Process Development for Scale-Up of a Novel 3,5-Substituted Thiazolidine-2,4-dione Compound as a Potent Inhibitor for Estrogen-Related Receptor 1
Li, Xun, Russell, Ronald K, Spink, Jan, Ballentine, Scott, Teleha, Christopher, Branum, Shawn, Wells, Kenneth, Beauchamp, Derek, Patch, Raymond, Huang, Hui, Player, Mark, Murray, William
Published in Organic process research & development (21.02.2014)
Published in Organic process research & development (21.02.2014)
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Lab-Scale Preparation of a Novel Cyclopenta[b]furan Chemokine Receptor Antagonist
Teleha, Christopher A, Branum, Shawn, Zhang, Yongzheng, Reuman, Michael E, Van Der Steen, Luc, Verbeek, Marc, Fawzy, Nagy, Leo, Gregory C, Winters, Michael P, Kang, Fu-An, Kolpak, Michael, Beauchamp, Derek A, Lanter, James C, Russell, Ronald K, Sui, Zhihua, Vanbaelen, Hilde
Published in Organic process research & development (19.12.2014)
Published in Organic process research & development (19.12.2014)
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Lab-Scale Preparation of a Novel Carbocyclic Chemokine Receptor Antagonist
Teleha, Christopher A, Branum, Shawn, Zhang, Yongzheng, Reuman, Michael E, Van Der Steen, Luc, Verbeek, Marc, Fawzy, Nagy, Leo, Gregory C, Kang, Fu-An, Cai, Chaozhong, Kolpak, Michael, Beauchamp, Derek A, Wall, Mark J, Russell, Ronald K, Sui, Zhihua, Vanbaelen, Hilde
Published in Organic process research & development (19.12.2014)
Published in Organic process research & development (19.12.2014)
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Synthesis of Mavatrep: A Potent Antagonist of Transient Receptor Potential Vanilloid‑1
Wells, Kenneth M, Mehrman, Steven J, Abdel-Magid, Ahmed F, Ferraro, Caterina, Scott, Lorraine, Zhong, Hua Marlon, Teleha, Christopher A, Ballentine, Scott, Li, Xun, Russell, Ronald K, Spink, Jan M, Diamond, Craig, Youells, Scott, Zhang, Yongzheng, Tsay, Fuh-Rong, Cesco-Cancia, Sergio, Manzo, Stephen M, Beauchamp, Derek A
Published in Organic process research & development (20.11.2015)
Published in Organic process research & development (20.11.2015)
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An Efficient Synthesis of 3‑Substituted N‑Glycoside Indoles Useful as Sodium-Dependent Glucose Transporter Inhibitors
Li, Xun, Wells, Kenneth M, Branum, Shawn, Damon, Sandra, Youells, Scott, Beauchamp, Derek A, Palmer, David, Stefanick, Stephen, Russell, Ronald K, Murray, William
Published in Organic process research & development (16.11.2012)
Published in Organic process research & development (16.11.2012)
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Crystallization of a Cephalosporin and an ERR-1: Assembly of an Inexpensive Crystallization Platform
Wells, Kenneth M, Beauchamp, Derek A, Fermier, Adam, Wu, Wenju, Mehrman, Steven, Youells, Scott, Hu, Zhiyong, Li, Xun, Macielag, Mark J, Bignan, Gilles, Xu, Guozhang, Zhao, Bao-Ping, Huang, Lian, Weber, James, Gaul, Micheal D, Russell, Ronald K
Published in Crystal growth & design (06.11.2013)
Published in Crystal growth & design (06.11.2013)
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An Efficient Synthetic Process for Scale-Up Production of 4,5-Diamino-2-(trifluoromethyl)benzonitrile and 5-Bromo-3-(trifluoromethyl)benzene-1,2-diamine
Li, Xun, Ng, Raymond A, Zhang, Yongzheng, Russell, Ronald K, Sui, Zhihua
Published in Organic process research & development (15.05.2009)
Published in Organic process research & development (15.05.2009)
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Scalable Synthesis of the VEGF-R2 Kinase Inhibitor JNJ-17029259 Using Ultrasound-Mediated Addition of MeLi−CeCl3 to a Nitrile
Reuman, Michael, Beish, Sandra, Davis, Jeremy, Batchelor, Mark J, Hutchings, Martin C, Moffat, David F. C, Connolly, Peter J, Russell, Ronald K
Published in Journal of organic chemistry (01.02.2008)
Published in Journal of organic chemistry (01.02.2008)
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Regio- and diastereoselective ring-opening of (S)-(−)-2-(trifluoromethyl)oxirane with chiral 2,5-disubstituted tetrahydroquinolines in hexafluoro-2-propanol
Li, Xun, Russell, Ronald K, Chen, Hongfeng, Zhang, Yongzheng, Ballentine, Scott, Spink, Jan, Branum, Shawn, Liu, Fuqiang, Chen, Yanping, Rammeloo, Thomas, Aelterman, Wim, Sorgi, Kirk L, Murray, William V
Published in Green chemistry : an international journal and green chemistry resource : GC (01.01.2010)
Published in Green chemistry : an international journal and green chemistry resource : GC (01.01.2010)
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Synthesis of a 5-((Aryloxy)methyl)-3-(4-(trifluoromethyl)phenyl)[1,2,4]thiadiazole Derivative: A Promising PPARα,δ Agonist
Reuman, Michael, Hu, Zhiyong, Kuo, Gee-Hong, Li, Xun, Russell, Ronald K, Shen, Lan, Youells, Scott, Zhang, Yongzheng
Published in Organic process research & development (01.11.2007)
Published in Organic process research & development (01.11.2007)
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Synthesis of Tetracyclic Heterocompounds as Selective Estrogen Receptor Modulators. Part 3. Development of an Acid-Catalyzed Racemization Process for (S)-2,8-(Dimethoxy)-5-{4-[2-(1-piperidinyl)ethoxy]phenyl}−11,12-dihydro-5H-6,13-dioxabenzo[3,4]cyclohepta[1,2-a]naphthalene
Li, Xun, Russell, Ronald K, Horváth, András, Jain, Nareshkumar, Depré, Dominique, Ormerod, Dominic, Aelterman, Wim, Sui, Zhihua
Published in Organic process research & development (16.01.2009)
Published in Organic process research & development (16.01.2009)
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Synthesis of Tetracyclic Heterocompounds as Selective Estrogen Receptor Modulators. Part 2. Process Improvement for Scale-Up Of 2,5,8-Substituted 11,12-Dihydro-5H-6,13-dioxabenzo[3,4]cyclohepta-[1,2-a]naphthalene Derivatives
Li, Xun, Reuman, Michael, Russell, Ronald K, Youells, Scott, Beish, Sandra, Hu, Zhiyong, Branum, Shawn, Jain, Nareshkumar, Sui, Zhihua
Published in Organic process research & development (01.07.2007)
Published in Organic process research & development (01.07.2007)
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Synthesis of Tetracyclic Heterocompounds as Selective Estrogen Receptor Modulators. Part 1. Process Development for Scale-up of 2,5,8-Substituted 5,11-Dihydrochromeno[4,3-c]chromene Derivatives
Li, Xun, Reuman, Michael, Russell, Ronald K, Adams, Richard, Ma, Robert, Branum, Shawn, Youells, Scott, Roberts, Jerry, Jain, Nareshkumar, Kanojia, Ramesh, Sui, Zhihua
Published in Organic process research & development (01.05.2007)
Published in Organic process research & development (01.05.2007)
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Substituted Salicylanilides as Inhibitors of Two-Component Regulatory Systems in Bacteria
Macielag, Mark J, Demers, James P, Fraga-Spano, Stephanie A, Hlasta, Dennis J, Johnson, Sigmond G, Kanojia, Ramesh M, Russell, Ronald K, Sui, Zhihua, Weidner-Wells, Michele A, Werblood, Harvey, Foleno, Barbara D, Goldschmidt, Raul M, Loeloff, Michael J, Webb, Glenda C, Barrett, John F
Published in Journal of medicinal chemistry (30.07.1998)
Published in Journal of medicinal chemistry (30.07.1998)
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β-Alkylthio indolyl carbinols: Potent nonsteroidal antiandrogens with oral efficacy in a prostate cancer model
Lanter, James C., Fiordeliso, James J., Alford, Vernon C., Zhang, Xuqing, Wells, Kenneth M., Russell, Ronald K., Allan, George F., Lai, Muh-Tsann, Linton, Olivia, Lundeen, Scott, Sui, Zhihua
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
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Synthesis of Tetracyclic Heterocompounds as Selective Estrogen Receptor Modulators. Part 2. Process Improvement for Scale-Up of 2,5,8-Substituted 11,12-Dihydro-5H-6,13-dioxabenzo[3,4]cyclohepta-[1,2-a]naphthalene Derivatives
Li, Xun, Reuman, Michael, Russell, Ronald K, Youells, Scott, Beish, Sandra, Hu, Zhiyong, Branum, Shawn, Jain, Nareshkumar, Sui, Zhihua
Published in Organic process research & development (18.01.2008)
Published in Organic process research & development (18.01.2008)
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