Search Results - "RYDER, Hamish" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Characterization of Aclidinium Bromide, a Novel Inhaled Muscarinic Antagonist, with Long Duration of Action and a Favorable Pharmacological Profile

by Gavaldà, Amadeu, Miralpeix, Montserrat, Ramos, Israel, Otal, Raquel, Carreño, Cristina, Viñals, Marisa, Doménech, Teresa, Carcasona, Carla, Reyes, Blanca, Vilella, Dolors, Gras, Jordi, Cortijo, Julio, Morcillo, Esteban, Llenas, Jesús, Ryder, Hamish, Beleta, Jorge
Published in The Journal of pharmacology and experimental therapeutics (01.11.2009)

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Journal Article

Synthesis and Biological Activity of Pyrido[3′,2′:4,5]thieno[3,2-d]pyrimidines as Phosphodiesterase Type 4 Inhibitors

Synthesis and Biological Activity of Pyrido[3′,2′:4,5]thieno[3,2-d]pyrimidines as Phosphodiesterase Type 4 Inhibitors

by Taltavull, Joan, Serrat, Jordi, Gràcia, Jordi, Gavaldà, Amadeu, Andrés, Míriam, Córdoba, Mònica, Miralpeix, Montserrat, Vilella, Dolors, Beleta, Jorge, Ryder, Hamish, Pagès, Lluís
Published in Journal of medicinal chemistry (14.10.2010)

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Journal Article

Discovery of potent inhibitors of the lyso phospholipase autotaxin

Discovery of potent inhibitors of the lyso phospholipase autotaxin

by Shah, Pritom, Cheasty, Anne, Foxton, Caroline, Raynham, Tony, Farooq, Muddasar, Gutierrez, Irene Farre, Lejeune, Aurore, Pritchard, Michelle, Turnbull, Andrew, Pang, Leon, Owen, Paul, Boyd, Susan, Stowell, Alexandra, Jordan, Allan, Hamilton, Niall M., Hitchin, James R., Stockley, Martin, MacDonald, Ellen, Quesada, Mar Jimenez, Trivier, Elisabeth, Skeete, Jana, Ovaa, Huib, Moolenaar, Wouter H., Ryder, Hamish
Published in Bioorganic & medicinal chemistry letters (01.11.2016)

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Journal Article

Discovery of novel quaternary ammonium derivatives of (3 R)-quinuclidinyl carbamates as potent and long acting muscarinic antagonists

Discovery of novel quaternary ammonium derivatives of (3 R)-quinuclidinyl carbamates as potent and long acting muscarinic antagonists

by Prat, Maria, Buil, María Antonia, Fernández, Maria Dolors, Castro, Jordi, Monleón, Juan Manuel, Tort, Laia, Casals, Gaspar, Ferrer, Manuel, Huerta, Josep Maria, Espinosa, Sònia, López, Manuel, Segarra, Victor, Gavaldà, Amadeu, Miralpeix, Montserrat, Ramos, Israel, Vilella, Dolors, González, Marisa, Córdoba, Mònica, Cárdenas, Alvaro, Antón, Francisca, Beleta, Jorge, Ryder, Hamish
Published in Bioorganic & medicinal chemistry letters (01.06.2011)

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Journal Article

Synthesis and Biological Evaluation of 3,4-Diaryloxazolones: A New Class of Orally Active Cyclooxygenase-2 Inhibitors

Synthesis and Biological Evaluation of 3,4-Diaryloxazolones: A New Class of Orally Active Cyclooxygenase-2 Inhibitors

by Puig, Carles, Crespo, María I, Godessart, Núria, Feixas, Joan, Ibarzo, Javier, Jiménez, Juan-Miguel, Soca, Lídia, Cardelús, Ignasi, Heredia, Ascensión, Miralpeix, Montserrat, Puig, Jaume, Beleta, Jordi, Huerta, Josep M, López, Manel, Segarra, Victor, Ryder, Hamish, Palacios, José M
Published in Journal of medicinal chemistry (27.01.2000)

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Journal Article

Synthesis and Biological Evaluation of 2-Phenylpyran-4-ones: A New Class of Orally Active Cyclooxygenase-2 Inhibitors

Synthesis and Biological Evaluation of 2-Phenylpyran-4-ones: A New Class of Orally Active Cyclooxygenase-2 Inhibitors

by Caturla, Francisco, Jiménez, Juan-Miguel, Godessart, Núria, Amat, Mercè, Cárdenas, Alvaro, Soca, Lídia, Beleta, Jordi, Ryder, Hamish, Crespo, María I
Published in Journal of medicinal chemistry (15.07.2004)

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Journal Article

Design of a Biased Potent Small Molecule Inhibitor of the Bromodonnain and PHD Finger-Containing (BRPF) Proteins Suitable for Cellular and in Vivo Studies

Design of a Biased Potent Small Molecule Inhibitor of the Bromodonnain and PHD Finger-Containing (BRPF) Proteins Suitable for Cellular and in Vivo Studies

by Igoe, Niall, Bayle, Elliott D., Fedorov, Oleg, Tallant, Cynthia, Savitsky, Pavel, Rogers, Catherine, Owen, Dafydd R., Deb, Gauri, Somervaille, Tim C. P., Andrews, David M., Jones, Neil, Cheasty, Anne, Ryder, Hamish, Brennan, Paul E., Mueller, Susanne, Knapp, Stefan, Fish, Paul V.
Published in Journal of medicinal chemistry (26.01.2017)

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Journal Article

Design of a Biased Potent Small Molecule Inhibitor of the Bromodomain and PHD Finger-Containing (BRPF) Proteins Suitable for Cellular and in Vivo Studies

Design of a Biased Potent Small Molecule Inhibitor of the Bromodomain and PHD Finger-Containing (BRPF) Proteins Suitable for Cellular and in Vivo Studies

by Igoe, Niall, Bayle, Elliott D, Fedorov, Oleg, Tallant, Cynthia, Savitsky, Pavel, Rogers, Catherine, Owen, Dafydd R, Deb, Gauri, Somervaille, Tim C. P, Andrews, David M, Jones, Neil, Cheasty, Anne, Ryder, Hamish, Brennan, Paul E, Müller, Susanne, Knapp, Stefan, Fish, Paul V
Published in Journal of medicinal chemistry (26.01.2017)

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Journal Article

Discovery of potent inhibitors of the lysophospholipase autotaxin

Discovery of potent inhibitors of the lysophospholipase autotaxin

by Shah, Pritom, Cheasty, Anne, Foxton, Caroline, Raynham, Tony, Farooq, Muddasar, Gutierrez, Irene Farre, Lejeune, Aurore, Pritchard, Michelle, Turnbull, Andrew, Pang, Leon, Owen, Paul, Boyd, Susan, Stowell, Alexandra, Jordan, Allan, Hamilton, Niall M., Hitchin, James R., Stockley, Martin, MacDonald, Ellen, Quesada, Mar Jimenez, Trivier, Elisabeth, Skeete, Jana, Ovaa, Huib, Moolenaar, Wouter H., Ryder, Hamish
Published in Bioorganic & medicinal chemistry letters (15.11.2016)

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Journal Article

Pharmacological characterization of abediterol, a novel inhaled β(2)-adrenoceptor agonist with long duration of action and a favorable safety profile in preclinical models

by Aparici, Mònica, Gómez-Angelats, Mireia, Vilella, Dolors, Otal, Raquel, Carcasona, Carla, Viñals, Marisa, Ramos, Israel, Gavaldà, Amadeu, De Alba, Jorge, Gras, Jordi, Cortijo, Julio, Morcillo, Esteban, Puig, Carlos, Ryder, Hamish, Beleta, Jorge, Miralpeix, Montserrat
Published in The Journal of pharmacology and experimental therapeutics (01.08.2012)

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Journal Article

Discovery of Novel Quaternary Ammonium Derivatives of (3R)-Quinuclidinol Esters as Potent and Long-Acting Muscarinic Antagonists with Potential for Minimal Systemic Exposure after Inhaled Administration: Identification of (3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane Bromide (Aclidinium Bromide)

Discovery of Novel Quaternary Ammonium Derivatives of (3R)-Quinuclidinol Esters as Potent and Long-Acting Muscarinic Antagonists with Potential for Minimal Systemic Exposure after Inhaled Administration: Identification of (3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane Bromide (Aclidinium Bromide)

by Prat, María, Fernández, Dolors, Buil, M. Antonia, Crespo, María I, Casals, Gaspar, Ferrer, Manuel, Tort, Laia, Castro, Jordi, Monleón, Juan M, Gavaldà, Amadeu, Miralpeix, Montserrat, Ramos, Israel, Doménech, Teresa, Vilella, Dolors, Antón, Francisca, Huerta, Josep M, Espinosa, Sonia, López, Manuel, Sentellas, Sonia, González, Marisa, Albertí, Joan, Segarra, Victor, Cárdenas, Alvaro, Beleta, Jorge, Ryder, Hamish
Published in Journal of medicinal chemistry (27.08.2009)

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Journal Article

Synthesis and biological activity of pyrido[3′,2′:4,5]furo[3,2-d]pyrimidine derivatives as novel and potent phosphodiesterase type 4 inhibitors

Synthesis and biological activity of pyrido[3′,2′:4,5]furo[3,2-d]pyrimidine derivatives as novel and potent phosphodiesterase type 4 inhibitors

by Taltavull, Joan, Serrat, Jordi, Gràcia, Jordi, Gavaldà, Amadeu, Córdoba, Mònica, Calama, Elena, Montero, José Luis, Andrés, Míriam, Miralpeix, Montserrat, Vilella, Dolors, Hernández, Begoña, Beleta, Jorge, Ryder, Hamish, Pagès, Lluís
Published in European journal of medicinal chemistry (01.10.2011)

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Journal Article

Pharmacological Characterization of Abediterol, a Novel Inhaled β 2 -Adrenoceptor Agonist with Long Duration of Action and a Favorable Safety Profile in Preclinical Models

by Aparici, Mònica, Gómez-Angelats, Mireia, Vilella, Dolors, Otal, Raquel, Carcasona, Carla, Viñals, Marisa, Ramos, Israel, Gavaldà, Amadeu, De Alba, Jorge, Gras, Jordi, Cortijo, Julio, Morcillo, Esteban, Puig, Carlos, Ryder, Hamish, Beleta, Jorge, Miralpeix, Montserrat
Published in The Journal of pharmacology and experimental therapeutics (01.08.2012)

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Journal Article

Efficient three-step sequence for the deamination of α-aminoesters. Application to the synthesis of CysLT1 antagonists

Efficient three-step sequence for the deamination of α-aminoesters. Application to the synthesis of CysLT1 antagonists

by González, Alfredo, Pérez, Daniel, Puig, Carles, Ryder, Hamish, Sanahuja, Jordi, Solé, Laia, Bach, Jordi
Published in Tetrahedron letters (10.06.2009)

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Journal Article

Discovery and characterization of 4 '-(2-Furyl)-N-pyridin-3-yl-4,5 '-bipyrimidin-2 '-amine (LAS38096), a potent, selective, and efficacious A(2B) adenosine receptor antagonist

Discovery and characterization of 4 '-(2-Furyl)-N-pyridin-3-yl-4,5 '-bipyrimidin-2 '-amine (LAS38096), a potent, selective, and efficacious A(2B) adenosine receptor antagonist

by Vidal, Bernat, Nueda, Arsenio, Esteve, Cristina, Domenech, Teresa, Benito, Sonia, Reinoso, Raquel F., Pont, Merce, Calbet, Marta, Lopez, Rosa, Cadavid, Maria Isabel, Loza, Maria Isabel, Cardenas, Alvaro, Godessart, Nuria, Beleta, Jorge, Warrellow, Graham, Ryder, Hamish
Published in Journal of medicinal chemistry (31.05.2007)

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Journal Article

Discovery and Characterization of 4‘-(2-Furyl)-N-pyridin-3-yl-4,5‘-bipyrimidin-2‘-amine (LAS38096), a Potent, Selective, and Efficacious A2B Adenosine Receptor Antagonist

Discovery and Characterization of 4‘-(2-Furyl)-N-pyridin-3-yl-4,5‘-bipyrimidin-2‘-amine (LAS38096), a Potent, Selective, and Efficacious A2B Adenosine Receptor Antagonist

by Vidal, Bernat, Nueda, Arsenio, Esteve, Cristina, Domenech, Teresa, Benito, Sonia, Reinoso, Raquel F, Pont, Mercè, Calbet, Marta, López, Rosa, Cadavid, María Isabel, Loza, María Isabel, Cárdenas, Álvaro, Godessart, Núria, Beleta, Jorge, Warrellow, Graham, Ryder, Hamish
Published in Journal of medicinal chemistry (31.05.2007)

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Journal Article

Reversal of P-glycoprotein mediated multidrug resistance by novel anthranilamide derivatives

Reversal of P-glycoprotein mediated multidrug resistance by novel anthranilamide derivatives

by Roe, Michael, Folkes, Adrian, Ashworth, Philip, Brumwell, Julie, Chima, Lal, Hunjan, Sukhjit, Pretswell, Ian, Dangerfield, Wendy, Ryder, Hamish, Charlton, Peter
Published in Bioorganic & medicinal chemistry letters (22.02.1999)

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Journal Article

New pyrrolopyrimidin-6-yl benzenesulfonamides : Potent A2B adenosine receptor antagonists

New pyrrolopyrimidin-6-yl benzenesulfonamides : Potent A2B adenosine receptor antagonists

by ESTEVE, Cristina, NUEDA, Arsenio, DIAZ, José Luis, BELETA, Jorge, CARDENAS, Alvaro, LOZOYA, Estrella, CADAVID, Maria Isabel, LOZA, Maria Isabel, RYDER, Hamish, VIDAV, Bernat
Published in Bioorganic & medicinal chemistry letters (15.07.2006)

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Journal Article

COMBINATIONS COMPRISING ANTIMUSCARINIC AGENTS AND CORTICOSTEROIDS

COMBINATIONS COMPRISING ANTIMUSCARINIC AGENTS AND CORTICOSTEROIDS

by GRAS ESCARDO JORDI, ORVIZ DIAZ PIO, RYDER HAMISH, LLENAS CALVO JESUS
Year of Publication 15.03.2013

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Patent

Synthesis and structure-activity relationships of novel histamine H-1 antagonists: Indolylpiperidinyl benzoic acid derivatives

Synthesis and structure-activity relationships of novel histamine H-1 antagonists: Indolylpiperidinyl benzoic acid derivatives

by Fonquerna, S, Miralpeix, M, Pages, L, Puig, C, Cardus, A, Anton, F, Cardenas, A, Vilella, D, Aparici, M, Calaf, E, Prieto, J, Gras, J, Huerta, JM, Warrellow, G, Beleta, J, Ryder, H
Published in Journal of medicinal chemistry (02.12.2004)

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