Structure-based development of new RAS-effector inhibitors from a combination of active and inactive RAS-binding compounds
Cruz-Migoni, Abimael, Canning, Peter, Quevedo, Camilo E., Bataille, Carole J. R., Bery, Nicolas, Miller, Ami, Russell, Angela J., Phillips, Simon E. V., Carr, Stephen B., Rabbitts, Terence H.
Published in Proceedings of the National Academy of Sciences - PNAS (12.02.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (12.02.2019)
Get full text
Journal Article
KRAS-specific inhibition using a DARPin binding to a site in the allosteric lobe
Bery, Nicolas, Legg, Sandrine, Debreczeni, Judit, Breed, Jason, Embrey, Kevin, Stubbs, Christopher, Kolasinska-Zwierz, Paulina, Barrett, Nathalie, Marwood, Rose, Watson, Jo, Tart, Jon, Overman, Ross, Miller, Ami, Phillips, Christopher, Minter, Ralph, Rabbitts, Terence H
Published in Nature communications (13.06.2019)
Published in Nature communications (13.06.2019)
Get full text
Journal Article
Small molecule inhibitors of RAS-effector protein interactions derived using an intracellular antibody fragment
Quevedo, Camilo E, Cruz-Migoni, Abimael, Bery, Nicolas, Miller, Ami, Tanaka, Tomoyuki, Petch, Donna, Bataille, Carole J R, Lee, Lydia Y W, Fallon, Phillip S, Tulmin, Hanna, Ehebauer, Matthias T, Fernandez-Fuentes, Narcis, Russell, Angela J, Carr, Stephen B, Phillips, Simon E V, Rabbitts, Terence H
Published in Nature communications (09.08.2018)
Published in Nature communications (09.08.2018)
Get full text
Journal Article
BRET-based RAS biosensors that show a novel small molecule is an inhibitor of RAS-effector protein-protein interactions
Bery, Nicolas, Cruz-Migoni, Abimael, Bataille, Carole Jr, Quevedo, Camilo E, Tulmin, Hanna, Miller, Ami, Russell, Angela, Phillips, Simon Ev, Carr, Stephen B, Rabbitts, Terence H
Published in eLife (10.07.2018)
Published in eLife (10.07.2018)
Get full text
Journal Article
Distinct pathways regulated by menin and by MLL1 in hematopoietic stem cells and developing B cells
Li, Bin E., Gan, Tao, Meyerson, Matthew, Rabbitts, Terence H., Ernst, Patricia
Published in Blood (19.09.2013)
Published in Blood (19.09.2013)
Get full text
Journal Article
Exploring the surfaceome of Ewing sarcoma identifies a new and unique therapeutic target
Town, Jennifer, Pais, Helio, Harrison, Sally, Stead, Lucy F., Bataille, Carole, Bunjobpol, Wilawan, Zhang, Jing, Rabbitts, Terence H.
Published in Proceedings of the National Academy of Sciences - PNAS (29.03.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (29.03.2016)
Get full text
Journal Article
Surfaceome interrogation using an RNA-seq approach highlights leukemia initiating cell biomarkers in an LMO2 T cell transgenic model
Pais, Helio, Ruggero, Katia, Zhang, Jing, Al-Assar, Osama, Bery, Nicolas, Bhuller, Ravneet, Weston, Victoria, Kearns, Pamela R, Mecucci, Cristina, Miller, Ami, Rabbitts, Terence H
Published in Scientific reports (08.04.2019)
Published in Scientific reports (08.04.2019)
Get full text
Journal Article
Progressive 3q Amplification Consistently Targets SOX2 in Preinvasive Squamous Lung Cancer
MCCAUGHAN, Frank, POLE, Jessica C. M, BANKIER, Alan T, KONFORTOV, Bernard A, CARROLL, Bernadette, FALZON, Mary, RABBITTS, Terence H, GEORGE, P. Jeremy, DEAR, Paul H, RABBITTS, Pamela H
Published in American journal of respiratory and critical care medicine (01.07.2010)
Published in American journal of respiratory and critical care medicine (01.07.2010)
Get full text
Journal Article
The role of Slit-Robo signaling in the generation, migration and morphological differentiation of cortical interneurons
Andrews, William, Barber, Melissa, Hernadez-Miranda, Luis R., Xian, Jian, Rakic, Sonja, Sundaresan, Vasi, Rabbitts, Terence H., Pannell, Richard, Rabbitts, Pamela, Thompson, Hannah, Erskine, Lynda, Murakami, Fujio, Parnavelas, John G.
Published in Developmental biology (15.01.2008)
Published in Developmental biology (15.01.2008)
Get full text
Journal Article
Selection and Characterization of a Nanobody Biosensor of GTP-Bound RHO Activities
Keller, Laura, Bery, Nicolas, Tardy, Claudine, Ligat, Laetitia, Favre, Gilles, Rabbitts, Terence H, Olichon, Aurélien
Published in Antibodies (Basel) (09.01.2019)
Published in Antibodies (Basel) (09.01.2019)
Get full text
Journal Article
Salmonella-based platform for efficient delivery of functional binding proteins to the cytosol
Chabloz, Antoine, Schaefer, Jonas V, Kozieradzki, Ivona, Cronin, Shane J F, Strebinger, Daniel, Macaluso, Francesca, Wald, Jiri, Rabbitts, Terence H, Plückthun, Andreas, Marlovits, Thomas C, Penninger, Josef M
Published in Communications biology (03.07.2020)
Published in Communications biology (03.07.2020)
Get full text
Journal Article