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Published in Science advances (01.10.2021)
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Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases
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Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
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Journal Article
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A2A Receptor Antagonists and Their Biological Evaluation
Basu, Sujay, Barawkar, Dinesh A, Thorat, Sachin, Shejul, Yogesh D, Patel, Meena, Naykodi, Minakshi, Jain, Vaibhav, Salve, Yogesh, Prasad, Vandna, Chaudhary, Sumit, Ghosh, Indraneel, Bhat, Ganesh, Quraishi, Azfar, Patil, Harish, Ansari, Shariq, Menon, Suraj, Unadkat, Vishal, Thakare, Rhishikesh, Seervi, Madhav S, Meru, Ashwinkumar V, De, Siddhartha, Bhamidipati, Ravi K, Rouduri, Sreekanth R, Palle, Venkata P, Chug, Anita, Mookhtiar, Kasim A
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
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Journal Article
Design and synthesis of novel xanthine derivatives as potent and selective A 2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Patel, Meena, Waman, Yogesh, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Naykodi, Minakshi, Goswami, Arnab, Reddy, B Srinivasa, Prasad, Vandna, Chaturvedi, Sandhya, Quraishi, Azfar, Menon, Suraj, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Ghosh, Indraneel, Mustafa, Syed, De, Siddhartha, Jain, Vaibhav, Banerjee, Ena Ray, Rouduri, Sreekanth R, Palle, Venkata P, Chugh, Anita, Mookhtiar, Kasim A
Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
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Journal Article
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A 2A Receptor Antagonists and Their Biological Evaluation
Basu, Sujay, Barawkar, Dinesh A, Thorat, Sachin, Shejul, Yogesh D, Patel, Meena, Naykodi, Minakshi, Jain, Vaibhav, Salve, Yogesh, Prasad, Vandna, Chaudhary, Sumit, Ghosh, Indraneel, Bhat, Ganesh, Quraishi, Azfar, Patil, Harish, Ansari, Shariq, Menon, Suraj, Unadkat, Vishal, Thakare, Rhishikesh, Seervi, Madhav S, Meru, Ashwinkumar V, De, Siddhartha, Bhamidipati, Ravi K, Rouduri, Sreekanth R, Palle, Venkata P, Chug, Anita, Mookhtiar, Kasim A
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
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Journal Article
Discovery of Potent and Selective A2A Antagonists with Efficacy in Animal Models of Parkinson’s Disease and Depression
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Naykodi, Minakshi, Shejul, Yogesh D, Patel, Meena, Thorat, Sachin, Panmand, Anil, Kashinath, K, Bonagiri, Rajesh, Prasad, Vandna, Bhat, Ganesh, Quraishi, Azfar, Chaudhary, Sumit, Magdum, Amol, Meru, Ashwinkumar V, Ghosh, Indraneel, Bhamidipati, Ravi K, Raje, Amol A, Madgula, Vamsi L. M, De, Siddhartha, Rouduri, Sreekanth R, Palle, Venkata P, Chugh, Anita, Hariharan, Narayanan, Mookhtiar, Kasim A
Published in ACS medicinal chemistry letters (10.08.2017)
Published in ACS medicinal chemistry letters (10.08.2017)
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Journal Article
Design and synthesis of novel xanthine derivatives as potent and selective A(2B) adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases
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Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
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Journal Article
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A(2A) Receptor Antagonists and Their Biological Evaluation
Basu, Sujay, Barawkar, Dinesh A., Thorat, Sachin, Shejul, Yogesh D., Patel, Meena, Naykodi, Minakshi, Jain, Vaibhav, Salve, Yogesh, Prasad, Vandna, Chaudhary, Sumit, Ghosh, Indraneel, Bhat, Ganesh, Quraishi, Azfar, Patil, Harish, Ansari, Shariq, Menon, Suraj, Unadkat, Vishal, Thakare, Rhishikesh, Seervi, Madhav S., Meru, Ashwinkumar V., De, Siddhartha, Bhamidipati, Ravi K., Rouduri, Sreekanth R., Palle, Venkata P., Chug, Anita, Mookhtiar, Kasim A.
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
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Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions
Shaikh, Nadim S., Iyer, Jitesh P., Munot, Yogesh S., Mukhopadhyay, Partha P., Raje, Amol A., Nagaraj, Ranganayaki, Jamdar, Vijay, Gavhane, Ravindra, Lohote, Mahendra, Sherkar, Prasad, Bala, Madhu, Petla, Rajkanth, Meru, Ashwinkumar, Umrani, Dhananjay, Rouduri, Sreekanth, Joshi, Sachin, Reddy, Satyanarayan, Kandikere, Vishwottam, Bhuniya, Debnath, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
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Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis
Thakkar, Mahesh, Bhuniya, Debnath, Kaduskar, Rahul, Mengawade, Tanaji, Naik, Keshav, Salunkhe, Videsh, Bhalerao, Amit, Kurhade, Santosh, Mavinahalli, Jagadeesh, Jain, Vaibhav, Petla, Rajkanth, Avaragolla, Satheesh, Ray, Swagatam, Rouduri, Sreekanth, Dhanave, Avinash, De, Siddhartha, Pathade, Vishal, Tambe, Ashwini, Raje, Amol A., Madgula, Vamsi, Joshi, Sachin, Nadeem, Ahmed, bala, Madhu, Umrani, Dhananjay, Hariharan, Narayanan, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
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Journal Article
Discovery and evaluation of 1 H -pyrrolo[2,3- b ]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis
Thakkar, Mahesh, Bhuniya, Debnath, Kaduskar, Rahul, Mengawade, Tanaji, Naik, Keshav, Salunkhe, Videsh, Bhalerao, Amit, Kurhade, Santosh, Mavinahalli, Jagadeesh, Jain, Vaibhav, Petla, Rajkanth, Avaragolla, Satheesh, Ray, Swagatam, Rouduri, Sreekanth, Dhanave, Avinash, De, Siddhartha, Pathade, Vishal, Tambe, Ashwini, Raje, Amol A., Madgula, Vamsi, Joshi, Sachin, Nadeem, Ahmed, bala, Madhu, Umrani, Dhananjay, Hariharan, Narayanan, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry letters (01.04.2017)
Published in Bioorganic & medicinal chemistry letters (01.04.2017)
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Journal Article
Discovery of Potent and Selective A(2A) Antagonists with Efficacy in Animal Models of Parkinson's Disease and Depression
Basu, Sujay, Barawkar, Dinesh A., Ramdas, Vidya, Naykodi, Minakshi, Shejul, Yogesh D., Patel, Meena, Thorat, Sachin, Panmand, Anil, Kashinath, K., Bonagiri, Rajesh, Prasad, Vandna, Bhat, Ganesh, Quraishi, Azfar, Chaudhary, Sumit, Magdum, Amol, Meru, Ashwinkumar V., Ghosh, Indraneel, Bhamidipati, Ravi K., Raje, Amol A., Madgula, Vamsi L. M., De, Siddhartha, Rouduri, Sreekanth R., Palle, Venkata P., Chugh, Anita, Hariharan, Narayanan, Mookhtiar, Kasim A.
Published in ACS medicinal chemistry letters (01.08.2017)
Published in ACS medicinal chemistry letters (01.08.2017)
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Journal Article
A 2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Waman, Yogesh, Patel, Meena, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Bonagiri, Rajesh, Jadhav, Dilip, Mukhopadhyay, Partha, Prasad, Vandna, Reddy, B Srinivasa, Goswami, Arnab, Chaturvedi, Sandhya, Menon, Suraj, Quraishi, Azfar, Ghosh, Indraneel, Dusange, Sushant, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Thakre, Rhishikesh, Bedse, Gaurav, Rouduri, Sreekanth, Gundu, Jayasagar, Palle, Venkata P, Chugh, Anita, Mookhtiar, Kasim A
Published in European journal of medicinal chemistry (15.02.2017)
Published in European journal of medicinal chemistry (15.02.2017)
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Journal Article
A2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives
Basu, Sujay, Barawkar, Dinesh A., Ramdas, Vidya, Waman, Yogesh, Patel, Meena, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Bonagiri, Rajesh, Jadhav, Dilip, Mukhopadhyay, Partha, Prasad, Vandna, Reddy, B. Srinivasa, Goswami, Arnab, Chaturvedi, Sandhya, Menon, Suraj, Quraishi, Azfar, Ghosh, Indraneel, Dusange, Sushant, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Thakre, Rhishikesh, Bedse, Gaurav, Rouduri, Sreekanth, Gundu, Jayasagar, Palle, Venkata P., Chugh, Anita, Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (15.02.2017)
Published in European journal of medicinal chemistry (15.02.2017)
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Journal Article