexylamines as high-affinity .sigma. receptor ligands
Radesca, Lilian, Bowen, Wayne D, Di Paolo, Lisa, De Costa, Brian R
Published in Journal of medicinal chemistry (01.10.1991)
Published in Journal of medicinal chemistry (01.10.1991)
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METHODS FOR PREPARING MAYTANSINOID DERIVATIVES WITH SELF-IMMOLATIVE PEPTIDE LINKERS
RADESCA, Lilian, CAMERON, Mark, HAGUE, Andrew, AHMED, Ijaz, OH, Lynette
Year of Publication 21.03.2024
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Year of Publication 21.03.2024
Patent
Development of Novel, Potent, and Selective Dopamine Reuptake Inhibitors through Alteration of the Piperazine Ring of 1-[2-(Diphenylmethoxy)ethyl]- and 1-[2-[Bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazines (GBR 12935 and GBR 12909)
Matecka, Dorota, Rothman, Richard B, Radesca, Lilian, de Costa, Brian R, Dersch, Christina M, Partilla, John S, Pert, Agu, Glowa, John R, Wojnicki, Francis H. E, Rice, Kenner C
Published in Journal of medicinal chemistry (22.11.1996)
Published in Journal of medicinal chemistry (22.11.1996)
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Journal Article
Synthesis of HIV-1 Reverse Transcriptase Inhibitor DMP 266
Radesca, Lilian A., Lo†, Young S., Moore, James R., Pierce, Michael E.
Published in Synthetic communications (01.12.1997)
Published in Synthetic communications (01.12.1997)
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Synthesis and biological evaluation of conformationally restricted 2-(1-pyrrolidinyl)-N-[2-(3,4-dichlorophenyl)ethyl]-N-methylethylenediamines as .sigma. receptor ligands. 1. Pyrrolidine, piperidine, homopiperidine, and tetrahydroisoquinoline classes
De Costa, Brian R, Dominguez, Celia, He, Xiao Shu, Williams, Wanda, Radesca, Lilian, Bowen, Wayne
Published in Journal of medicinal chemistry (01.11.1992)
Published in Journal of medicinal chemistry (01.11.1992)
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Synthesis and receptor binding properties of fluoro- and iodo-substituted high-affinity .sigma.-receptor ligands: identification of potential PET and SPECT .sigma.-receptor imaging agents
De Costa, Brian, Radesca, Lilian, Dominguez, Celia, Di Paolo, Lisa, Bowen, Wayne D
Published in Journal of medicinal chemistry (01.06.1992)
Published in Journal of medicinal chemistry (01.06.1992)
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Synthesis and evaluation of N-substituted cis-N-methyl-2-(1-pyrrolidinyl)cyclohexylamines as high affinity .sigma. receptor ligands. Identification of a new class of highly potent and selective .sigma. receptor probes
De Costa, Brian R, Bowen, Wayne D, Thurkauf, Andrew, Finn, Daniel T, Vazirani, Sondra, Rothman, Richard B, Band, Linda, Contreras, Patricia C, Gray, Nancy M
Published in Journal of medicinal chemistry (01.11.1990)
Published in Journal of medicinal chemistry (01.11.1990)
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