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Published in Peptides (New York, N.Y. : 1980) (01.10.2009)
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Novel pharmacological MC4R agonists can efficiently activate mutated MC4R from obese patient with impaired endogenous agonist response
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Anticancer Activity of BIM-46174, a New Inhibitor of the Heterotrimeric G alpha /G beta gamma Protein Complex
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Published in Cancer research (Chicago, Ill.) (15.09.2006)
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Identification of a novel series of benzimidazoles as potent and selective antagonists of the human melanocortin-4 receptor
Poitout, Lydie, Brault, Valérie, Sackur, Carole, Bernetière, Sonia, Camara, José, Plas, Pascale, Roubert, Pierre
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
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Anticancer activity of BIM-46174, a new inhibitor of the heterotrimeric Gα/Gβγ protein complex
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Published in Cancer research (Chicago, Ill.) (15.09.2006)
Published in Cancer research (Chicago, Ill.) (15.09.2006)
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Abstract 2795: Safety profile and therapeutic potential in breast cancer of STX140, an original tubulin binding agent
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Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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3-Thio-1,2,4-triazoles, novel somatostatin sst2/sst5 agonists
CONTOUR-GALCERA, Marie-Odile, SIDHU, Alban, PLAS, Pascale, ROUBERT, Pierre
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
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Identification of Potent Non-Peptide Somatostatin Antagonists with sst3 Selectivity
Poitout, Lydie, Roubert, Pierre, Contour-Galcéra, Marie-Odile, Moinet, Christophe, Lannoy, Jacques, Pommier, Jacques, Plas, Pascale, Bigg, Dennis, Thurieau, Christophe
Published in Journal of medicinal chemistry (30.08.2001)
Published in Journal of medicinal chemistry (30.08.2001)
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Novel melanocortin-4 receptor agonists that decrease food intake and body weight
Dong, Jesse Z, DeOliveira, Daniel B, Halem, Heather A, Taylor, John E, Roubert, Pierre, Plas, Pascale, Culler, Michael D, Zhang, Jundong
Published in Advances in experimental medicine and biology (2009)
Published in Advances in experimental medicine and biology (2009)
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Anticancer activity of BIM-46174, a new inhibitor of the heterotrimeric Galpha/Gbetagamma protein complex
Prévost, Grégoire P, Lonchampt, Marie O, Holbeck, Susan, Attoub, Samir, Zaharevitz, Daniel, Alley, Mike, Wright, John, Brezak, Marie C, Coulomb, Hélène, Savola, Ann, Huchet, Marion, Chaumeron, Sophie, Nguyen, Quang-Dé, Forgez, Patricia, Bruyneel, Erik, Bracke, Mark, Ferrandis, Eric, Roubert, Pierre, Demarquay, Danièle, Gespach, Christian, Kasprzyk, Philip G
Published in Cancer research (Chicago, Ill.) (15.09.2006)
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Published in Cancer research (Chicago, Ill.) (15.09.2006)
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Identification of Potent Non-Peptide Somatostatin Antagonists with sst 3 Selectivity
Poitout, Lydie, Roubert, Pierre, Contour-Galcéra, Marie-Odile, Moinet, Christophe, Lannoy, Jacques, Pommier, Jacques, Plas, Pascale, Bigg, Dennis, Thurieau, Christophe
Published in Journal of medicinal chemistry (01.08.2001)
Published in Journal of medicinal chemistry (01.08.2001)
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Synthesis of substituted imidazopyrazines as ligands for the human somatostatin receptor subtype 5
Contour-Galcéra, Marie-Odile, Poitout, Lydie, Moinet, Christophe, Morgan, Barry, Gordon, Tom, Roubert, Pierre, Thurieau, Christophe
Published in Bioorganic & medicinal chemistry letters (12.03.2001)
Published in Bioorganic & medicinal chemistry letters (12.03.2001)
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NOVEL BENZIMIDAZOLE AND IMIDAZOPYRIDINE DERIVATIVES AND USE THEREOF AS A MEDICAMENT
POITOUT LYDIE, SACKUR CAROLE, PLAS PASCALE, BRAULT VALERIE, ROUBERT PIERRE
Year of Publication 31.07.2013
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Year of Publication 31.07.2013
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Angiotensin II and phorbol-esters potently down-regulate endothelin (ET-1) binding sites in vascular smooth muscle cells
Roubert, Pierre, Gillard, Véronique, Plas, Pascale, Guillon, Jean-Michel, Chabrier, Pierre-Etienne, Braquet, Pierre
Published in Biochemical and biophysical research communications (31.10.1989)
Published in Biochemical and biophysical research communications (31.10.1989)
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NOVEL BENZIMIDAZOLE AND IMIDAZOPYRIDINE DERIVATIVES AND USE THEREOF AS A MEDICAMENT
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Year of Publication 13.12.2012
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Year of Publication 13.12.2012
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