Effect of Flexibility, Lipophilicity, and the Location of Polar Residues on the Passive Membrane Permeability of a Series of Cyclic Decapeptides
Wang, Shuzhe, König, Gerhard, Roth, Hans-Jörg, Fouché, Marianne, Rodde, Stephane, Riniker, Sereina
Published in Journal of medicinal chemistry (09.09.2021)
Published in Journal of medicinal chemistry (09.09.2021)
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Journal Article
Rationalization of the Membrane Permeability Differences in a Series of Analogue Cyclic Decapeptides
Witek, Jagna, Wang, Shuzhe, Schroeder, Benjamin, Lingwood, Robin, Dounas, Andreas, Roth, Hans-Jörg, Fouché, Marianne, Blatter, Markus, Lemke, Oliver, Keller, Bettina, Riniker, Sereina
Published in Journal of chemical information and modeling (28.01.2019)
Published in Journal of chemical information and modeling (28.01.2019)
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Journal Article
Lessons for Oral Bioavailability: How Conformationally Flexible Cyclic Peptides Enter and Cross Lipid Membranes
Linker, Stephanie M., Schellhaas, Christian, Kamenik, Anna S., Veldhuizen, Mac M., Waibl, Franz, Roth, Hans-Jörg, Fouché, Marianne, Rodde, Stephane, Riniker, Sereina
Published in Journal of medicinal chemistry (23.02.2023)
Published in Journal of medicinal chemistry (23.02.2023)
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Journal Article
Polar/apolar interfaces modulate the conformational behavior of cyclic peptides with impact on their passive membrane permeability
Linker, Stephanie M, Schellhaas, Christian, Ries, Benjamin, Roth, Hans-Jörg, Fouché, Marianne, Rodde, Stephane, Riniker, Sereina
Published in RSC advances (16.02.2022)
Published in RSC advances (16.02.2022)
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Journal Article
Design and Development of a Cyclic Decapeptide Scaffold with Suitable Properties for Bioavailability and Oral Exposure
Fouché, Marianne, Schäfer, Michael, Berghausen, Jörg, Desrayaud, Sandrine, Blatter, Markus, Piéchon, Philippe, Dix, Ina, Martin Garcia, Aimar, Roth, Hans-Jörg
Published in ChemMedChem (19.05.2016)
Published in ChemMedChem (19.05.2016)
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Journal Article
Back Cover: Design and Development of a Cyclic Decapeptide Scaffold with Suitable Properties for Bioavailability and Oral Exposure (ChemMedChem 10/2016)
Fouché, Marianne, Schäfer, Michael, Berghausen, Jörg, Desrayaud, Sandrine, Blatter, Markus, Piéchon, Philippe, Dix, Ina, Martin Garcia, Aimar, Roth, Hans-Jörg
Published in ChemMedChem (19.05.2016)
Published in ChemMedChem (19.05.2016)
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Journal Article
Complex molecules: do they add value?
Selzer, Paul, Roth, Hans-Jörg, Ertl, Peter, Schuffenhauer, Ansgar
Published in Current opinion in chemical biology (01.06.2005)
Published in Current opinion in chemical biology (01.06.2005)
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Journal Article
Automated Parallel Synthesis of N-Alkylated-?-Amino Methyl Esters in Gram Quantities
Sylvie Chamoin, Hans-Jörg Roth, Carsten Borek, Aline Jary, Hugues Maillot
Published in Chimia (01.05.2003)
Published in Chimia (01.05.2003)
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Journal Article
Quality Control in Combinatorial Chemistry: Determinations of Amounts and Comparison of the “Purity” of LC−MS-Purified Samples by NMR, LC−UV and CLND
Letot, Elodie, Koch, Guido, Falchetto, Rocco, Bovermann, Günter, Oberer, Lukas, Roth, Hans-Jörg
Published in Journal of combinatorial chemistry (01.05.2005)
Published in Journal of combinatorial chemistry (01.05.2005)
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Journal Article
COMPOUNDS AND COMPOSITIONS AS LXR MODULATORS
SAEZ ENRIQUE, CHAMOIN SYLVIE, ELLIS DAVID A, CHIANELLI DONATELLA, NABAKKA JULIET, MOLTENI VALENTINA, LI XIAOLIN, ROTH HANS-JORG
Year of Publication 05.03.2009
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Year of Publication 05.03.2009
Patent
COMPOUNDS AND COMPOSITIONS AS LXR MODULATORS
LI, XIAOLIN, ROTH, HANS-JORG, ELLIS, DAVID A, SAEZ, ENRIQUE, CHAMOIN, SYLVIE, CHIANELLI, DONATELLA, NABAKKA, JULIET, MOLTENI, VALENTINA
Year of Publication 30.07.2008
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Year of Publication 30.07.2008
Patent